中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [11]
采集方式
OAI收割 [11]
内容类型
期刊论文 [11]
发表日期
2024 [2]
2023 [1]
2022 [2]
2021 [1]
2020 [1]
2013 [2]
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Asymmetric macrocyclization enabled by Rh(III)-catalyzed C-H activation: Enantioenriched macrocyclic inhibitor of Zika virus infection
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2024, 卷号: 35, 期号: 11, 页码: 6
作者:
Chen, Chao
;
Yu, Wenwen
;
Huang, Guangen
;
Ren, Xuelian
;
Chen, Xiangli
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/09/26
C -H activation
Carboamidation
Enantioselective macrocyclization
Anti-Zika virus activity
Controlled Reversible N-Terminal Modification of Peptides and Proteins
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2024, 卷号: 146, 期号: 34, 页码: 23752-23763
作者:
Lin, Zeng
;
Liu, Bo
;
Lu, Mengru
;
Wang, Yongqin
;
Ren, Xuelian
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/09/26
Discovery and Structural Optimization of Covalent ZAP-70 Kinase Inhibitors against Psoriasis
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 15
作者:
Rao, Danni
;
Yang, Tao
;
Feng, Huixu
;
An, Qi
;
Zhang, Shaofeng
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2023/10/17
SLL-627 Is a Highly Selective and Potent ? Opioid Receptor (KOR) Agonist with an Unexpected Nonreduction in Locomotor Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 16
作者:
Kong, Linghui
;
Shu, Xuelian
;
Tang, Siyuan
;
Ye, Rongrong
;
Sun, Huijiao
  |  
收藏
  |  
浏览/下载:60/0
  |  
提交时间:2022/08/30
A Traceless Site-Specific Conjugation on Native Antibodies Enables Efficient One-Step Payload Assembly
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2022, 页码: 11
作者:
Zeng, Yue
;
Shi, Wei
;
Dong, Qian
;
Li, Wanzhen
;
Zhang, Jianxin
  |  
收藏
  |  
浏览/下载:71/0
  |  
提交时间:2022/08/30
Acyl Transfer
Anti-Tumor
One-Step Synthesis
Site-Specific ADCs
Thioester
Discovery of a potent, selective, and covalent ZAP-70 kinase inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 219, 页码: 12
作者:
Rao, Danni
;
Li, Heng
;
Ren, Xuelian
;
Sun, Yaoliang
;
Wen, Cuiyun
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2021/08/17
Zeta-chain associated protein kinase 70 kDa (ZAP-70)
Covalent inhibitor
T cell
Autoimmune diseases
Manipulating the Click Reactivity of Dibenzoazacyclooctynes: From Azide Click Component to Caged Acylation Reagent by Silver Catalysis
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2020, 页码: 6
作者:
Shi, Wei
;
Tang, Feng
;
Ao, Jiwei
;
Yu, Qun
;
Liu, Junjie
  |  
收藏
  |  
浏览/下载:140/0
  |  
提交时间:2020/12/21
acylation
click chemistry
peptides
rearrangements
silver
Structure-Based Design and Synthesis of C-1- and C-4-Modified Analogs of Zanamivir as Neuraminidase Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 3, 页码: 671-684
作者:
Feng, Enguang
;
Shin, Woo-Jin
;
Zhu, Xuelian
;
Li, Jian
;
Ye, Deju
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
Toll-like receptor 4/nuclear factor-kappa B signaling pathway is involved in ACTG-toxin H-mediated anti-inflammatory effect
期刊论文
OAI收割
MOLECULAR AND CELLULAR BIOCHEMISTRY, 2013, 卷号: 374, 期号: 1-2, 页码: 29-36
作者:
Yang, Xinying
;
Zhang, Guojian
;
Tang, Xuelian
;
Jiao, Jieying
;
Kim, Sung Yeon
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
ACTG-toxin H
LPS
TLR4/NF kappa B
Efficacy and Toxicity of 5-Fluorouracil in Colon Cancer Treatment of a Mouse Syngeneic Model
期刊论文
OAI收割
Journal of South China Agricultural University, 2012, 卷号: 33, 期号: 4, 页码: 535-538
作者:
Tang Xuelian
;
Fu Jinghua
;
Park Hyun
;
Yang Xinying
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
5-fluorouracil
efficacy
toxicity
colon cancer