中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [72]
生物物理研究所 [2]
大连化学物理研究所 [2]
上海营养与健康研究所 [2]
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OAI收割 [78]
内容类型
期刊论文 [77]
会议论文 [1]
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2024 [8]
2023 [3]
2022 [6]
2021 [4]
2020 [1]
2019 [1]
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Immunology [2]
Cell Biolo... [1]
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浏览/检索结果:
共78条,第1-10条
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Synthesis and Biological Activity of Tetracyclic Dispiro Core Derivatives of Natural Products Dispirocochlearoids A-C
期刊论文
OAI收割
ORGANIC LETTERS, 2024, 卷号: 26, 期号: 45, 页码: 9654-9658
作者:
Pei, Junping
;
Wang, Ying
;
Shi, Shengjie
;
Chen, Linhai
;
Yin, Jianpeng
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/12/11
Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/02/28
metabolic diseases
ATP-citrate lyase (ACLY)
lipogenesis
ACLY inhibitors
dienyldicarboxylic acid
A brain-to-gut signal controls intestinal fat absorption
期刊论文
OAI收割
NATURE, 2024, 页码: 27
作者:
Lyu, Qianqian
;
Xue, Wenzhi
;
Liu, Ruixin
;
Ma, Qinyun
;
Kasaragod, Vikram Babu
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/11/26
Discovery of GPR84 Fluorogenic Probes Based on a Novel Antagonist for GPR84 Bioimaging
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 16
作者:
Xiao, Yufeng
;
Chen, Jing
;
Li, Shaoxian
;
Zhang, Qing
;
Liu, Yin
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/08/22
Simultaneous determination of BGT-002 and its acyl glucuronide metabolite ZM326E-M2 in human plasma by liquid chromatography-tandem mass spectrometry and its application to a pharmacokinetic study
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2024, 卷号: 243, 页码: 8
作者:
Zhu, Xueran
;
Cui, Shumin
;
Liu, Xinjing
;
Zhang, Mei
;
Xie, Zhifu
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/05/31
ATP-Citrate Lyase
BGT-002
Acyl glucuronide metabolite
Pseudo-MRM
LC-MS/MS
Pharmacokinetics
Polyphenol Compound 18a Modulates UCP1-Dependent Thermogenesis to Counteract Obesity
期刊论文
OAI收割
BIOMOLECULES, 2024, 卷号: 14, 期号: 6, 页码: 21
作者:
Wen, Xueping
;
Song, Yufei
;
Zhang, Mei
;
Kang, Yiping
;
Chen, Dandan
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/08/22
18a
adipocytes
polyphenols
thermogenesis
UCP1
Discovery of betulinic acid derivatives as gut-restricted TGR5 agonists: Balancing the potency and physicochemical properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 144, 页码: 18
作者:
Zhuo, Ning
;
Yun, Ying
;
Zhang, Chenlu
;
Guo, Shimeng
;
Yin, Jianpeng
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2024/03/25
Type 2 Diabetes
TGR5 agonist
Betulinic acid
Gut-restricted
Gallbladder-filling effects
Kinetophores
Design, Synthesis, and Structure-Activity Relationship of Novel Potent and Highly Selective Cysteinyl Leukotriene Receptor 1 (CysLT1R) Antagonists
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 1, 页码: 259-276
作者:
Wang Jingyi
;
Liu Jinyu
;
Chen Dongsheng
;
Chen Huayan
;
Xie Xin
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收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/05/07
cysteinyl leukotriene
cysteinyl leukotriene receptor 1 (CysLT1R)
selective antagonists
Design and Synthesis Studies of α-Methylene-γ-butyrolactones Antagonists of GPR52
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2023, 卷号: 43, 期号: 11, 页码: 3916-3929
作者:
Shen, Donghang
;
Li, Xin
;
Guo, Shimeng
;
Xie, Xin
;
Nan, Fajun
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/02/27
Huntingdon's disease
G protein-coupled receptor
GPR52
alpha-methylene-gamma-butyrolactones
antagonist
Ligand activation mechanisms of human KCNQ2 channel
期刊论文
OAI收割
Nature communications, 2023, 卷号: 14, 期号: 1, 页码: 6632
作者:
Ma, Demin
;
Zheng, Yueming
;
Li, Xiaoxiao
;
Zhou, Xiaoyu
;
Yang, Zhenni
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2024/03/26