中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [80]
生物物理研究所 [2]
大连化学物理研究所 [2]
上海营养与健康研究所 [2]
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OAI收割 [86]
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期刊论文 [85]
会议论文 [1]
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2025 [7]
2024 [8]
2023 [3]
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2021 [4]
2020 [1]
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Immunology [2]
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Novel thieno[2,3-b]pyridine derivatives protect islet through DRAK2 kinase inhibition
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 301, 页码: 18
作者:
Lian, Kaiyue
;
Li, Ruihan
;
Lu, Yuting
;
Song, Gaolei
;
Zhang, Xinwen
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The enedioic acid analog 326E alleviates metabolic dysfunction-associated steatohepatitis via dual targeting at ACLY and PPARα
期刊论文
OAI收割
CELL METABOLISM, 2025, 卷号: 37, 期号: 11, 页码: 2149-2166
作者:
Xie, Zhifu
;
Cheng, Long
;
Hu, Yue
;
Song, Gaolei
;
Wang, Fan
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Mechanism of hydroxamic acid group metabolism to carboxylic acid: Oxidation versus hydrolysis
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2025, 卷号: 53, 期号: 10, 页码: 11
作者:
Huang, Xiyue
;
Zhou, Lei
;
Chen, Huixian
;
Sun, Xiaowei
;
Cao, Mengyi
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Dual Roles of IRE1α Inhibition in Reversing Mitochondrial ROS-Induced CD8+T Cell Senescence and Exerting Direct Anti-Tumor Effects in Multiple Myeloma
期刊论文
OAI收割
CLINICAL LYMPHOMA MYELOMA & LEUKEMIA, 2025, 卷号: 25, 页码: 2
作者:
Wan, Yike
;
Wang, Jingjing
;
Chen, Mengping
;
Wang, Junying
;
Nan, Fajun
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Discovery of Novel Tridentate Alkenyl Diacid Derivatives as Potent ATP Citrate Lyase Inhibitors for the Treatment of Hepatocellular Carcinoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 15, 页码: 15598-15616
作者:
Yang, Yurou
;
Zhai, Jimao
;
Wang, Fan
;
Song, Gaolei
;
Xu, Honghong
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Dual roles of IRE1α inhibition in reversing mitochondrial ROS-induced CD8
+
T-cell senescence and exerting direct antitumor effects in multiple myeloma
期刊论文
OAI收割
JOURNAL FOR IMMUNOTHERAPY OF CANCER, 2025, 卷号: 13, 期号: 5, 页码: 13
作者:
Wan, Yike
;
Wang, Jingjing
;
Chen, Mengping
;
Wang, Junying
;
Nan, Fajun
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Phosphatidylinositol 4,5-bisphosphate activation mechanism of human KCNQ5
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 14, 页码: 11
作者:
Yang, Zhenni
;
Zheng, Yueming
;
Ma, Demin
;
Wang, Long
;
Zhang, Jiatong
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A Phase I Study to Evaluate the Safety, Tolerability, Pharmacokinetics of BGT-002, a Novel ATP-Citrate Lyase Inhibitor, in Healthy Chinese Subjects
期刊论文
OAI收割
DRUG DESIGN DEVELOPMENT AND THERAPY, 2025, 卷号: 19, 页码: 1783-1794
作者:
Liu, Yun
;
Yu, Chengyin
;
Zhang, Yifan
;
Xie, Zhifu
;
Wang, Yating
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Synthesis and Biological Activity of Tetracyclic Dispiro Core Derivatives of Natural Products Dispirocochlearoids A-C
期刊论文
OAI收割
ORGANIC LETTERS, 2024, 卷号: 26, 期号: 45, 页码: 9654-9658
作者:
Pei, Junping
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Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
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