中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [4]
合肥物质科学研究院 [1]
采集方式
OAI收割 [5]
内容类型
期刊论文 [5]
发表日期
2022 [2]
2021 [1]
2020 [1]
2012 [1]
学科主题
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Cryo-EM structures of cancer-specific helical and kinase domain mutations of PI3K alpha
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 46, 页码: 11
作者:
Liu, Xiao
;
Zhou, Qingtong
;
Hart, Jonathan R.
;
Xu, Yingna
;
Yang, Su
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2023/10/17
phosphoinositide 3-kinase (PI3K)
mass spectrometry
mutants
Nanobodies and chemical cross-links advance the structural and functional analysis of PI3K alpha
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 38, 页码: 9
作者:
Hart, Jonathan R.
;
Liu, Xiao
;
Pan, Chen
;
Liang, Anyi
;
Ueno, Lynn
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2023/10/17
phosphoinositide 3-kinase (PI3K)
nanobody
conformational changes
chemical cross-linking
mass spectrometry
Cryo-EM structures of PI3K alpha reveal conformational changes during inhibition and activation
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 45, 页码: 9
作者:
Liu, Xiao
;
Yang, Su
;
Hart, Jonathan R.
;
Xu, Yingna
;
Zou, Xinyu
  |  
收藏
  |  
浏览/下载:69/0
  |  
提交时间:2022/01/04
phosphoinositide 3-kinase (PI3K)
activation
inhibition
activity-dependent conformational changes
Emerging roles of class I PI3K inhibitors in modulating tumor microenvironment and immunity
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:
Sun, Pu
;
Meng, Ling-hua
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2020/12/21
phosphoinositide 3-kinase (PI3K)
PI3K inhibitors
tumor microenvironment
immune cells
immunotherapy
The crossregulation between ERK and PI3K signaling pathways determines the tumoricidal efficacy of MEK inhibitor
期刊论文
OAI收割
JOURNAL OF MOLECULAR CELL BIOLOGY, 2012, 卷号: 4
-
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/10/26
KINASE KINASE-1/2 INHIBITOR
PHOSPHOINOSITIDE 3-KINASE-GAMMA
ADVANCED CANCERS
LUNG-CANCER
CELL LUNG
PHASE-II
RESISTANCE
ROBUSTNESS
ACTIVATION
MUTATIONS
systems biology
mathematical model
ERK pathway
PI3K pathway
MEK inhibitor
resistance
robustness
biochemical control analysis