中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共175条,第1-10条 帮助

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Heterocycle-fused phenylcyclohexylamines as novel multi-target antagonists of N-methyl-D-aspartate (NMDA) receptor and monoamine transporter for treating depression 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 291, 页码: 20
作者:  
Zheng, Fuqiang;  Hu, Zhengtao;  Chen, Hai;  Cheng, Jiaxin;  Hou, Qiongqiong
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Design and Development of a Novel Oral 4′-Fluorouridine Double Prodrug VV261 against SFTSV 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 9, 页码: 9811-9826
作者:  
Cheng, Yong;  Zheng, Wei;  Dong, Xinru;  Sun, Tengxiao;  Xu, Mengwei
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Design, Synthesis, and Biological Evaluation of Peptidomimetic Tetrahydropyrrole Spirodihydroindolones as SARS-CoV-2 3CL Protease Inhibitors 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 16, 期号: 5, 页码: 790-796
作者:  
Hu, Liuyan;  Zhao, Zhi;  Zhang, Shujing;  Yang, Lei;  Cui, Wenjie
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Structural Similarity in Natural Products Leading to Sample Misidentification: A Case Study of the Bisbenzylisoquinoline Alkaloids Oxyacanthine and Berbamine 期刊论文  OAI收割
JOURNAL OF NATURAL PRODUCTS, 2025, 卷号: 88, 期号: 1, 页码: 191-198
作者:  
Cheng, Yan;  Akramov, Davlat;  Yakhshilikova, Lola;  Zhu, Chengwei;  Lu, Jie
  |  收藏  |  浏览/下载:17/0  |  提交时间:2025/04/01
Discovery of peptidomimetic spiropyrrolidine derivatives as novel 3CLpro inhibitors against SARS-CoV-2 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 281, 页码: 22
作者:  
Guma, Samuel Desta;  Zhou, Zhaoyin;  Song, Kang;  Yang, Feipu;  Suo, Jin
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/12/11
F-CPI: A Multimodal Deep Learning Approach for Predicting Compound Bioactivity Changes Induced by Fluorine Substitution 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 13
作者:  
Zhang, Qian;  Yin, Wenhai;  Chen, Xinyao;  Zhou, Aimin;  Zhang, Guixu
  |  收藏  |  浏览/下载:14/0  |  提交时间:2025/02/28
Direct Reductive N-alkylation of Amines with Carboxylic Esters 期刊论文  OAI收割
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2024, 页码: 7
作者:  
Zhang, Yuxuan;  Bonku, Emmanuel Mintah;  Yang, Xingbang;  Zhu, Fuqiang;  Jiang, Xiangrui
  |  收藏  |  浏览/下载:14/0  |  提交时间:2025/01/14
Design, synthesis, and evaluation of novel oxyacanthine derivatives for anti-SARS-CoV-2 activity 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 113, 页码: 5
作者:  
Lu, Jie;  Cheng, Yan;  Zhang, Yumin;  Wang, Yi;  Xia, Bingqing
  |  收藏  |  浏览/下载:9/0  |  提交时间:2025/02/28
Discovery of the potent covalent inhibitor with an acrylate warhead for SARS-CoV-2 3CL protease 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 112, 页码: 5
作者:  
Shen, Wen;  Chen, Xinyao;  Zhou, Liping;  Cheng, Yan;  Zhang, Yan
  |  收藏  |  浏览/下载:26/0  |  提交时间:2024/10/21
Iron-Catalyzed Cross-Coupling Reactions of Alkyl Grignard Reagents with Alkenyl Carbonate 期刊论文  OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2024, 页码: 8
作者:  
Qin, Hongjian;  Yang, Xingbang;  Mintah Bonku, Emmanuel;  Zhu, Fuqiang;  Abduahadi, Safomuddin
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/12/11