中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [16]
上海光学精密机械研... [12]
近代物理研究所 [9]
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OAI收割 [81]
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期刊论文 [74]
会议论文 [7]
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2024 [2]
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Plant Scie... [2]
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Discovery of Novel 2-Aminopyridine-Based and 2-Aminopyrimidine-Based Derivatives as Potent CDK/HDAC Dual Inhibitors for the Treatment of Refractory Solid Tumors and Hematological Malignancies
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 17, 页码: 15220-15245
作者:
Saidahmatov, Abdusaid
;
Li, Jianan
;
Xu, Shihao
;
Hu, Xiaobei
;
Gao, Xiangqian
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/10/21
Discovery of a Highly Potent, Selective and Efficacious USP7 Degrader for the Treatment of Acute Lymphoblastic Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 20
作者:
Xu, Miaomiao
;
Fu, Jingfeng
;
Pei, Yuan
;
Li, Mengna
;
Kan, Weijuan
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/08/22
Discovery of 5-trifluoromethyl-2-aminopyrimidine derivatives as potent dual inhibitors of FLT3 and CHK1
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:
Deng, Minjie
;
Gao, Yue
;
Wang, Peipei
;
Du, Wenjing
;
Xu, Gaoya
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2024/02/19
Discovery of 2-Aminopyrimidine Derivatives as Potent Dual FLT3/CHK1 Inhibitors with Significantly Reduced hERG Inhibitory Activities
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:
Li, Xuemei
;
Wang, Peipei
;
Wang, Chang
;
Jin, Tingting
;
Xu, Ran
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/10/17
Preventive and therapeutic benefits of nelfinavir in rhesus macaques and human beings infected with SARS-CoV-2
期刊论文
OAI收割
Signal Transduction and Targeted Therapy, 2023, 卷号: 8, 期号: 5, 页码: 2384-2391
作者:
Xu, Zhijian
;
Shi, Danrong
;
Han, Jianbao
;
Ling, Yun
;
Jiang, Xiangrui
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2024/03/27
Design, Synthesis, and Biological Evaluation of 2-Aminothiazole Derivatives as Novel Checkpoint Kinase 1 (CHK1) Inhibitors
期刊论文
OAI收割
CHEMMEDCHEM, 2023, 页码: 19
作者:
Deng, Minjie
;
Wang, Peipei
;
Long, Xiubing
;
Xu, Gaoya
;
Wang, Chang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/04/10
2-aminothiazole
CHK1 inhibitors
antiproliferation
hematologic malignancies
biological activity
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors
期刊论文
OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:
Zang, Yi
;
Su, Mingbo
;
Wang, Qingxing
;
Cheng, Xi
;
Zhang, Wenru
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/03/27
high-throughput screening
SARS
CoV-2
main
papain-like
proteases
The genomic characteristics and pathogenicity of a mammalian orthoreovirus within a new lineage from wild pika in plateau
期刊论文
OAI收割
VIROLOGICA SINICA, 2023, 卷号: 38, 期号: 6
作者:
Zong, Kexin
;
Guo, Yuanyuan
;
Song, Jingdong
;
Liu, Maoshun
;
Hao, Junfeng
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/11/27
Grassland changes and adaptive management on the Qinghai-Tibetan Plateau
期刊论文
OAI收割
NATURE REVIEWS EARTH & ENVIRONMENT, 2022, 页码: 16
作者:
Wang, Yanfen
;
Lv, Wangwang
;
Xue, Kai
;
Wang, Shiping
;
Zhang, Lirong
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2022/09/26
Grassland changes and adaptive management on the Qinghai-Tibetan Plateau
期刊论文
OAI收割
NATURE REVIEWS EARTH & ENVIRONMENT, 2022, 卷号: 3, 期号: 10, 页码: 668-683
作者:
Wang, Yanfen
;
Lv, Wangwang
;
Xue, Kai
;
Wang, Shiping
;
Zhang, Lirong
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2022/09/26