中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [20]
地理科学与资源研究所 [5]
西安光学精密机械研究... [2]
中国科学院大学 [1]
地球化学研究所 [1]
生态环境研究中心 [1]
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期刊论文 [27]
专利 [2]
会议论文 [1]
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2025 [2]
2024 [5]
2023 [3]
2022 [2]
2020 [4]
2019 [2]
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题名升序
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(+)-Borneol Enhances the Antiseizure Effects of Retigabine by both Pharmacokinetic and Pharmacodynamic Interaction
期刊论文
OAI收割
NEUROCHEMICAL RESEARCH, 2025, 卷号: 50, 期号: 3, 页码: 13
作者:
Xu, Haiyan
;
Wu, Zhidan
;
Wang, Pei
;
Gong, Jili
;
Qiu, Li
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/06/23
Epilepsy
Retigabine
(+)-Borneol
Synergistic interaction
KCNQ channels
Electrophysiological Abnormalities and Pharmacological Corrections of Pathogenic Missense Variants in KCNQ3
期刊论文
OAI收割
NEUROSCIENCE BULLETIN, 2025, 页码: 11
作者:
Wu, Xiaorong
;
Gong, Jili
;
Qiu, Li
;
Yang, Guimei
;
Yuan, Hui
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/05/27
KCNQ3
Self-limited familial neonatal epilepsy
Neurodevelopmental disorder
Pynegabine
Amitriptyline
Electrophysiology
A novel isoquinoline alkaloid HJ-69 isolated from Zanthoxylum bungeanum attenuates inflammatory pain by inhibiting voltage-gated sodium and potassium channels
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2024, 卷号: 330, 页码: 12
作者:
Wang, Long
;
Hao, Haishuang
;
Meng, Xianhua
;
Zhang, Wenbo
;
Zhang, Yin
  |  
收藏
  |  
浏览/下载:120/0
  |  
提交时间:2024/11/05
HJ-69
Zanthoxylum bungeanum
Isoquinoline alkaloid
Nav
Kv
Inflammatory pain
Discovery of Novel Pyrimidine-Based Derivatives as Nav1.2 Inhibitors with Efficacy in Mouse Models of Epilepsy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15, 页码: 12912-12931
作者:
He, Guoxue
;
Zheng, Yueming
;
Chang, Shunzhen
;
Wang, Long
;
Yang, Xiaohao
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/09/26
Direct Identification of Complex Glycans via a Highly Sensitive Engineered Nanopore
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2024, 页码: 11
作者:
Yao, Guangda
;
Tian, Yinping
;
Ke, Wenjun
;
Fang, Jie
;
Ma, Shengzhou
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/05/22
Pharmacological inhibition of Kir4.1 evokes rapid-onset antidepressant responses
期刊论文
OAI收割
NATURE CHEMICAL BIOLOGY, 2024, 页码: 29
作者:
Zhou, Xiaoyu
;
Zhao, Cheng
;
Xu, Haiyan
;
Xu, Yixiang
;
Zhan, Li
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2024/03/25
An LQT2-related mutation in the voltage-sensing domain is involved in switching the gating polarity of hERG
期刊论文
OAI收割
BMC BIOLOGY, 2024, 卷号: 22, 期号: 1, 页码: 14
作者:
Liu, Zhipei
;
Wang, Feng
;
Yuan, Hui
;
Tian, Fuyun
;
Yang, Chuanyan
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2024/03/13
hERG
K525N
Gating Polarity
Voltage-Sensing Domain
LQT2
Discovery of selective NaV1.8 inhibitors based on 5-chloro-2-(4,4-difluor- oazepan-1-yl)-6-methyl nicotinamide scaffold for the treatment of pain
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 254, 页码: 12
作者:
Qin, Hui
;
Wei, Aihuan
;
Wang, Yunqi
;
Wang, Linlin
;
Xu, Haiyan
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2023/10/17
Pain
Non-addictive analgesics
Na V 1
8-selective inhibitors
Bicyclic aromatic groups
Design, Synthesis and Bioactivity of [3.3.3]Propellane-Based Voltage-Gated Calcium Channel alpha 2 delta Subunit Ligands
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2023, 卷号: 43, 期号: 6, 页码: 2226-2238
作者:
He Jinyan
;
Tian Fuyun
;
Wu Qingqing
;
Zheng Yueming
;
Chen Yuting
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2023/10/17
propellane
voltage-gated calcium channel
alpha 2 delta subunit
synthesis
bioactivity
structure-activity relationship
Characterization of the role of TMEM175 in an in vitro lysosomal H+ fluxes model
期刊论文
OAI收割
FEBS JOURNAL, 2023, 页码: 19
作者:
Yang, Chuanyan
;
Tian, Fuyun
;
Hu, Mei
;
Kang, Chunlan
;
Ping, Meixuan
  |  
收藏
  |  
浏览/下载:74/0
  |  
提交时间:2023/10/17
glycocalyx
H+ leak
lysosome acidification
proton channel
TMEM175