机构

• 上海药物研究所 [74]

采集方式

• OAI收割 [74]

内容类型

• 期刊论文 [74]

发表日期

• 2024 [1]
• 2023 [2]
• 2022 [3]
• 2021 [4]
• 2019 [5]
• 2018 [4]
• 更多

学科主题

筛选

浏览/检索结果: 共74条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择提交时间升序提交时间降序发表日期升序发表日期降序题名升序题名降序作者升序作者降序 Design, Synthesis, and Anti-tuberculosis Activity of Streptomycin Derivatives 期刊论文  OAI收割 LETTERS IN DRUG DESIGN & DISCOVERY, 2024, 卷号: 21, 期号: 4, 页码: 738-748 作者:  Zhang, Yinyong;  Zhao, Wenhao;  Yang, Yushe;  Zhou, Xianli;  Guo, Bin   |  收藏  |  浏览/下载：6/0  |  提交时间：2024/03/06 Multidrug-resistant  hydrazine  hydrazide  sulfonyl hydrazide  siderophore  synthesis  anti-tuberculosis activity   Discovery of a Novel Bifunctional Steroid Analog, YXG-158, as an Androgen Receptor Degrader and CYP17A1 Inhibitor for the Treatment of Enzalutamide-Resistant Prostate Cancer 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 14, 页码: 9972-9991 作者:  Wang, Ao;  Luo, Xianggang;  Meng, Xin;  Lu, Zhengyu;  Chen, Kaixian   |  收藏  |  浏览/下载：9/0  |  提交时间：2023/10/17 Efficient Kilogram-Scale Synthesis of a Novel Oxazolidinone Antibacterial Candidate YG-056SP 期刊论文  OAI收割 ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2023, 页码: 12 作者:  Zhang, Yinyong;  Yang, Yushe;  Meng, Xin;  Zhou, Xianli;  Guo, Bin   |  收藏  |  浏览/下载：16/0  |  提交时间：2023/04/10 oxazolidinone  asymmetric reduction  fused ring  process development  crystal transformation   Design, Synthesis, and Biological Evaluation of Androgen Receptor Degrading and Antagonizing Bifunctional Steroidal Analogs for the Treatment of Advanced Prostate Cancer 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 22 作者:  Wang, Ao;  Luo, Xianggang;  Wang, Yawan;  Meng, Xin;  Lu, Zhengyu   |  收藏  |  浏览/下载：30/0  |  提交时间：2022/11/11 Design, Synthesis, and Structure-Activity Relationship Studies of Bisamide Derivatives of Amphotericin B with Potent Efficacy and Low Toxicity 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 17 作者:  Ma, Huijun;  Qian, Anran;  Zheng, Yazhou;  Meng, Xin;  Wang, Ting   |  收藏  |  浏览/下载：14/0  |  提交时间：2023/04/10 Discovery of Thieno[2,3-e]indazole Derivatives as Novel Oral Selective Estrogen Receptor Degraders with Highly Improved Antitumor Effect and Favorable Druggability br 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 7, 页码: 5724-5750 作者:  Lu, Zhengyu;  Cao, Yangzhi;  Zhang, Dan;  Meng, Xin;  Guo, Bin   |  收藏  |  浏览/下载：16/0  |  提交时间：2022/08/16 Design, Synthesis, and Biological Evaluation of Novel Pyrimido[4,5-b]indole Derivatives Against Gram-Negative Multidrug-Resistant Pathogens 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8644-8665 作者:  Kong, Qidi;  Pan, Wei;  Xu, Heng;  Xue, Yaru;  Guo, Bin   |  收藏  |  浏览/下载：33/0  |  提交时间：2021/08/17 Improved Practical Synthesis of DY-038, an Oral Available Antiplatelet Agent 期刊论文  OAI收割 CHEMISTRYSELECT, 2021, 卷号: 6, 期号: 13, 页码: 3183-3186 作者:  Cao, Yangzhi;  Kong, Deyu;  Sun, Lulu;  Meng, Xin;  Zhang, Yinyong   |  收藏  |  浏览/下载：29/0  |  提交时间：2021/08/17 antiplatelet agent  cyclization  DY-038  process development  sulfonamides   Recent advances in antibacterial agents 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 35, 页码: 8 作者:  Kong, Qidi;  Yang, Yushe   |  收藏  |  浏览/下载：14/0  |  提交时间：2021/05/24 Antimicrobial resistance  Antibacterial agents  Gram-negative bacteria  Gram-positive bacteria   Design, synthesis and biological evaluation of novel thiohydantoin derivatives as potent androgen receptor antagonists for the treatment of prostate cancer 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 31, 页码: 13 作者:     |  收藏  |  浏览/下载：12/0  |  提交时间：2021/05/24 Androgen receptor  Novel thiohydantoin derivatives  Androgen receptor antagonists  Prostate cancer