中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [22]
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内容类型
发表日期
  • 2019 [22]
学科主题
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浏览/检索结果: 共22条,第1-10条 帮助

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Common activation mechanism of class A GPCRs 期刊论文  OAI收割
ELIFE, 2019, 卷号: 8, 页码: 31
作者:  
Zhou, Qingtong;  Yang, Dehua;  Wu, Meng;  Guo, Yu;  Guo, Wangjing
  |  收藏  |  浏览/下载:76/0  |  提交时间:2020/07/01
Cancer Cell Membrane-Camouflaged Nanorods with Endoplasmic Reticulum Targeting for Improved Antitumor Therapy 期刊论文  OAI收割
ACS APPLIED MATERIALS & INTERFACES, 2019, 卷号: 11, 期号: 50, 页码: 46614-46625
作者:  
Zhang, Wei;  Yu, Miaorong;  Xi, Ziyue;  Nie, Di;  Dai, Zhuo
  |  收藏  |  浏览/下载:44/0  |  提交时间:2020/07/01
A Novel Allosteric Inhibitor of Phosphoglycerate Mutase 1 Suppresses Growth and Metastasis of Non-Small-Cell Lung Cancer 期刊论文  OAI收割
CELL METABOLISM, 2019, 卷号: 30, 期号: 6, 页码: 1107-+
作者:  
Huang, Ke;  Liang, Qian;  Zhou, Ye;  Jiang, Lu-lu;  Gu, Wei-ming
  |  收藏  |  浏览/下载:81/0  |  提交时间:2020/07/01
DeepCPI: A Deep Learning-based Framework for Large-scale in silico Drug Screening 期刊论文  OAI收割
GENOMICS PROTEOMICS & BIOINFORMATICS, 2019, 卷号: 17, 期号: 5, 页码: 478-495
作者:  
Wan, Fangping;  Zhu, Yue;  Hu, Hailin;  Dai, Antao;  Cai, Xiaoqing
  |  收藏  |  浏览/下载:63/0  |  提交时间:2020/07/01
Preclinical evaluation of 3D185, a novel potent inhibitor of FGFR1/2/3 and CSF-1R, in FGFR-dependent and macrophage-dominant cancer models 期刊论文  OAI收割
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2019, 卷号: 38, 期号: 1, 页码: 16
作者:  
Peng, Xia;  Hou, Pengcong;  Chen, Yi;  Dai, Yang;  Ji, Yinchun
  |  收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
Discovery and Development of a Series of Pyrazolo[3,4-d]pyridazinone Compounds as the Novel Covalent Fibroblast Growth Factor Receptor Inhibitors by the Rational Drug Design 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 16, 页码: 7473-7488
作者:  
Wang, Yulan;  Dai, Yang;  Wu, Xiaowei;  Li, Fei;  Liu, Bo
  |  收藏  |  浏览/下载:38/0  |  提交时间:2020/07/01
Thymine DNA glycosylase recognizes the geometry alteration of minor grooves induced by 5-formylcytosine and 5-carboxylcytosine 期刊论文  OAI收割
CHEMICAL SCIENCE, 2019, 卷号: 10, 期号: 31, 页码: 7407-7417
作者:  
Fu, Tianran;  Liu, Liping;  Yang, Qing-Lin;  Wang, Yuxin;  Xu, Pan
  |  收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
Efficient Synthesis of Spirooxindole Pyrrolones by a Rhodium(III)-Catalyzed C-H Activation/Carbene Insertion/Lossen Rearrangement Sequence 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2019, 页码: 6
作者:  
  |  收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01
Cu-Mediated C-H Thioetherification of Arenes at Room Temperature 期刊论文  OAI收割
ORGANIC LETTERS, 2019, 卷号: 21, 期号: 15, 页码: 5981-5985
作者:  
Wang, Xing;  Yi, Xing;  Xu, Hui;  Dai, Hui-Xiong
  |  收藏  |  浏览/下载:7/0  |  提交时间:2020/07/01
Accelerating the Throughput of Affinity Mass Spectrometry-Based Ligand Screening toward a G Protein-Coupled Receptor 期刊论文  OAI收割
ANALYTICAL CHEMISTRY, 2019, 卷号: 91, 期号: 13, 页码: 8162-8169
作者:  
Lu, Yan;  Qin, Shanshan;  Zhang, Bingjie;  Dai, Antao;  Cai, Xiaoqing
  |  收藏  |  浏览/下载:25/0  |  提交时间:2020/07/01