中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
采集方式
内容类型
发表日期
学科主题
筛选

浏览/检索结果: 共6条,第1-6条 帮助

条数/页: 排序方式:
Discovery of Thiochroman Derivatives as Potent, Oral Selective Estrogen Receptor Degraders and Antagonists for the Treatment of Endocrine-Resistant Breast Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 23, 页码: 21545-21567
作者:  
Zhang, Dan;  Lu, Zhengyu;  He, Yongqi;  Leng, Xin-Yu;  Meng, Xin
  |  收藏  |  浏览/下载:19/0  |  提交时间:2025/01/06
Discovery of Thieno[2,3-e]indazole Derivatives as Novel Oral Selective Estrogen Receptor Degraders with Highly Improved Antitumor Effect and Favorable Druggability br 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 7, 页码: 5724-5750
作者:  
Lu, Zhengyu;  Cao, Yangzhi;  Zhang, Dan;  Meng, Xin;  Guo, Bin
  |  收藏  |  浏览/下载:26/0  |  提交时间:2022/08/16
Improved Practical Synthesis of DY-038, an Oral Available Antiplatelet Agent 期刊论文  OAI收割
CHEMISTRYSELECT, 2021, 卷号: 6, 期号: 13, 页码: 3183-3186
作者:  
Cao, Yangzhi;  Kong, Deyu;  Sun, Lulu;  Meng, Xin;  Zhang, Yinyong
  |  收藏  |  浏览/下载:48/0  |  提交时间:2021/08/17
Optimization of P2Y(12) Antagonist Ethyl 6-(4-((Benzylsulfonyl)carbarnoyl)piperidin-1-yl)-5-cyano-2-methylnicotinate (AZD1283) Led to the Discovery of an Oral Antiplatelet Agent with Improved Druglike Properties 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 6, 页码: 3088-3106
作者:  
Kong, Deyu;  Xue, Tao;  Guo, Bin;  Cheng, Jianjun;  Liu, Shunyin
  |  收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
Synthesis and biological evaluation of novel potent FFA1 agonists containing 2,3-dihydrobenzo[b][1,4]dioxine 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 848-852
作者:  
  |  收藏  |  浏览/下载:22/0  |  提交时间:2020/07/01
Improved synthesis of YT-14, a potent antibiotic to multidrug-resistant strains 期刊论文  OAI收割
JOURNAL OF CHEMICAL RESEARCH, 2018, 期号: 7, 页码: 354-360
作者:  
Wei, Jianhai;  Kong, Deyu;  Wang, Lei;  Zhang, Yinyong;  Hu, Wenhao
  |  收藏  |  浏览/下载:46/0  |  提交时间:2019/01/08