中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共86条,第1-10条 帮助

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Novel thieno[2,3-b]pyridine derivatives protect islet through DRAK2 kinase inhibition 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 301, 页码: 18
作者:  
Lian, Kaiyue;  Li, Ruihan;  Lu, Yuting;  Song, Gaolei;  Zhang, Xinwen
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The enedioic acid analog 326E alleviates metabolic dysfunction-associated steatohepatitis via dual targeting at ACLY and PPARα 期刊论文  OAI收割
CELL METABOLISM, 2025, 卷号: 37, 期号: 11, 页码: 2149-2166
作者:  
Xie, Zhifu;  Cheng, Long;  Hu, Yue;  Song, Gaolei;  Wang, Fan
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Mechanism of hydroxamic acid group metabolism to carboxylic acid: Oxidation versus hydrolysis 期刊论文  OAI收割
DRUG METABOLISM AND DISPOSITION, 2025, 卷号: 53, 期号: 10, 页码: 11
作者:  
Huang, Xiyue;  Zhou, Lei;  Chen, Huixian;  Sun, Xiaowei;  Cao, Mengyi
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Dual Roles of IRE1α Inhibition in Reversing Mitochondrial ROS-Induced CD8+T Cell Senescence and Exerting Direct Anti-Tumor Effects in Multiple Myeloma 期刊论文  OAI收割
CLINICAL LYMPHOMA MYELOMA & LEUKEMIA, 2025, 卷号: 25, 页码: 2
作者:  
Wan, Yike;  Wang, Jingjing;  Chen, Mengping;  Wang, Junying;  Nan, Fajun
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Discovery of Novel Tridentate Alkenyl Diacid Derivatives as Potent ATP Citrate Lyase Inhibitors for the Treatment of Hepatocellular Carcinoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 15, 页码: 15598-15616
作者:  
Yang, Yurou;  Zhai, Jimao;  Wang, Fan;  Song, Gaolei;  Xu, Honghong
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Dual roles of IRE1α inhibition in reversing mitochondrial ROS-induced CD8+ T-cell senescence and exerting direct antitumor effects in multiple myeloma 期刊论文  OAI收割
JOURNAL FOR IMMUNOTHERAPY OF CANCER, 2025, 卷号: 13, 期号: 5, 页码: 13
作者:  
Wan, Yike;  Wang, Jingjing;  Chen, Mengping;  Wang, Junying;  Nan, Fajun
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Phosphatidylinositol 4,5-bisphosphate activation mechanism of human KCNQ5 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 14, 页码: 11
作者:  
Yang, Zhenni;  Zheng, Yueming;  Ma, Demin;  Wang, Long;  Zhang, Jiatong
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A Phase I Study to Evaluate the Safety, Tolerability, Pharmacokinetics of BGT-002, a Novel ATP-Citrate Lyase Inhibitor, in Healthy Chinese Subjects 期刊论文  OAI收割
DRUG DESIGN DEVELOPMENT AND THERAPY, 2025, 卷号: 19, 页码: 1783-1794
作者:  
Liu, Yun;  Yu, Chengyin;  Zhang, Yifan;  Xie, Zhifu;  Wang, Yating
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Synthesis and Biological Activity of Tetracyclic Dispiro Core Derivatives of Natural Products Dispirocochlearoids A-C 期刊论文  OAI收割
ORGANIC LETTERS, 2024, 卷号: 26, 期号: 45, 页码: 9654-9658
作者:  
Pei, Junping
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Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors 期刊论文  OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:  
Cheng, Tingting;  Song, Gaolei;  Cheng, Long;  Wang, Fan;  Sun, Xinyu
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