中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [5]
采集方式
OAI收割 [5]
内容类型
期刊论文 [5]
发表日期
2021 [1]
2012 [1]
2011 [1]
2009 [1]
2008 [1]
学科主题
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Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel Arylaminoacetylhydrazone Derivatives Containing Carbazole Moiety
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 8, 页码: 3157-3170
作者:
Li Yingjun
;
Lin Ledi
;
Jin Kun
;
Gao Lixin
;
Sheng Li
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2021/11/04
protein tyrosine phosphatase 1B (PTP1B) inhibitor
carbazole
arylaminoacetylhydrazone
synthesis
molecular docking
Natural products possessing protein tyrosine phosphatase 1B (PTP1B) inhibitory activity found in the last decades
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 10, 页码: 1217-1245
作者:
Jiang, Cheng-shi
;
Liang, Lin-fu
;
Guo, Yue-wei
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08
natural products
phytochemistry
protein tyrosine phosphatase 1B (PTP1B)
inhibitor
structure-activity relationship (SAR)
type 2 diabetes
obesity
Monosaccharide as a Central Scaffold Toward the Construction of Salicylate-Based Bidentate PTP1B Inhibitors via Click Chemistry
期刊论文
OAI收割
BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2011, 卷号: 32, 期号: 3, 页码: 1000-1006
作者:
Tang, Yan-Hui
;
Hu, Min
;
He, Xiao-Peng
;
Fahnbulleh, Sando
;
Li, Cui
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
Monosaccharide
Structural preference
Click chemistry
Protein tyrosine phosphatase 1B (PTP1B) inhibitor
asesquiterpenequinonedysidinefromthespongedysideavillosaactivatestheinsulinpathwaythroughinhibitionofptpases
期刊论文
OAI收割
actapharmacologicasinica, 2009, 卷号: 30, 期号: 3, 页码: 333
作者:
Yu ZHANG
;
Yan LI
;
Yuewei GUO
;
Hualiang JIANG
;
Xu SHEN
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
TYROSINE-PHOSPHATASE 1B
STIMULATES GLUCOSE-UPTAKE
PROTEIN-KINASE INHIBITOR
3T3-L1 ADIPOCYTES
SELECTIVE INHIBITORS
GLUT4 TRANSLOCATION
PHOSPHOLIPASE A(2)
PLASMA-MEMBRANE
LEPTIN ACTION
SENSITIVITY
sesquiterpene quinone
dysidine
PTP1B
inhibitor
insulin
discoveryofanovelcompetitiveinhibitorofptp1bbyhighthroughputscreening
期刊论文
OAI收割
actapharmacologicasinica, 2008, 卷号: 29, 期号: 2, 页码: 278
作者:
Lei SHI
;
Haiping YU
;
Yueyang ZHOU
;
Junqin DU
;
Qiang SHEN
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
PROTEIN-TYROSINE PHOSPHATASE-1B
FAO HEPATOMA-CELLS
INSULIN SENSITIVITY
ADIPOSE-TISSUE
OVEREXPRESSION
RESISTANCE
OBESITY
1B
PTP-1B
GENE
high throughput screening
PTP1B
insulin receptor
phosphoryaltion
competitive inhibitor