中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共300条,第1-10条 帮助

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Structure-Activity Relationships of 2-(Arylthio)benzoic Acid FTO Inhibitors 期刊论文  OAI收割
ISRAEL JOURNAL OF CHEMISTRY, 2024, 页码: 13
作者:  
Yan, Chao;  Zhang, Qian;  Xiao, Pan;  Xie, Xinyun;  Li, Ming
  |  收藏  |  浏览/下载:28/0  |  提交时间:2024/03/25
Immunotherapy Innovations in the Fight against Osteosarcoma: Emerging Strategies and Promising Progress 期刊论文  OAI收割
PHARMACEUTICS, 2024, 卷号: 16, 期号: 2, 页码: 21
作者:  
Cheng, Shigao;  Wang, Huiyuan;  Kang, Xuejia;  Zhang, Hui
  |  收藏  |  浏览/下载:11/0  |  提交时间:2024/04/09
Targeting ST8SIA6-AS1 counteracts KRASG12C inhibitor resistance through abolishing the reciprocal activation of PLK1/c-Myc signaling 期刊论文  OAI收割
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2023, 卷号: 12, 期号: 1, 页码: 22
作者:  
Wang, Yafang;  Yao, Mingyue;  Li, Cheng;  Yang, Kexin;  Qin, Xiaolong
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/01/26
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:  
Zhang, Jingyu;  Duan, Haiting;  Gui, Renzhao;  Wu, Mingfei;  Shen, Liteng
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/19
Discovery of 5-trifluoromethyl-2-aminopyrimidine derivatives as potent dual inhibitors of FLT3 and CHK1 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:  
Deng, Minjie;  Gao, Yue;  Wang, Peipei;  Du, Wenjing;  Xu, Gaoya
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/02/19
Preclinical and early clinical studies of a novel compound SYHA1813 that efficiently crosses the blood-brain barrier and exhibits potent activity against glioblastoma 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4748-4764
作者:  
Liu, Yingqiang;  Zhan, Zhengsheng;  Kang, Zhuang;  Li, Mengyuan;  Lv, Yongcong
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/01/26
Design, synthesis and biological evaluation of 2-aminopyrimidine derivatives as potent FLT3 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 96, 页码: 5
作者:  
Lian, Xuanmin;  Gao, Yue;  Li, Xuemei;  Wang, Peipei;  Tong, Lexian
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/12/11
Discovery, Structure-Activity Relationship and In Vitro Anticancer Activity of Small-Molecule Inhibitors of the Protein-Protein Interactions between AF9/ENL and AF4 or DOT1L 期刊论文  OAI收割
CANCERS, 2023, 卷号: 15, 期号: 21, 页码: 28
作者:  
Li, Xin;  Wu, Xiaowei;  Nie, Shenyou;  Zhao, Jidong;  Yao, Yuan
  |  收藏  |  浏览/下载:7/0  |  提交时间:2023/12/19
Chemical Inhibitors Targeting the Oncogenic m6A Modifying Proteins 期刊论文  OAI收割
ACCOUNTS OF CHEMICAL RESEARCH, 2023, 卷号: 56, 期号: 21, 页码: 3010-3022
作者:  
Huang, Yue;  Xia, Wenyang;  Dong, Ze;  Yang, Cai-Guang
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/12/11
Development of PI3Kγ selective inhibitors: the strategies and application 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 10
作者:  
Gu, Dong-Yan;  Zhang, Meng-Meng;  Li, Jia;  Zhou, Yu-Bo;  Sheng, Rong
  |  收藏  |  浏览/下载:4/0  |  提交时间:2023/12/08