中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海神经科学研究所 [23]
上海药物研究所 [5]
昆明植物研究所 [4]
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中国科学院大学 [1]
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期刊论文 [32]
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TRP (transient receptor potential) ion channel family: structures, biological functions and therapeutic interventions for diseases
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 38
作者:
Zhang, Miao
;
Ma, Yueming
;
Ye, Xianglu
;
Zhang, Ning
;
Pan, Lei
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
Synthesis of AC1903 analogs as potent transient receptor potential canonical channel 4/5 inhibitors and biological evaluation
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 68, 页码: 11
作者:
Chen, Lili
;
Zhang, Zhuang
;
Tian, Hongtao
;
Jiang, Shan
;
Ji, Yunyun
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/11/11
TRPC5
AC1903
Podocyte
FSGS
Keratinocyte
Proliferation
Inflammation
Discovery of novel modulators targeting human TRPC5: Docking-based virtual screening, molecular dynamics simulation and binding af fi nity predication
期刊论文
OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2021, 卷号: 102, 页码: 107795
作者:
Liu,Bin
;
Zhang,Wei
;
Guo,Sheng
;
Zuo,Zhili
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/04/02
hTRPC5
Homology modeling
Molecular docking
Molecular dynamics simulation
Virtual screening
INHIBITOR
CHANNELS
GROMACS
POTENT
AMBER
IDENTIFICATION
CONSTRAINTS
INTEGRATION
AMYGDALA
Pyrazolopyrimidines as Potent Stimulators for Transient Receptor Potential Canonical 3/6/7 Channels
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 11, 页码: 4680-4692
作者:
Qu, Chunrong
;
Ding, Mingmin
;
Zhu, Yingmin
;
Lu, Yungang
;
Du, Juan
  |  
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2019/01/08
Benzimidazole derivative M084 extends the lifespan of Caenorhabditis elegans in a DAF-16/FOXO-dependent way
期刊论文
OAI收割
MOLECULAR AND CELLULAR BIOCHEMISTRY, 2017, 卷号: 426, 期号: 1-2, 页码: 101-109
作者:
Ding, Ai-Jun
;
Wu, Gui-Sheng
;
Tang, Bin
;
Hong, Xuechuan
;
Zhu, Michael X.
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2017/05/19
Aging
Benzimidazole derivative M084
Caenorhabditis elegans
Lifespan
Acute Treatment with a Novel TRPC4/C5 Channel Inhibitor Produces Antidepressant and Anxiolytic-Like Effects in Mice
期刊论文
OAI收割
PLOS ONE, 2015, 卷号: 10, 期号: 8
作者:
Yang, Li-Ping
;
Jiang, Fang-Jie
;
Wu, Gui-Sheng
;
Deng, Ke
;
Wen, Meng
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2016/01/19
Identification and optimization of 2-aminobenzimidazole derivatives as novel inhibitors of TRPC4 and TRPC5 channels
期刊论文
OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2015, 卷号: 172, 期号: 14, 页码: 3495-3509
作者:
Zhu, Yingmin
;
Lu, Yungang
;
Qu, Chunrong
;
Miller, Melissa
;
Tian, Jinbin
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2015/12/15
Ca2+ signaling initiated by canonical transient receptor potential channels in dendritic development
期刊论文
OAI收割
NEUROSCIENCE BULLETIN, 2015, 卷号: 31, 期号: 3, 页码: 351-356
作者:
Feng, SJ
;
He, ZH
;
Li, HY
;
Wang, YZ
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2015/12/30
NEURITE OUTGROWTH
TRPC CHANNELS
NEUROTROPHIC FACTORS
HIPPOCAMPAL-NEURONS
CATION CHANNEL
GROWTH CONES
BRAIN
CELLS
BDNF
NEUROBLASTS
Crucial role of TRPC6 in maintaining the stability of HIF-1 alpha in glioma cells under hypoxia
期刊论文
OAI收割
JOURNAL OF CELL SCIENCE, 2015, 卷号: 128, 期号: 17, 页码: 3317-3329
作者:
Li, SS
;
Wang, JK
;
Wei, Y
;
Liu, YJ
;
Ding, X
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2015/12/30
SMOOTH-MUSCLE-CELLS
OPERATED CA2+ CHANNELS
CALCIUM OSCILLATIONS
CANCER METABOLISM
TUMOR-SUPPRESSOR
INDUCIBLE FACTOR-1-ALPHA
PROLYL HYDROXYLATION
ENDOTHELIAL-CELLS
DENDRITIC GROWTH
CATION CHANNELS
Canonical transient receptor potential 4 and its small molecule modulators
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2015, 卷号: 58, 期号: 1, 页码: 39-47
作者:
Fu Jie
;
Gao ZhaoBing
;
Shen Bing
;
Zhu, Michael X.
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
TRPC4 channel
non-selective cation channel
G protein coupled receptors
small molecular modulators
G proteins
excitation
contraction
Ca2+ signaling