中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [16]
采集方式
OAI收割 [16]
内容类型
期刊论文 [16]
发表日期
2020 [16]
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发表日期:2020
专题:上海药物研究所
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Large-scale Generation of Functional and Transplantable Hepatocytes and Cholangiocytes from Human Endoderm Stem Cells
期刊论文
OAI收割
CELL REPORTS, 2020, 卷号: 33, 期号: 10, 页码: 24
作者:
Feng, Sisi
;
Wu, Jiaying
;
Qiu, Wei-Lin
;
Yang, Li
;
Deng, Xiaogang
  |  
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2021/05/24
Synthesis of Axially Chiral Olefin-Oxazoline Ligands via Pd-Catalyzed Multiple C-H Functionalization
期刊论文
OAI收割
ORGANIC LETTERS, 2020, 卷号: 22, 期号: 23, 页码: 9169-9173
作者:
Li, Ling-Jun
;
Chen, Jun-Jie
;
Feng, Chen-Fei
;
Li, Han-Yuan
;
Wang, Xing
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2021/05/24
Chemical constituents from the South China sea soft coral Sinularia humilis
期刊论文
OAI收割
NATURAL PRODUCT RESEARCH, 2020, 页码: 7
作者:
Li, Jie
;
Huan, Xia-Juan
;
Wu, Meng-Jun
;
Chen, Zi-Hui
;
Chen, Bao
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2021/05/24
Soft coral
Sinularia humilis
diterpenoids
capnosane
Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (ROR gamma t) modulators: insights into different protein behaviors with "short" and "long" inverse agonists
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Yu, Ming-cheng
;
Yang, Feng
;
Ding, Xiao-yu
;
Sun, Nan-nan
;
Jiang, Zheng-yuan
  |  
收藏
  |  
浏览/下载:95/0
  |  
提交时间:2020/12/24
RORγ
t
cocrystal structures
MD simulation
“
short”
inverse agonists
agonists
“
long”
inverse agonists
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:
Lv, Kaikai
;
Chen, Weicong
;
Chen, Danqi
;
Mou, Jie
;
Zhang, Huijie
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/12/21
Design, synthesis and biological evaluation of potent EGFR kinase inhibitors against 19D/T790M/C797S mutation
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 16, 页码: 6
作者:
Su, Zhicheng
;
Yang, Tingyuan
;
Wang, Jie
;
Lai, Mengzhen
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2020/12/24
EGFR
NSCLC
C797S
Discovery of novel USP8 inhibitors via Ubiquitin-Rho-110 fluorometric assay based high throughput screening
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 9
作者:
Han, Jie
;
Tian, Yucheng
;
Yu, Liang
;
Zhang, Qilin
;
Xu, Xi
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2020/12/24
Ubiquitination
High throughput screening
Drug discovery
USP8
Targeting FTO Suppresses Cancer Stem Cell Maintenance and Immune Evasion
期刊论文
OAI收割
CANCER CELL, 2020, 卷号: 38, 期号: 1, 页码: 79-+
作者:
Su, Rui
;
Dong, Lei
;
Li, Yangchan
;
Gao, Min
;
Han, Li
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2020/12/24
Heterogeneous immunogenomic features and distinct escape mechanisms in multifocal hepatocellular carcinoma
期刊论文
OAI收割
JOURNAL OF HEPATOLOGY, 2020, 卷号: 72, 期号: 5, 页码: 896-908
作者:
Dong, Liang-qing
;
Peng, Li-hua
;
Ma, Li-jie
;
Liu, Dong-bing
;
Zhang, Shu
  |  
收藏
  |  
浏览/下载:81/0
  |  
提交时间:2020/07/01
Hepatocellular carcinoma
Tumor heterogeneity
Tumor microenvironment
Immunoediting
Neoantigen
TREK Channel Family Activator with a Well-Defined Structure-Activation Relationship for Pain and Neurogenic Inflammation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 7, 页码: 3665-3677
作者:
Qiu, Yunguang
;
Huang, Lu
;
Fu, Jie
;
Han, Chenxia
;
Fang, Jing
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2020/07/01