中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [107]
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Benzothiazole amide analogues as antagonists of TRPC 6 channels: A therapeutic approach for kidney fibrosis
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 291, 页码: 16
作者:
Ren, Chunlin
;
Xu, Qiding
;
Luo, Qiusi
;
Qiao, Xue
;
Ding, Taotao
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/06/23
Transient receptor potential canonical 6
channels
Antagonist
Renal fibrosis
Benzothiazole derivatives
Unilateral ureteral obstruction
Diverse Secondary Metabolites From the
Ligia exotica-
Derived Fungus
Diaporthe melitensis
HZ-1
期刊论文
OAI收割
CHEMISTRY & BIODIVERSITY, 2025, 页码: 7
作者:
Zhu, Ming-Xin
;
Hao, Yi
;
Yan, Bing-Yuan
;
Jin, Yang
;
Gao, Zhen
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/06/23
antibacterial activities
Diaporthe melitensis
Ligia exotica
marine natural products
Enhancing fluorescent probe design through multilayer interaction convolutional networks: advancing biosensing and bioimaging precision
期刊论文
OAI收割
CHEMICAL SCIENCE, 2025, 页码: 8
作者:
Ma, Gongcheng
;
Ding, Qihang
;
Zhang, Yuding
;
Zeng, Xiaodong
;
Zhu, Kai
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/06/23
Development of
99m
Tc-labeled melanin-targeted probes for SPECT imaging of melanoma
期刊论文
OAI收割
EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2025, 页码: 14
作者:
Tao, Ji
;
Cao, Rui
;
Lei, Zhe
;
Wang, Xiao
;
Luo, Renli
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/06/23
Melanoma
Melanin
(99m)Technetium
SPECT
Imaging probe
Exploring and expanding the natural chemical space of bacterial diterpenes
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 9
作者:
Wei, Xiuting
;
Ning, Wenbo
;
Mccadden, Caitlin A.
;
Alsup, Tyler A.
;
Li, Zining
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/06/23
Design, Synthesis, and Biological Evaluation of Peptidomimetic Tetrahydropyrrole Spirodihydroindolones as SARS-CoV-2 3CL Protease Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 16, 期号: 5, 页码: 790-796
作者:
Hu, Liuyan
;
Zhao, Zhi
;
Zhang, Shujing
;
Yang, Lei
;
Cui, Wenjie
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/06/23
COVID-19
SARS-CoV-2
3CL protease
Peptidomimetic inhibitors
Tetrahydropyrrole spirodihydroindolone
Discovery of 2,4-quinazolinedione derivatives as LC3B recruiters in the facilitation of protein complex degradations
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 287, 页码: 10
作者:
Zeng, Yanping
;
Xiao, Jian
;
Shi, Li
;
Li, Yangsha
;
Xu, Yuanxin
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2025/04/01
LC3B
CDK9
Degradation
Protein complex
Apigenin alleviates inflammation as a natural IRAK4 inhibitor
期刊论文
OAI收割
PHYTOMEDICINE, 2025, 卷号: 139, 页码: 12
作者:
Gongpan, Pianchou
;
Xu, Tingting
;
Zhang, Yufei
;
Ji, Kailong
;
Kong, Lingmei
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/04/24
Apigenin
IRAK4 inhibitor
Anti-inflammation
NF-kappa B
MAPK pathways
Ulcerative colitis
Phomaligol J, a New Cyclohexenone With Antibacterial Activity From a Pufferfish-Associated Fungus
Aspergillus austwickii
期刊论文
OAI收割
CHEMISTRY & BIODIVERSITY, 2025, 页码: 6
作者:
Du, Wang-Yang
;
Wang, Hui-Fang
;
Sun, Ruo-Nan
;
Jin, Yang
;
Wang, Hai-Feng
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/05/27
antibacterial activity
Aspergillus austwickii
associated
cyclohexenone
pufferfish
Design, Synthesis, and biological evaluation of 7H-Pyrrolo[2,3-d] pyrimidines as potent HPK1 kinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 119, 页码: 13
作者:
Wu, Feifei
;
Li, Huiyu
;
Li, Weiqiang
;
Zhang, Laishun
;
An, Qi
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/04/01
Optimization
Hematopoietic progenitor kinase 1
Inhibitor
Cancer immunotherapy