中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [14]
合肥物质科学研究院 [3]
广州生物医药与健康研... [1]
上海营养与健康研究所 [1]
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OAI收割 [19]
内容类型
期刊论文 [18]
学位论文 [1]
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2023 [3]
2022 [3]
2021 [4]
2020 [2]
2019 [2]
2018 [2]
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学科主题
Biochemist... [1]
Biophysics [1]
生物化学与分子生物学 [1]
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浏览/检索结果:
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Degradation of Cyclin-Dependent Kinase 9/Cyclin T1 by Optimized Microtubule-Associated Protein 1 Light Chain 3 Beta-Recruiting Coumarin Analogs
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 17
作者:
Zeng, Yanping
;
Xiao, Jian
;
Xu, Yuanxin
;
Wei, Fan
;
Tian, Lina
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/10/17
Predicting and overcoming resistance to CDK9 inhibitors for cancer therapy
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13
作者:
Hua, Chen
;
Shena, Lijuan
;
Zoua, Fengming
;
Wua, Yun
;
Wanga, Beilei
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/11/10
Acquired resistance mutations
CDK9 inhibitors
Transcription
Single nucleotide polymorphisms
BAY1251152
Discovery of HyT-Based Degraders of CDK9-Cyclin T1 Complex
期刊论文
OAI收割
CHEMISTRY & BIODIVERSITY, 2023, 页码: 10
作者:
Lin, Rongkun
;
Yang, Jie
;
Liu, Ting
;
Wang, Mingyu
;
Ke, Chongrong
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/10/17
CDK9
cyclin T1
degrader
hydrophobic tag
protein degradation
Inhibition of the dopamine transporter promotes lysosome biogenesis and ameliorates Alzheimer's disease-like symptoms in mice
期刊论文
OAI收割
ALZHEIMERS & DEMENTIA, 2022, 页码: 15
作者:
Yin, Limin
;
Zhou, Jianhui
;
Li, Tianyou
;
Wang, Xinghua
;
Xue, Wenlong
  |  
收藏
  |  
浏览/下载:76/0
  |  
提交时间:2022/11/11
Alzheimer's disease
CDK9
dopamine transporter
lysosome biogenesis
TFEB
Discovery of Small-Molecule Degraders of the CDK9-Cyclin T1 Complex for Targeting Transcriptional Addiction in Prostate Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 16, 页码: 11034-11057
作者:
Li, Jiacheng
;
Liu, Ting
;
Song, Yuanli
;
Wang, Mingyu
;
Liu, Liping
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/21
CDK9 inhibitors in cancer research
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2022
作者:
Huang, Zhi
;
Wang, Tianqi
;
Wang, Cheng
;
Fan, Yan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2022/12/23
Discovery of Potent and Selective CDK9 Degraders for Targeting Transcription Regulation in Triple-Negative Breast Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14822-14847
作者:
Wei, Dan
;
Wang, Hanlin
;
Zeng, Qinghe
;
Wang, Wenjing
;
Hao, Bingbing
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2021/12/16
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:
Han, Xu
;
Song, Ning
;
Saidahmatov, Abdusaid
;
Wang, Peipei
;
Wang, Yong
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2021/12/16
Efficient Synthesis and Docking Analysis of Selective CDK9 Inhibitor NVP-2
期刊论文
OAI收割
Pharmaceutical Fronts, 2021, 期号: 3, 页码: E50-E55
作者:
Saidahmatov, Abdusaid
;
Liang, Xue-Wu
;
Shi, Yuqiang
;
Han, Xu
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/14
NVP-2
CDK9 inhitor
efficient synthesis
docking analysis
Discovery of selective CDK9 degraders with enhancing antiproliferative activity through PROTAC conversion
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 11
作者:
Qiu, Xiaqiu
;
Li, Yuanqing
;
Yu, Bin
;
Ren, Jie
;
Huang, Huidan
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2021/05/24
CDK9
Antitumor
PROTAC
AML
Degrader