中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Discovery of a highly potent CECR2 bromodomain inhibitor with 7H-pyrrolo[2,3-d] pyrimidine scaffold

期刊论文  OAI收割

BIOORGANIC CHEMISTRY, 2022, 卷号: 123, 页码: 12
作者:  
Lu, Haibo;  Lu, Tian;  Zu, Shijia;  Duan, Zhe;  Guang, Yiman
  |  收藏  |  浏览/下载:24/0  |  提交时间:2022/08/16
Inhibition of the deubiquitinating enzyme USP47 as a novel targeted therapy for hematologic malignancies expressing mutant EZH2 期刊论文  OAI收割
LEUKEMIA, 2022
作者:  
Yang, Jing;  Weisberg, Ellen L.;  Qi, Shuang;  Ni, Wei;  Mei, Husheng
  |  收藏  |  浏览/下载:68/0  |  提交时间:2022/02/14
Brominated Polythiophene Reduces the Efficiency-Stability-Cost Gap of Organic and Quantum Dot Hybrid Solar Cells 期刊论文  OAI收割
ADVANCED ENERGY MATERIALS, 2022, 卷号: 12, 期号: 35, 页码: 2201975
作者:  
Liu, Junwei;  Liu, Yang;  Wang, Jingjing;  Li, Haojin;  Zhou, Kangkang
  |  收藏  |  浏览/下载:2/0  |  提交时间:2023/11/09
Context and auto-interaction are all you need: Towards context embedding based QoS prediction via automatic feature interaction for high quality cloud API delivery 期刊论文  OAI收割
Future Generation Computer Systems, 2021, 卷号: 128, 期号: 2022, 页码: 265-281
作者:  
Zhen Chen;  Maosheng Pan;  Pengfei He;  Wenchao Qi;  Linlin Liu
  |  收藏  |  浏览/下载:51/0  |  提交时间:2021/11/17
Discovery of a subtype-selective, covalent inhibitor against palmitoylation pocket of TEAD3 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 10, 页码: 3206-3219
作者:  
Lu, Tian;  Li, Yong;  Lu, Wenchao;  Spitters, Twgm;  Fang, Xueyu
  |  收藏  |  浏览/下载:45/0  |  提交时间:2021/12/01
Selectively targeting FLT3-ITD mutants over FLT3-wt by a novel inhibitor for acute myeloid leukemia 期刊论文  OAI收割
HAEMATOLOGICA, 2021, 卷号: 106
作者:  
Wang, Aoli;  Hu, Chen;  Chen, Cheng;  Liang, Xiaofei;  Wang, Beilei
  |  收藏  |  浏览/下载:46/0  |  提交时间:2021/04/26
Network-based analysis with primary cells reveals drug response landscape of acute myeloid leukemia 期刊论文  OAI收割
EXPERIMENTAL CELL RESEARCH, 2020, 卷号: 393
作者:  
Chen, Cheng;  Wang, Li;  Li, Lili;  Wang, Aoli;  Huang, Tao
  |  收藏  |  浏览/下载:43/0  |  提交时间:2020/11/26
Discovery of a highly selective VEGFR2 kinase inhibitor CHMFL-VEGFR2-002 as a novel anti-angiogenesis agent 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2020, 卷号: 10
作者:  
Jiang, Zongru;  Wang, Li;  Liu, Xuesong;  Chen, Cheng;  Wang, Beilei
  |  收藏  |  浏览/下载:42/0  |  提交时间:2020/11/26
Discovery and characterization of a novel highly potent and selective type II native and drug-resistant V299L mutant BCR-ABL inhibitor (CHMFL-ABL-039) for Chronic Myeloid Leukemia (CML) 期刊论文  OAI收割
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 6, 页码: 877-885
作者:  
Wu, Jiaxin;  Wang, Aoli;  Li, Xixiang;  Chen, Cheng
  |  收藏  |  浏览/下载:76/0  |  提交时间:2019/11/27
Discovery of 2-(4-Chloro-3-(trifluoromethyl)phenyl)-N-(4-((6,7-dimethoxyquinolin-4-yl)oxy)phenyl)acetamide (CHMFL-KIT-64) as a Novel Orally Available Potent Inhibitor against Broad-Spectrum Mutants of 期刊论文  OAI收割
J. Med. Chem., 2019
作者:  
Yun Wu;  Beilei Wang;  Junjie Wang;  Qi S(亓爽);  Fengming Zou
  |  收藏  |  浏览/下载:41/0  |  提交时间:2020/10/20