中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [16]
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内容类型
发表日期
  • 2020 [16]
学科主题
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Large-scale Generation of Functional and Transplantable Hepatocytes and Cholangiocytes from Human Endoderm Stem Cells 期刊论文  OAI收割
CELL REPORTS, 2020, 卷号: 33, 期号: 10, 页码: 24
作者:  
Feng, Sisi;  Wu, Jiaying;  Qiu, Wei-Lin;  Yang, Li;  Deng, Xiaogang
  |  收藏  |  浏览/下载:75/0  |  提交时间:2021/05/24
Synthesis of Axially Chiral Olefin-Oxazoline Ligands via Pd-Catalyzed Multiple C-H Functionalization 期刊论文  OAI收割
ORGANIC LETTERS, 2020, 卷号: 22, 期号: 23, 页码: 9169-9173
作者:  
Li, Ling-Jun;  Chen, Jun-Jie;  Feng, Chen-Fei;  Li, Han-Yuan;  Wang, Xing
  |  收藏  |  浏览/下载:15/0  |  提交时间:2021/05/24
Chemical constituents from the South China sea soft coral Sinularia humilis 期刊论文  OAI收割
NATURAL PRODUCT RESEARCH, 2020, 页码: 7
作者:  
Li, Jie;  Huan, Xia-Juan;  Wu, Meng-Jun;  Chen, Zi-Hui;  Chen, Bao
  |  收藏  |  浏览/下载:16/0  |  提交时间:2021/05/24
Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (ROR gamma t) modulators: insights into different protein behaviors with "short" and "long" inverse agonists 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:  
Yu, Ming-cheng;  Yang, Feng;  Ding, Xiao-yu;  Sun, Nan-nan;  Jiang, Zheng-yuan
  |  收藏  |  浏览/下载:95/0  |  提交时间:2020/12/24
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:  
Lv, Kaikai;  Chen, Weicong;  Chen, Danqi;  Mou, Jie;  Zhang, Huijie
  |  收藏  |  浏览/下载:22/0  |  提交时间:2020/12/21
Design, synthesis and biological evaluation of potent EGFR kinase inhibitors against 19D/T790M/C797S mutation 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 16, 页码: 6
作者:  
Su, Zhicheng;  Yang, Tingyuan;  Wang, Jie;  Lai, Mengzhen;  Tong, Linjiang
  |  收藏  |  浏览/下载:62/0  |  提交时间:2020/12/24
EGFR  NSCLC  C797S  
Discovery of novel USP8 inhibitors via Ubiquitin-Rho-110 fluorometric assay based high throughput screening 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 9
作者:  
Han, Jie;  Tian, Yucheng;  Yu, Liang;  Zhang, Qilin;  Xu, Xi
  |  收藏  |  浏览/下载:39/0  |  提交时间:2020/12/24
Targeting FTO Suppresses Cancer Stem Cell Maintenance and Immune Evasion 期刊论文  OAI收割
CANCER CELL, 2020, 卷号: 38, 期号: 1, 页码: 79-+
作者:  
Su, Rui;  Dong, Lei;  Li, Yangchan;  Gao, Min;  Han, Li
  |  收藏  |  浏览/下载:40/0  |  提交时间:2020/12/24
Heterogeneous immunogenomic features and distinct escape mechanisms in multifocal hepatocellular carcinoma 期刊论文  OAI收割
JOURNAL OF HEPATOLOGY, 2020, 卷号: 72, 期号: 5, 页码: 896-908
作者:  
Dong, Liang-qing;  Peng, Li-hua;  Ma, Li-jie;  Liu, Dong-bing;  Zhang, Shu
  |  收藏  |  浏览/下载:81/0  |  提交时间:2020/07/01
TREK Channel Family Activator with a Well-Defined Structure-Activation Relationship for Pain and Neurogenic Inflammation 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 7, 页码: 3665-3677
作者:  
Qiu, Yunguang;  Huang, Lu;  Fu, Jie;  Han, Chenxia;  Fang, Jing
  |  收藏  |  浏览/下载:36/0  |  提交时间:2020/07/01