中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共155条,第1-10条 帮助

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Design, synthesis and bio-evaluation of 2,5-disubstituted thiazole derivatives for potential treatment of acute myeloid leukemia through targeting CDK9 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2025, 卷号: 160, 页码: 16
作者:  
Chen, Sumeng;  Huang, Jindi;  Zhang, Shipeng;  Zheng, Xinni;  Chen, Hongming
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 18, 页码: 15469-15481
作者:  
Wu, Xinyuan;  Pan, Jiayi;  Fan, Rufeng;  Zhang, Yiwei;  Wang, Chao
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:  
Wu, Xinyuan;  Li, Shunyao;  Liang, Ting;  Yu, Qing;  Zhang, Yiwei
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Phosphatidylinositol 4,5-bisphosphate activation mechanism of human KCNQ5 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 14, 页码: 11
作者:  
Yang, Zhenni;  Zheng, Yueming;  Ma, Demin;  Wang, Long;  Zhang, Jiatong
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
A holistic strategy for the in-depth discrimination and authentication of 16 citrus herbs and associated commercial products based on machine learning techniques and non-targeted metabolomics 期刊论文  OAI收割
JOURNAL OF CHROMATOGRAPHY A, 2025, 卷号: 1745, 页码: 12
作者:  
Huang, Yu-shi;  An, Ya-ling;  Zheng, Yue-yuan;  Zhao, Wen-jie;  Song, Chun-qian
  |  收藏  |  浏览/下载:17/0  |  提交时间:2025/04/01
Time-Dependent Regulation of Sleep-Wakefulness and Electroencephalographic Characteristics by Spontaneous Running in Male Mice 期刊论文  OAI收割
JOURNAL OF SLEEP RESEARCH, 2025, 页码: 16
作者:  
Zhou, Wufang;  Zhou, Jialin;  Lu, Qianyu;  Wang, Long;  Liang, Yutao
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/05/27
Current landscape of metal-organic framework-mediated nucleic acid delivery and therapeutics 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2025, 卷号: 672, 页码: 21
作者:  
Feng, Shiwei;  Li, Yan;  Tan, Zheng;  Shen, Shiyang
  |  收藏  |  浏览/下载:11/0  |  提交时间:2025/04/01
An efficient deep learning-based strategy to screen inhibitors for GluN1/GluN3A receptor 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 9
作者:  
Wang, Ze-chen;  Zeng, Yue;  Sun, Jin-yuan;  Chen, Xue-qin;  Wu, Hao-chen
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/04/24
Development of novel epoxyketone macrocyclic peptidyl proteasome inhibitors through OPA-mediated one-step cyclization of unprotected peptides 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2025, 卷号: 156, 页码: 16
作者:  
Zeng, Gongruixue;  Xu, Gaoya;  Gao, Lixin;  Zheng, Xiaoli;  Chi, Xinglong
  |  收藏  |  浏览/下载:13/0  |  提交时间:2025/04/01
Harnessing the Magic Methyl Effect: Discovery of CLPP-2068 as a Novel HsClpP Activator for the Treatment of Diffuse Large B-Cell Lymphoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 4, 页码: 4287-4307
作者:  
Sun, Mingyang;  Chen, Beijing;  Teng, Dan;  Zhao, Hongshen;  Liao, Yilie
  |  收藏  |  浏览/下载:16/0  |  提交时间:2025/04/01