中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共58条,第1-10条 帮助

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Ginkgetin Alleviates Inflammation and Senescence by Targeting STING 期刊论文  OAI收割
ADVANCED SCIENCE, 2024, 页码: 15
作者:  
Liu, Yadan;  Ye, Jialin;  Fan, Zisheng;  Wu, Xiaolong;  Zhang, Yinghui
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/12/16
An updated patent review of SOS1 inhibitors (2022-present) 期刊论文  OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2024, 页码: 15
作者:  
Zhou, Guizhen;  Zhou, Chuan;  Ma, Xinyi;  Xu, Jiahang;  Zhou, Zehui
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/12/11
Design, synthesis, and bioevaluation of SOS1 PROTACs derived from pyrido [2,3- d ]pyrimidin-7-one-based SOS1 inhibitor 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 107, 页码: 9
作者:  
Wang, Kun;  Zhou, Zehui;  Ma, Xinyi;  Xu, Jiahang;  Xu, Wangyang
  |  收藏  |  浏览/下载:21/0  |  提交时间:2024/07/12
Roles of photochemical consumption of VOCs on regional background O3 concentration and atmospheric reactivity over the pearl river estuary, Southern China 期刊论文  OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2024, 卷号: 928, 页码: 10
作者:  
Sun, Jiayin;  Yu, Xiaoyu;  Ling, Zhenhao;  Fang, Guizhen;  Ming, Lili
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/09/13
Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRASG12D 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:  
Zhou, Chuan;  Fan, Zisheng;  Gu, Yuejiao;  Ge, Zhiming;  Tao, Zhaofan
  |  收藏  |  浏览/下载:25/0  |  提交时间:2024/02/27
Discovery of a Potent, Cooperative, and Selective SOS1 PROTAC ZZ151 with In Vivo Antitumor Efficacy in KRAS-Mutant Cancers 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 6, 页码: 4197-4214
作者:  
Zhou, Zehui;  Zhou, Guizhen;  Zhou, Chuan;  Fan, Zisheng;  Cui, Rongrong
  |  收藏  |  浏览/下载:24/0  |  提交时间:2024/03/27
Design, Synthesis, and Biological Evaluation of Bipyridazine Derivatives as Stimulator of Interferon Genes (STING) Receptor Agonists 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 5, 页码: 3327-3347
作者:  
Shan, Bin;  Hou, Hui;  Zhang, Keke;  Li, Rui;  Shen, Chang
  |  收藏  |  浏览/下载:22/0  |  提交时间:2024/03/27
Design, Synthesis, and Bioevaluation of Pyrido[2,3-d]pyrimidin-7-ones as Potent SOS1 Inhibitors 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2023, 页码: 183-190
作者:  
Liu, Meiying;  Zhou, Guizhen;  Su, Wenhong;  Gu, Yuejiao;  Gao, Mingshan
  |  收藏  |  浏览/下载:23/0  |  提交时间:2024/03/27
Discovery of ARF1-targeting inhibitor demethylzeylasteral as a potential agent against breast cancer 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 5, 页码: 2619-2622
作者:  
Chang, Jie;  Yang, Ruirui;  Chen, Lifan;  Fan, Zisheng;  Zhou, Jingyi
  |  收藏  |  浏览/下载:44/0  |  提交时间:2022/08/16
Discovery of the First-in-Class Agonist-Based SOS1 PROTACs Effective in Human Cancer Cells Harboring Various KRAS Mutations 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 5, 页码: 3923-3942
作者:  
Zhou, Chuan;  Fan, Zisheng;  Zhou, Zehui;  Li, Yupeng;  Cui, Rongrong
  |  收藏  |  浏览/下载:55/0  |  提交时间:2022/06/15