中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共81条,第1-10条 帮助

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Discovery of Novel 2-Aminopyridine-Based and 2-Aminopyrimidine-Based Derivatives as Potent CDK/HDAC Dual Inhibitors for the Treatment of Refractory Solid Tumors and Hematological Malignancies 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 17, 页码: 15220-15245
作者:  
Saidahmatov, Abdusaid;  Li, Jianan;  Xu, Shihao;  Hu, Xiaobei;  Gao, Xiangqian
  |  收藏  |  浏览/下载:20/0  |  提交时间:2024/10/21
Discovery of a Highly Potent, Selective and Efficacious USP7 Degrader for the Treatment of Acute Lymphoblastic Leukemia 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 20
作者:  
Xu, Miaomiao;  Fu, Jingfeng;  Pei, Yuan;  Li, Mengna;  Kan, Weijuan
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/08/22
Discovery of 5-trifluoromethyl-2-aminopyrimidine derivatives as potent dual inhibitors of FLT3 and CHK1 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:  
Deng, Minjie;  Gao, Yue;  Wang, Peipei;  Du, Wenjing;  Xu, Gaoya
  |  收藏  |  浏览/下载:25/0  |  提交时间:2024/02/19
Discovery of 2-Aminopyrimidine Derivatives as Potent Dual FLT3/CHK1 Inhibitors with Significantly Reduced hERG Inhibitory Activities 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:  
Li, Xuemei;  Wang, Peipei;  Wang, Chang;  Jin, Tingting;  Xu, Ran
  |  收藏  |  浏览/下载:24/0  |  提交时间:2023/10/17
Preventive and therapeutic benefits of nelfinavir in rhesus macaques and human beings infected with SARS-CoV-2 期刊论文  OAI收割
Signal Transduction and Targeted Therapy, 2023, 卷号: 8, 期号: 5, 页码: 2384-2391
作者:  
Xu, Zhijian;  Shi, Danrong;  Han, Jianbao;  Ling, Yun;  Jiang, Xiangrui
  |  收藏  |  浏览/下载:39/0  |  提交时间:2024/03/27
Design, Synthesis, and Biological Evaluation of 2-Aminothiazole Derivatives as Novel Checkpoint Kinase 1 (CHK1) Inhibitors 期刊论文  OAI收割
CHEMMEDCHEM, 2023, 页码: 19
作者:  
Deng, Minjie;  Wang, Peipei;  Long, Xiubing;  Xu, Gaoya;  Wang, Chang
  |  收藏  |  浏览/下载:21/0  |  提交时间:2023/04/10
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors 期刊论文  OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:  
Zang, Yi;  Su, Mingbo;  Wang, Qingxing;  Cheng, Xi;  Zhang, Wenru
  |  收藏  |  浏览/下载:23/0  |  提交时间:2024/03/27
The genomic characteristics and pathogenicity of a mammalian orthoreovirus within a new lineage from wild pika in plateau 期刊论文  OAI收割
VIROLOGICA SINICA, 2023, 卷号: 38, 期号: 6
作者:  
Zong, Kexin;  Guo, Yuanyuan;  Song, Jingdong;  Liu, Maoshun;  Hao, Junfeng
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/11/27
Grassland changes and adaptive management on the Qinghai-Tibetan Plateau 期刊论文  OAI收割
NATURE REVIEWS EARTH & ENVIRONMENT, 2022, 页码: 16
作者:  
Wang, Yanfen;  Lv, Wangwang;  Xue, Kai;  Wang, Shiping;  Zhang, Lirong
  |  收藏  |  浏览/下载:48/0  |  提交时间:2022/09/26
Grassland changes and adaptive management on the Qinghai-Tibetan Plateau 期刊论文  OAI收割
NATURE REVIEWS EARTH & ENVIRONMENT, 2022, 卷号: 3, 期号: 10, 页码: 668-683
作者:  
Wang, Yanfen;  Lv, Wangwang;  Xue, Kai;  Wang, Shiping;  Zhang, Lirong
  |  收藏  |  浏览/下载:46/0  |  提交时间:2022/09/26