中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共190条,第1-10条 帮助

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Fluorescence-Coupled Ubiquitination Assay as a High-Throughput Screening Strategy for Novel Cereblon Degraders 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 10111-10127
作者:  
Deng, Yanan;  Yang, Shiling;  Xu, Hesong;  Ding, Xiyao;  Xu, Ying
  |  收藏  |  浏览/下载:3/0  |  提交时间:2025/06/23
Design, synthesis and pharmacological evaluation of 1,2,3,4-tetrahydrobenzofuro[2,3-c] pyridine derivatives as p21-activated kinase 4 inhibitors for treatment of pancreatic cancer 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 1, 页码: 438-466
作者:  
Li, Yang;  Fang, Yan;  Chen, Xiaoyu;  Tong, Linjiang;  Feng, Fang
  |  收藏  |  浏览/下载:16/0  |  提交时间:2025/04/01
Pathfinding Pulsar Observations with the CVN Incorporating the FAST 期刊论文  OAI收割
CHINESE PHYSICS LETTERS, 2024, 卷号: 41, 期号: 11, 页码: 117501
作者:  
Yan, Zhen;  Shen, Zhiqiang;  Jiang, Peng;  Zhang, Bo
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/12/06
Structure-Based Drug Design of 2-Amino-[1,1′-biphenyl]-3-carboxamide Derivatives as Selective PKMYT1 Inhibitors for the Treatment of CCNE1-Amplified Breast Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:  
Wang, Chaofan;  Fang, Yan;  Zhou, Ziqin;  Liu, Zhuoheng;  Feng, Fang
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/09/26
Branched-chain amino acid transaminase 1 confers EGFR-TKI resistance through epigenetic glycolytic activation 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 17
作者:  
Zhang, Tao;  Pan, Zilu;  Gao, Jing;  Wu, Qingqing;  Bai, Gang
  |  收藏  |  浏览/下载:25/0  |  提交时间:2024/10/21
Discovery of a Covalent Inhibitor That Overcame Resistance to Venetoclax in AML Cells Overexpressing BFL-1 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 36
作者:  
Lou, Jianfeng;  Zhou, Qianqian;  Lyu, Xilin;  Cen, Xinyi;  Liu, Chen
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/08/22
GFPBW1, a β-glucan from Grifola frondosa as vaccine adjuvant: APCs activation and maturation 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 11
作者:  
He, Xiang;  Lu, Jiang-ling;  Liao, Wen-feng;  Long, Yi-ru;  Zhang, Xing
  |  收藏  |  浏览/下载:18/0  |  提交时间:2024/08/20
Mapping Brain Synergy Dysfunction in Schizophrenia: Understanding Individual Differences and Underlying Molecular Mechanisms 期刊论文  OAI收割
ADVANCED SCIENCE, 2024, 页码: 16
作者:  
Ding, Chaoyue;  Li, Ang;  Xie, Sangma;  Tian, Xiaohan
  |  收藏  |  浏览/下载:22/0  |  提交时间:2024/09/09
Discovery of a novel BTK inhibitor S-016 and identification of a new strategy for the treatment of lymphomas including BTK inhibitor-resistant lymphomas 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 11
作者:  
Song, Pei-ran;  Wan, Zhi-peng;  Huang, Ge-ge;  Song, Zi-lan;  Zhang, Tao
  |  收藏  |  浏览/下载:75/0  |  提交时间:2024/07/12
Pharmacokinetics, mass balance, and metabolism of [14C]envonalkib (TQ-B3139), a novel ALK tyrosine kinase inhibitor, in healthy Chinese subjects 期刊论文  OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2024, 页码: 11
作者:  
Ma, Sheng;  Wang, Xin;  Yan, Shu;  Miao, Liyan;  Wan, Xiaojing
  |  收藏  |  浏览/下载:27/0  |  提交时间:2024/05/07