中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
采集方式
OAI收割 [7]
内容类型
期刊论文 [7]
发表日期
2022 [7]
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发表日期:2022
专题:上海药物研究所
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Structure-Based Design of Tropane Derivatives as a Novel Series of CCR5 Antagonists with Broad-Spectrum Anti-HIV-1 Activities and Improved Oral Bioavailability
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 24, 页码: 16526-16540
作者:
Xie, Xiong
;
Zheng, Yu-Gui
;
Chen, Huan
;
Li, Jian
;
Luo, Rong-Hua
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/04/10
Multimodule characterization of immune subgroups in intrahepatic cholangiocarcinoma reveals distinct therapeutic vulnerabilities
期刊论文
OAI收割
JOURNAL FOR IMMUNOTHERAPY OF CANCER, 2022, 卷号: 10, 期号: 7, 页码: 14
作者:
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/08/30
tumor microenvironment
cytotoxicity
immunologic
drug therapy
combination
Copy Number Analyses Identified a Novel Gene: APOBEC3A Related to Lipid Metabolism in the Pathogenesis of Preeclampsia
期刊论文
OAI收割
FRONTIERS IN CARDIOVASCULAR MEDICINE, 2022, 卷号: 9, 页码: 13
作者:
Liu, Nan
;
Guo, Yu-Na
;
Wang, Xiao-Jin
;
Ma, Jue
;
He, Yun-Ting
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/08/16
preeclampsia
APOBEC3A
lipid metabolism
copy number variation
genetics
Genome-wide gain-of-function screening identifies EZH2 mediating resistance to PI3K alpha inhibitors in oesophageal squamous cell carcinoma
期刊论文
OAI收割
CLINICAL AND TRANSLATIONAL MEDICINE, 2022, 卷号: 12, 期号: 5, 页码: 17
作者:
Xing, Hui
;
Gao, Mengshi
;
Wang, Yuxiang
;
Zhang, Xu
;
Shi, Jiajie
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2022/08/16
CDKNIA
cell cycle
CRISPR-SAM
CYH33
ESCC
EZH2
PI3K alpha inhibitor
resistance
Characterization of a small-molecule inhibitor targeting NEMO/IKK beta to suppress colorectal cancer growth
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2022, 卷号: 7, 期号: 1, 页码: 13
作者:
Yu, Zhenlong
;
Gao, Jian
;
Zhang, Xiaolei
;
Peng, Yulin
;
Wei, Wenlong
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/06/15
Metabolite profiles and mass balance of fuzuloparib, a novel poly (ADP-ribose) polymerase inhibitor, in subjects with advanced solid cancers
期刊论文
OAI收割
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 2022, 页码: 14
作者:
Bian, Yicong
;
Meng, Jian
;
Ma, Sheng
;
Li, Guangze
;
Wang, Yuya
  |  
收藏
  |  
浏览/下载:79/0
  |  
提交时间:2022/06/15
fuzuloparib
mass balance
metabolite profiles
PARP
pharmacokinetics
Comprehensive Transcriptome Profiling of NAFLD- and NASH-Induced Skeletal Muscle Dysfunction
期刊论文
OAI收割
FRONTIERS IN ENDOCRINOLOGY, 2022, 卷号: 13, 页码: 14
作者:
Guo, Mingwei
;
Xiang, Liping
;
Yao, Jing
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2022/08/30
NAFLD
NASH
quadriceps muscle
lipid deposition
insulin resistance
myokines