中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共5条,第1-5条 帮助

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First ATG101-recruiting small molecule degrader for selective CDK9 degradation via autophagy-lysosome pathway 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 5, 页码: 2612-2624
作者:  
Zhong, Ye;  Xu, Jing;  Cao, Huiying;  Gao, Jie;  Ding, Shaoyue
  |  收藏  |  浏览/下载:25/0  |  提交时间:2025/07/25
Cross-Linking Profiling of Molecular Glue Degrader-Induced E3 Ligase Interactome to Expand Target Space 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 13
作者:  
Xu, Yali;  Zhao, Wensi;  Nie, Hui-Jun;  Wang, Jiamin;  Fu, Jingjing
  |  收藏  |  浏览/下载:37/0  |  提交时间:2025/05/27
Discovery of HyT-Based Degraders of CDK9-Cyclin T1 Complex 期刊论文  OAI收割
CHEMISTRY & BIODIVERSITY, 2023, 页码: 10
作者:  
Lin, Rongkun;  Yang, Jie;  Liu, Ting;  Wang, Mingyu;  Ke, Chongrong
  |  收藏  |  浏览/下载:61/0  |  提交时间:2023/10/17
Structure-based rational design enables efficient discovery of a new selective and potent AKT PROTAC degrader 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 238, 页码: 15
作者:  
Zhu, Cheng-Liang;  Luo, Xiaomin;  Tian, Tian;  Rao, Zijian;  Wang, Hanlin
  |  收藏  |  浏览/下载:76/0  |  提交时间:2022/08/16
Design, Synthesis, and Biological Evaluation of IRAK4-Targeting PROTACs 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 12, 期号: 1, 页码: 82-87
作者:  
Chen, Yun;  Ning, Yi;  Bai, Gang;  Tong, Linjiang;  Zhang, Tao
  |  收藏  |  浏览/下载:88/0  |  提交时间:2021/05/24