中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
西安光学精密机械研究... [2]
上海硅酸盐研究所 [2]
地理科学与资源研究所 [1]
上海生物化学与细胞生... [1]
云南天文台 [1]
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采集方式
OAI收割 [16]
内容类型
期刊论文 [16]
发表日期
2024 [6]
2023 [2]
2022 [1]
2021 [1]
2020 [1]
2019 [1]
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学科主题
天文学 [1]
天文学::星系与宇宙... [1]
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Discovery of a Potent, selective and orally bioavailable CDK9 degrader for targeting transcription regulation in Triple-Negative breast cancer
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 153, 页码: 16
作者:
Nie, Hui-Jun
;
Li, Ben-Fu
;
Sun, Jingya
;
Yuan, Yali
;
Zhang, Zhi-Gao
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/11/26
Triple-negative breast cancer
Targeting transcription regulation
Orally bioavailable degrader
PROTAC
Cyclin-dependent Kinase 9
Physical mechanism-based simulation methods for soil and ground heat flux from observations at multi-sites
期刊论文
OAI收割
JOURNAL OF HYDROLOGY, 2024, 卷号: 645, 页码: 132168
作者:
Liu, Zhaofei
;
Jiang, Dong
;
Wang, Rui
;
Hao, Mengmeng
;
Zhang, Xingxing
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/12/20
Ground heat flux
Soil heat flux
Simulation
Gradient method
Calorimetry method
Triple collocation
Tibetan Plateau
Radioactive ADME Demonstrates ARV-110's High Druggability Despite Low Oral Bioavailability
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 15
作者:
He, Yifei
;
Zheng, Yuandong
;
Zhu, Chenggu
;
Lei, Peng
;
Yu, Jinghua
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/09/26
Discovery of Orally Bioavailable and Potent CDK9 Inhibitors for Targeting Transcription Regulation in Triple-Negative Breast Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 12, 页码: 10035-10056
作者:
Wang, Wen-Jing
;
Gao, Lixin
;
Wang, Simei
;
Huang, Wensi
;
Meng, Xin-Yu
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/08/20
Metabolism investigation of the peptide-drug conjugate LN005 in rats using UHPLC-HRMS
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2024, 卷号: 238, 页码: 11
作者:
Wang, Weiqiang
;
Chen, Chong
;
Luo, Jing
;
Tang, Chongzhuang
;
Zheng, Yuandong
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2024/01/16
LN005
Metabolism
Peptide -drug conjugates
UHPLC-HRMS
Doxorubicin
Metabolite characterisation of the peptide-drug conjugate LN005 in liver S9s by UHPLC-Orbitrap-HRMS
期刊论文
OAI收割
XENOBIOTICA, 2024, 页码: 9
作者:
Yuan, Yali
;
Wang, Weiqiang
;
Luo, Jing
;
Tang, Chongzhuang
;
Zheng, Yuandong
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/02/19
peptide-drug conjugate
PDC
LN005
metabolite identification
liver S9s
A validated LC-MS/MS method for the quantification of bevacizumab in rat, cynomolgus monkey, and human serum
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2023, 卷号: 235, 页码: 11
作者:
Zhou, Ainan
;
Yu, Jinghua
;
Wu, Yali
;
Xue, Hao
;
Zhong, Dafang
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/10/17
Monoclonal antibody
Bevacizumab
LC-MS
MS
Surrogate peptide
Pharmacokinetics
Serum
Covalent Binding Mechanism of Furmonertinib and Osimertinib With Human Serum AlbuminS
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2023, 卷号: 51, 期号: 1, 页码: 8-16
作者:
Wu, Yali
;
Chen, Lili
;
Chen, Jian
;
Xue, Hao
;
He, Qingfeng
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/27
A Census of Optically Dark Massive Galaxies in the Early Universe from Magnification by Lensing Galaxy Clusters
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL, 2022, 卷号: 926, 期号: 2
作者:
Shu, Xinwen
;
Yang, Lei
;
Liu, Daizhong
;
Wang, Wei-Hao
;
Wang, Tao
  |  
收藏
  |  
浏览/下载:78/0
  |  
提交时间:2022/03/16
Recent progress of integrated circuits and optoelectronic chips
期刊论文
OAI收割
SCIENCE CHINA-INFORMATION SCIENCES, 2021, 卷号: 64, 期号: 10, 页码: 201401
作者:
Hao, Yue
;
Xiang, Shuiying
;
Han, Genquan
;
Zhang, Jincheng
;
Ma, Xiaohua
;
Zhu, Zhangming
;
Guo, Xingxing
;
Zhang, Yahui
;
Han, Yanan
;
Song, Ziwei
;
Liu, Yan
;
Yang, Ling
;
Zhou, Hong
;
Shi, Jiangyi
;
Zhang, Wei
;
Xu, Min
;
Zhao, Weisheng
;
Pan, Biao
;
Huang, Yangqi
;
Liu,
  |  
收藏
  |  
浏览/下载:64/0
  |  
提交时间:2022/03/28