中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Design, Synthesis, and Pharmacological Evaluation of Quinazoline and Quinoline Derivatives as Potent ENPP1 Inhibitors for Cancer Immunotherapy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 18
作者:
He, Jie
;
Ma, Xiaoyu
;
Sun, Jia
;
Chen, Manman
;
Xu, Lan
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2025/04/01
Design, synthesis and pharmacological evaluation of 1,2,3,4-tetrahydrobenzofuro[2,3-c] pyridine derivatives as p21-activated kinase 4 inhibitors for treatment of pancreatic cancer
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 1, 页码: 438-466
作者:
Li, Yang
;
Fang, Yan
;
Chen, Xiaoyu
;
Tong, Linjiang
;
Feng, Fang
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/04/01
P21-activated kinase 4
Tetrahydrobenzofuro[2
3-c]pyridine
Structure-activity relationship
Allosteric inhibitor
Pharmacokinetics properties
Kinase selectivity
Pancreatic cancer
Immune infiltration
Attentional network deficits in patients with migraine: behavioral and electrophysiological evidence
期刊论文
OAI收割
JOURNAL OF HEADACHE AND PAIN, 2024, 卷号: 25, 期号: 1, 页码: 16
作者:
Chen, Yuxin
;
Xie, Siyuan
;
Zhang, Libo
;
Li, Desheng
;
Su, Hui
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/12/09
Migraine
Attention
Electroencephalography (EEG)
Vigilance
Hypersensitivity
Machine learning
Zinc isotope perspective on global carbon cycling during the onset of the late Paleozoic icehouse
期刊论文
OAI收割
GEOLOGY, 2024, 页码: 6
作者:
Zhong, Yutian
;
Chen, Jitao
;
Liu, Sheng-Ao
;
Yuan, Chengshuai
;
Gao, Biao
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/03/28
Brain-to-brain synchrony increased during interpersonal touch in romantic lovers: an EEG-based hyperscanning study
期刊论文
OAI收割
BMC PSYCHOLOGY, 2024, 卷号: 12, 期号: 1, 页码: 14
作者:
Zhou, Chenghao
;
Jiang, Xiaowei
;
Chen, Yanan
;
Ge, Chunlei
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/11/18
EEG-based hyperscanning
Interpersonal touch
Brain-to-brain synchrony
Romantic love
Dynamic interpersonal functional connectivity
GeneCompass: deciphering universal gene regulatory mechanisms with a knowledge-informed cross-species foundation model
期刊论文
OAI收割
CELL RESEARCH, 2024, 页码: 16
作者:
Yang, Xiaodong
  |  
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2024/12/06
Sesquiterpene lactones from
Tithonia diversifolia
with ferroptosis-inducing activities
期刊论文
OAI收割
PHYTOCHEMISTRY, 2024, 卷号: 226, 页码: 12
作者:
Ding, Ao-Xue
;
Shan, Yi -Ming
;
Li, Chen-Yue
;
Qin, Guo -Qing
;
Chen, Tong
  |  
收藏
  |  
浏览/下载:88/0
  |  
提交时间:2024/08/22
Tithonia diversifolia
Asteraceae
Sesquiterpene lactones
Ferroptosis
Cytotoxic effects
Molecular Dynamics Insights into Mechanical Stability, Elastic Properties, and Fracture Behavior of PHOTH-Graphene
期刊论文
OAI收割
MATERIALS, 2024, 卷号: 17, 期号: 19, 页码: 20
作者:
Peng, Qing
;
Chen, Gen
;
Huang, Zeyu
;
Chen, Xue
;
Li, Ao
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/11/14
PHOTH-graphene
mechanical property
MD
defects
hydrogen functionalization
Characterization and noncovalent inhibition of the K63-deubiquitinase activity of SARS-cov-2 PLpro
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2024, 卷号: 228, 页码: 12
作者:
Liu, Xin
;
Zheng, Miao
;
Zhang, Hongqing
;
Feng, Bo
;
Li, Jiaqi
  |  
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2024/10/21
Discovery of a Highly Potent and Selective BRD9 PROTAC Degrader Based on E3 Binder Investigation for the Treatment of Hematological Tumors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 28
作者:
Duan, Haiting
;
Zhang, Jingyu
;
Gui, Renzhao
;
Lu, Yang
;
Pang, Ao
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/08/20