中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [24]
西双版纳热带植物园 [1]
高能物理研究所 [1]
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OAI收割 [25]
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期刊论文 [25]
会议论文 [1]
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2025 [1]
2022 [1]
2021 [1]
2017 [2]
2016 [5]
2015 [1]
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学科主题
Chemistry [2]
Pharmacolo... [1]
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Applications of innovative synthetic strategies in anticancer drug discovery: The driving force of new chemical reactions
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 119, 页码: 36
作者:
Wang, Han
;
Ma, Xiaolong
;
Sun, Longkang
;
Bi, Tongyu
;
Yang, Weibo
  |  
收藏
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浏览/下载:33/0
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提交时间:2025/04/01
Synthetic methodologies
Medicinal chemistry
New chemical reactions
Anticancer drug discovery
Conserved protein targets for developing pan-coronavirus drugs based on sequence and 3D structure similarity analyses
期刊论文
OAI收割
COMPUTERS IN BIOLOGY AND MEDICINE, 2022, 卷号: 145, 页码: 105455
作者:
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收藏
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浏览/下载:32/0
  |  
提交时间:2024/03/21
Pharmaceutical informatics
Drug design
Target discovery
Medicinal chemistry
Broad-spectrum drugs
1,2-Difunctionalized bicyclo[1.1.1]pentanes: Long-sought-after mimetics for ortho/ meta-substituted arenes
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 28, 页码: 5
作者:
Zhao, Jin-Xin
;
Chang, Yu-Xuan
;
He, Chi
;
Burke, Benjamin J.
;
Collins, Michael R.
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2021/11/04
synthesis
medicinal chemistry
bioisosteres
Carbohydrate Synthesis For Medicinal Chemistry: Part 1. O-Glycosides
会议论文
OAI收割
作者:
Gu XY(顾相应)
;
Yin Q(尹强)
;
Liu X(刘筱)
;
Jiang RW(姜如炜)
;
Chen GH(陈国华)
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
In
O-Glycosides
Part 1
Carbohydrate Synthesis For Medicinal Chemistry
discoveryofpotent24difluorolinkerpolyadpribosepolymerase1inhibitorswithenhancedwatersolubilityandinvivoanticancerefficacy
期刊论文
OAI收割
actapharmacologicasinica, 2017, 卷号: 38, 期号: 11, 页码: 1521
作者:
Chen Wenhua
;
Song Shanshan
;
Ql Minghui
;
Huan Xiajuan
;
Wang Yingqing
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/07/01
PARP INHIBITORS
MEDICINAL CHEMISTRY
DRUG DISCOVERY
CANCER
THERAPY
DESIGN
FLUORINE
SUCCESS
PREDICT
METRICS
PARP-1 inhibitor
olaparib
breast cancer
BRCA-deficient tumors
Tailor-Made alpha-Amino Acids in the Pharmaceutical Industry: Synthetic Approaches to (1R,2S)-1-Amino-2-vinylcyclopropane-1-carboxylic Acid (Vinyl-ACCA)
期刊论文
OAI收割
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2016, 期号: 16, 页码: 2757-2774
作者:
Sato, Tatsunori
;
Izawa, Kunisuke
;
Luis Acena, Jose
;
Liu, Hong
;
Soloshonok, Vadim A.
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收藏
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浏览/下载:22/0
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提交时间:2019/01/08
Asymmetric synthesis
Amino acids
Medicinal chemistry
Drug design
Antiviral agents
First Total Synthesis of the Marine Natural Brominated Polyunsaturated Lipid Xestospongenyne as a Potent Pancreatic Lipase Inhibitory Agent
期刊论文
OAI收割
SYNLETT, 2016, 卷号: 27, 期号: 3, 页码: 391-394
作者:
Gong, Jing-Xu
;
Wang, He-Yao
;
Yao, Li-Gong
;
Li, Xu-Wen
;
Guo, Yue-Wei
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收藏
  |  
浏览/下载:48/0
  |  
提交时间:2019/01/08
lipids
xestospongenyne
total synthesis
medicinal chemistry
natural products
Counting on natural products for drug design
期刊论文
OAI收割
NATURE CHEMISTRY, 2016, 卷号: 8, 期号: 6, 页码: 531-541
Rodrigues, T
;
Reker, D
;
Schneider, P
;
Schneider, G
收藏
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浏览/下载:29/0
  |  
提交时间:2017/01/12
CATALYTIC ENANTIOSELECTIVE SYNTHESIS
INSPIRED COMPOUND COLLECTION
DIVERSITY-ORIENTED SYNTHESIS
RELEVANT CHEMICAL SPACE
TARGET PREDICTION
MACROMOLECULAR TARGETS
COMBINATORIAL LIBRARY
NETWORK PHARMACOLOGY
MEDICINAL CHEMISTRY
LIGAND DISCOVERY
Structure-Based Discovery of PDEs Inhibitors
期刊论文
OAI收割
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2016, 卷号: 16, 期号: 9, 页码: 917-933
作者:
Li, Li
;
Chen, Wuyan
;
Chen, Tiantian
;
Ren, Jing
;
Xu, Yechun
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
Crystal structure
Cyclic nucleotide signalling pathway
Family-selective inhibitor
Medicinal chemistry
Phosphodiesterases
Structure-based drug design
Small-Molecule Therapeutics for Ebola Virus (EBOV) Disease Treatment
期刊论文
OAI收割
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2016, 期号: 1, 页码: 8-16
作者:
Izawa, Kunisuke
;
Luis Acena, Jose
;
Wang, Jiang
;
Soloshonok, Vadim A.
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/01/08
Synthetic methods
Medicinal chemistry
Drug design
Antiviral agents