中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [21]
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Chemical Inhibitors Targeting the Oncogenic m6A Modifying Proteins 期刊论文  OAI收割
ACCOUNTS OF CHEMICAL RESEARCH, 2023, 卷号: 56, 期号: 21, 页码: 3010-3022
作者:  
Huang, Yue;  Xia, Wenyang;  Dong, Ze;  Yang, Cai-Guang
  |  收藏  |  浏览/下载:7/0  |  提交时间:2023/12/11
High-Throughput-Methyl-Reading (HTMR) assay: a solution based on nucleotide methyl-binding proteins enables large-scale screening for DNA/RNA methyltransferases and demethylases 期刊论文  OAI收割
NUCLEIC ACIDS RESEARCH, 2022, 卷号: 50, 期号: 2, 页码: 14
作者:  
Xiao, Senhao;  Guo, Siqi;  Han, Jie;  Sun, Yanli;  Wang, Mingchen
  |  收藏  |  浏览/下载:29/0  |  提交时间:2022/06/15
Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (ROR gamma t) modulators: insights into different protein behaviors with "short" and "long" inverse agonists 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:  
Yu, Ming-cheng;  Yang, Feng;  Ding, Xiao-yu;  Sun, Nan-nan;  Jiang, Zheng-yuan
  |  收藏  |  浏览/下载:93/0  |  提交时间:2020/12/24
Antibody-free enzyme-assisted chemical approach for detection of N-6-methyladenosine 期刊论文  OAI收割
NATURE CHEMICAL BIOLOGY, 2020, 页码: 12
作者:  
Wang, Ye;  Xiao, Yu;  Dong, Shunqing;  Yu, Qiong;  Jia, Guifang
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
Discovery of alkyl bis(oxy)dibenzimidamide derivatives as novel protein arginine methyltransferase 1 (PRMT1) inhibitors 期刊论文  OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2017, 卷号: 90, 期号: 6, 页码: 1260-1270
作者:  
Zhang, Wei-yao;  Lu, Wen-chao;  Jiang, Hao;  Lv, Zheng-bing;  Xie, Yi-qian
  |  收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
Structural Characterization of Mannoglucan from Dendrobium nobile Lindl and the Neuritogenesis-Induced Effect of Its Acetylated Derivative on PC-12 Cells 期刊论文  OAI收割
POLYMERS, 2017, 卷号: 9, 期号: 9
作者:  
Jin, Can;  Du, Zhenyun;  Lin, Liyan;  Zhou, Lishuang;  Li, Saijuan
  |  收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
m(6)A RNA Methylation Regulates the Self-Renewal and Tumorigenesis of Glioblastoma Stem Cells 期刊论文  OAI收割
CELL REPORTS, 2017, 卷号: 18, 期号: 11, 页码: 2622-2634
作者:  
Cui, Qi;  Shi, Hailing;  Ye, Peng;  Li, Li;  Qu, Qiuhao
  |  收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08
Fluorescein Derivatives as Bifunctional Molecules for the Simultaneous Inhibiting and Labeling of FTO Protein 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2015, 卷号: 137, 期号: 43, 页码: 13736-13739
作者:  
Wang, Tianlu;  Hong, Tingting;  Huang, Yue;  Su, Haomiao;  Wu, Fan
  |  收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
Design, Synthesis, and Biological Evaluation of Novel Nonsteroidal FarnesoidX Receptor (FXR) Antagonists: Molecular Basis of FXR Antagonism 期刊论文  OAI收割
CHEMMEDCHEM, 2015, 卷号: 10, 期号: 7, 页码: 1184-1199
作者:  
Huang, Huang;  Si, Pei;  Wang, Lei;  Xu, Yong;  Xu, Xin
  |  收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08
Development of beta-amino-carbonyl compounds as androgen receptor antagonists 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 5, 页码: 664-673
作者:  
Zhang, Zhi-yun;  Zhu, Yan-hui;  Zhou, Cai-hong;  Liu, Qing;  Lu, Hui-li
  |  收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08