中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [19]
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Design, synthesis of novel benzimidazole derivatives as ENL inhibitors suppressing leukemia cells viability via downregulating the expression of MYC 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 248, 页码: 14
作者:  
Guo, Siqi;  Jia, Tongguan
  |  收藏  |  浏览/下载:20/0  |  提交时间:2023/04/10
Synthesis and pharmacological validation of fluorescent diarylsulfonylurea analogues as NLRP3 inhibitors and imaging probes 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 237, 页码: 13
作者:  
Zhao, Jiannan;  Li, Yongling;  Ma, Jing;  Liu, Jingting;  Xiao, Ruoxuan
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/08/16
Structure-Based of a Series of NSD2-PWWP1 Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 13, 页码: 9459-9477
作者:  
Li, Na;  Yang, Hong;  Liu, Ke;  Zhou, Liwei;  Huang, Yuting
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/03/21
Structural insights into hormone recognition by the human glucose-dependent insulinotropic polypeptide receptor 期刊论文  OAI收割
ELIFE, 2021, 卷号: 10, 页码: 20
作者:  
Zhao, Fenghui;  Zhang, Chao;  Zhou, Qingtong;  Hang, Kaini;  Zou, Xinyu
  |  收藏  |  浏览/下载:32/0  |  提交时间:2021/08/17
Structural insights into the lipid and ligand regulation of serotonin receptors 期刊论文  OAI收割
NATURE, 2021, 页码: 25
作者:  
Xu, Peiyu;  Huang, Sijie;  Zhang, Huibing;  Mao, Chunyou;  Zhou, X. Edward
  |  收藏  |  浏览/下载:18/0  |  提交时间:2021/05/24
Structural basis for activation of the growth hormone-releasing hormone receptor 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 10
作者:  
Zhou, Fulai;  Zhang, Huibing;  Cong, Zhaotong;  Zhao, Li-Hua;  Zhou, Qingtong
  |  收藏  |  浏览/下载:32/0  |  提交时间:2020/12/21
Allosteric Regulation of Hsp90 alpha's Activity by Small Molecules Targeting the Middle Domain of the Chaperone 期刊论文  OAI收割
ISCIENCE, 2020, 卷号: 23, 期号: 2, 页码: 46
作者:  
Zhou, Chen;  Zhang, Chi;  Zhu, Hongwen;  Liu, Zhijun;  Su, Haixia
  |  收藏  |  浏览/下载:69/0  |  提交时间:2020/07/01
Discovery of novel CBP bromodomain inhibitors through TR-FRET-based high-throughput screening 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 2, 页码: 286-292
作者:  
Zhang, Feng-cai;  Sun, Zhong-ya;  Liao, Li-ping;  Zuo, Yu;  Zhang, Dan
  |  收藏  |  浏览/下载:48/0  |  提交时间:2020/07/01
Structure and dynamics of the active human parathyroid hormone receptor-1 期刊论文  OAI收割
SCIENCE, 2019, 卷号: 364, 期号: 6436, 页码: 148-+
作者:  
Zhao, Li-Hua;  Ma, Shanshan;  Sutkeviciute, Ieva;  Shen, Dan-Dan;  Zhou, X. Edward
  |  收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Crystal structure of the Frizzled 4 receptor in a ligand-free state 期刊论文  OAI收割
NATURE, 2018, 卷号: 560, 期号: 7720, 页码: 666-+
作者:  
Yang, Shifan;  Wu, Yiran;  Xu, Ting-Hai;  de Waal, Parker W.;  He, Yuanzheng
  |  收藏  |  浏览/下载:81/0  |  提交时间:2019/01/08