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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [153]
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OAI收割 [153]
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期刊论文 [152]
会议论文 [1]
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2022 [3]
2021 [5]
2020 [6]
2019 [4]
2018 [5]
2017 [7]
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Chemistry [4]
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共153条,第1-10条
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专题:上海药物研究所
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Discovery of YFJ-36: Design, Synthesis, and Antibacterial Activities of Catechol-Conjugated β-Lactams against Gram-Negative Bacteria
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:
Liu, Fangjun
;
Kou, Qunhuan
;
Li, Hongyuan
;
Cao, Yangzhi
;
Chen, Meng
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/22
Enantioselective Assembly of α, β-Diamine Acid Derivatives via Three-Component Reaction of α-H Diazoacetates with Sulfonamides and Imines
期刊论文
OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2023, 页码: 8
作者:
Sha, Hongkai
;
Xie, Xiongda
;
Zhang, Dan
;
Hu, Wenhao
;
Kang, Zhenghui
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/03/13
asymmetric three-component reaction
alpha, beta-diamine acid
metal carbenes
ammonium ylide
alpha-H diazoacetates
Simultaneous determination of almonertinib and its active metabolite HAS-719 in human plasma by LC-MS/MS: Evaluation of pharmacokinetic interactions
期刊论文
OAI收割
JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 2022, 卷号: 1197, 页码: 7
作者:
Liu, Lu
;
Yang, Le
;
Li, Wei
;
Chen, Xiaoyan
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/08/16
Almonertinib
LC -MS
MS
Active metabolite (HAS-719)
Pharmacokinetic drug-drug interaction
Quantification of the major circulating metabolite of BS1801, an ebselen analog, in human plasma
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2022, 卷号: 212, 页码: 10
作者:
Tian, Qianqian
;
Jiang, Jinfang
;
Yin, Hanwei
;
Ma, Jiao
;
Deng, Guozhen
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/06/15
BS1801
Ebselen
Circulating metabolite
Human plasma
LC-MS/MS
Berberine and its derivatives represent as the promising therapeutic agents for inflammatory disorders
期刊论文
OAI收割
PHARMACOLOGICAL REPORTS, 2022, 页码: 13
作者:
Lu, Qiukai
;
Fu, Yifan
;
Li, Heng
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/06/15
Allergy
Berberine
Inflammation
Ulcerative colitis
A camptothecin-based, albumin-binding prodrug enhances efficacy and safety in vivo
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 226, 页码: 11
作者:
Cheng, Zhiyang
;
Huang, Ying
;
Shen, Qianqian
;
Zhao, Yangrong
;
Wang, Lei
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2021/11/04
Cancer
beta-glucuronidase
Bioconjugation
Albumin
Camptothecin
A validated HPLC-MS/MS method for determination of simmitecan and its metabolite chimmitecan in human plasma and its application to a pharmacokinetic study in Chinese patients with advanced solid tumor
期刊论文
OAI收割
JOURNAL OF SEPARATION SCIENCE, 2021, 页码: 8
作者:
Zhou, Jun
;
Zhan, Yan
;
Zhong, Dafang
;
Chen, Xiaoyan
;
Zhang, Yifan
  |  
收藏
  |  
浏览/下载:81/0
  |  
提交时间:2021/11/04
chimmitecan
mass spectrometry
pharmacokinetics
simmitecan
solid tumors
Interfacial interactions and structures of protic ionic liquids on a graphite surface: A first-principles study and comparison with aprotic ionic liquids
期刊论文
OAI收割
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2021, 页码: 11
作者:
Lu, Yunxiang
;
Xu, Yanmin
;
Lu, Ling
;
Xu, Zhijian
;
Liu, Honglai
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2021/11/04
Quantification of Usaramine and its N-Oxide Metabolite in Rat Plasma Using Liquid Chromatography-Tandem Mass Spectrometry
期刊论文
OAI收割
JOURNAL OF ANALYTICAL TOXICOLOGY, 2021, 卷号: 46, 期号: 5, 页码: 512-518
作者:
Lin, Feifei
;
Ma, Yan
;
Pan, Anni
;
Ye, Yang
;
Liu, Jia
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2022/08/16
Characterization and quantitative determination of henagliflozin metabolites in humans
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2021, 卷号: 192, 页码: 8
作者:
Chen, Zhendong
;
Li, Liang
;
Zhan, Yan
;
Zhang, Yifan
;
Liu, Haiyan
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2021/05/24
Henagliflozin
Metabolism
LC-MS/MS