中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [48]
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期刊论文 [180]
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HIF-1 alpha inhibition in macrophages preserves acute liver failure by reducing IL-1 beta production
期刊论文
OAI收割
FASEB JOURNAL, 2023, 卷号: 37, 期号: 9, 页码: 12
作者:
Kong, Xiangrong
;
Liu, Wei
;
Zhang, Xinwen
;
Zhou, Chendong
;
Sun, Xinyu
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
acute liver failure
cell death
HIF-1 alpha inhibitor
interleukin-1 beta
macrophage
Discovery of novel triazine derivatives as potent retinoic acid receptor-related orphan receptor gamma t (ROR gamma t) inverse agonists
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 256, 页码: 18
作者:
Lu, Lixue
;
Chen, Song
;
Yu, Mingcheng
;
Zhou, Ronghui
;
Guo, Siqi
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/10/17
ROR gamma t
Triazines
Inverse agonist
Psoriasis
Autoimmune diseases
Design, synthesis and pharmacological evaluation of 2,3-dihydrobenzo-furan IRAK4 inhibitors for the treatment of diffuse large B-cell lymphoma
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 256, 页码: 16
作者:
Chen, Yun
;
Ning, Yi
;
Chen, Zhiwei
;
Xue, Yaping
;
Wu, Qingyun
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Apoptosis
Diffuse large B-Cell lymphoma
Interleukin-1 receptor associated kinase 4
Structure-based drug design
2
3-Dihydrobenzofuran
A novel anti-PD-L1/IL-15 immunocytokine overcomes resistance to PD-L1 blockade and elicits potent antitumor immunity
期刊论文
OAI收割
MOLECULAR THERAPY, 2023, 卷号: 31, 期号: 1, 页码: 66-77
作者:
Shi, Wenqiang
;
Lv, Liangyin
;
Liu, Nan
;
Wang, Hui
;
Wang, Yang
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/04/10
Targeting CSF-1R represents an effective strategy in modulating inflammatory diseases
期刊论文
OAI收割
PHARMACOLOGICAL RESEARCH, 2023, 卷号: 187, 页码: 17
作者:
Xiang, Caigui
;
Li, Heng
;
Tang, Wei
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
CSF-1R
CSF-1
IL-34
Inflammatory diseases
Myeloid cells
ASK120067 potently suppresses B-cell or T-cell malignancies in vitro and in vivo by inhibiting BTK and ITK
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 9
作者:
Song, Peiran
;
Bai, Gang
;
Chan, Shingpan
;
Zhang, Tao
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2023/04/10
Bruton's tyrosine kinase
interleukin-2-inducible T cell kinase
ASK120067
B-cell lymphoma
T-cell leukemia
E3 ubiquitin ligase NEDD4L negatively regulates inflammation by promoting ubiquitination of MEKK2
期刊论文
OAI收割
EMBO REPORTS, 2022
作者:
Li, Hui
;
Wang, Ning
;
Jiang, Yu
;
Wang, Haofei
;
Xin, Zengfeng
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2022/12/22
IL-17R signaling
inflammation
MEKK2
NEDD4L
ubiquitination
Artemisinin analog SM934 alleviates epithelial barrier dysfunction via inhibiting apoptosis and caspase-1-mediated pyroptosis in experimental colitis
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 18
作者:
Shao, Meijuan
;
Yan, Yuxi
;
Zhu, Fenghua
;
Yang, Xiaoqian
;
Qi, Qing
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/11/11
SM934
colitis
intestinal epithelial barrier
apoptosis
pyroptosis
NLRP3/caspase-1/GSDMD
MAPK/NF-kB
Synthesis of AC1903 analogs as potent transient receptor potential canonical channel 4/5 inhibitors and biological evaluation
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 68, 页码: 11
作者:
Chen, Lili
;
Zhang, Zhuang
;
Tian, Hongtao
;
Jiang, Shan
;
Ji, Yunyun
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/11/11
TRPC5
AC1903
Podocyte
FSGS
Keratinocyte
Proliferation
Inflammation
Anti-inflammatory activity of Anchusa italica Retz. in LPS-stimulated RAW264.7 cells mediated by the Nrf2/HO-1, MAPK and NF-κB signaling pathways
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2022, 卷号: 286, 期号: 3, 页码: 1-9
作者:
Duan, XM (Duan, Xiaomei) [1] , [2]
;
Li, J (Li, Jun) [1] , [2]
;
Cui, JX (Cui, Jingxue) [1] , [2]
;
Dong, YW (Dong, Yuwei) [1] , [2]
;
Xin, XL (Xin, Xuelei) [1] , [2]
  |  
收藏
  |  
浏览/下载:158/0
  |  
提交时间:2022/05/17
Boraginaceae
Anchusa italica Retz.
Anti-inflammatory