中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
地理科学与资源研究所 [4]
植物研究所 [3]
成都生物研究所 [2]
武汉植物园 [2]
南海海洋研究所 [1]
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OAI收割 [22]
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期刊论文 [23]
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2025 [3]
2024 [2]
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2020 [3]
2018 [4]
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Pharmacokinetics and Safety of TPN171 (a PDE5 Inhibitor) in Patients With Mild or Moderate Hepatic Impairment Versus Participants With Normal Hepatic Function: A Phase I Study
期刊论文
OAI收割
CLINICAL PHARMACOLOGY IN DRUG DEVELOPMENT, 2025, 页码: 7
作者:
Zhou, Jing
;
Zhang, Hong
;
Ding, Yanhua
;
Wang, Zhen
;
Wang, Yu
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/06/23
hepatic impairment
pharmacokinetics
phosphodiesterase-5 inhibitor
TPN171
Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:
Wu, Xinyuan
;
Li, Shunyao
;
Liang, Ting
;
Yu, Qing
;
Zhang, Yiwei
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/06/23
Activity-based protein profiling data
Covalent DNA-encoded chemical library
Covalent ligand selection
Lysine-targeting covalent inhibitors
A Phase I Study to Evaluate the Pharmacokinetics and Safety of TPN171 (a PDE5 Inhibitor) in Adults with Renal Impairment
期刊论文
OAI收割
CLINICAL PHARMACOLOGY IN DRUG DEVELOPMENT, 2025, 页码: 8
作者:
Fu, Ping
;
Song, Yi
;
Hu, Chao
;
Yong, Xiaolan
;
Yu, Yang
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/06/23
pharmacokinetics
phosphodiesterase 5 inhibitor
renal impairment
safety
TPN171
Enhancing the Predictive Power of Machine Learning Models through a Chemical Space Complementary DEL Screening Strategy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 12
作者:
Suo, Yanrui
;
Qian, Xu
  |  
收藏
  |  
浏览/下载:98/0
  |  
提交时间:2024/11/26
A Vancomycin-Templated DNA-Encoded Library for Combating Drug-Resistant Bacteria
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3778-3794
作者:
Guan, Dongliang
;
Liu, Jiaxiang
;
Chen, Feifei
;
Li, Jian
;
Wang, Xiaowen
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/05/07
DNA-encoded focused indazole library synthesis by a palladium- mediated C-N(sp(2)) cross-coupling reaction between DNA-linked (hetero)aryl halides and aromatic nitrogen heterocycles
期刊论文
OAI收割
TETRAHEDRON LETTERS, 2022, 卷号: 96, 页码: 6
作者:
Yang, Juan
;
Xia, Shengdi
;
Liu, Jiaxiang
;
Yu, Zikun
;
Mei, Lianghe
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2022/08/16
Human-Climate Coupled Changes in Vegetation Community Complexity of China Since 1980s
期刊论文
OAI收割
EARTHS FUTURE, 2022, 卷号: 10, 期号: 7
作者:
Su, Yanjun
;
Guo, Qinghua
;
Guan, Hongcan
;
Hu, Tianyu
;
Jin, Shichao
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2024/03/07
vegetation community complexity
human activities
climate change
vegetation map
A visual and full-field method for detecting quench and normal zone propagation in HTS tapes
期刊论文
OAI收割
Superconductor Science and Technology, 2021, 卷号: 35, 期号: 2
作者:
Wang,Shudan
;
Guan,Mingzhi
;
Chen,Jiaxiang
;
Wang,Xingzhe
;
Zhou,Youhe
  |  
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2022/01/18
HTS coated tape
quench and propagation
quench detection method
thermoelastic strain-rate
DIC full-field technique
Diversified strategy for the synthesis of DNA-encoded oxindole libraries
期刊论文
OAI收割
CHEMICAL SCIENCE, 2021, 卷号: 12, 期号: 8, 页码: 2841-2847
作者:
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2021/05/24
An updated Vegetation Map of China (1:1000000)
期刊论文
OAI收割
SCIENCE BULLETIN, 2020, 卷号: 65, 期号: 13, 页码: 1125-1136
作者:
Su, Yanjun
;
Guo, Qinghua
;
Hu, Tianyu
;
Guan, Hongcan
;
Jin, Shichao
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2020/10/04