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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [54]
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西北高原生物研究所 [7]
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期刊论文 [94]
会议论文 [1]
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Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:
Wu, Xinyuan
;
Li, Shunyao
;
Liang, Ting
;
Yu, Qing
;
Zhang, Yiwei
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/06/23
Activity-based protein profiling data
Covalent DNA-encoded chemical library
Covalent ligand selection
Lysine-targeting covalent inhibitors
IHCH9033, a novel class I HDAC inhibitor, synergizes with FLT3 inhibitor and rescues quizartinib resistance in FLT3-ITD AML via enhancing DNA damage response
期刊论文
OAI收割
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2025, 卷号: 14, 期号: 1, 页码: 19
作者:
Yao, Mingyue
;
Yan, Wenzhong
;
Wang, Yafang
;
Zhao, Yu
;
Xu, Xiaowei
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2025/04/01
Acute myeloid leukemia
HDAC inhibitor
FLT3-ITD mutation
DNA damage response
Synergistic effect
Drug resistance
Harnessing the Magic Methyl Effect: Discovery of CLPP-2068 as a Novel
Hs
ClpP Activator for the Treatment of Diffuse Large B-Cell Lymphoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 4, 页码: 4287-4307
作者:
Sun, Mingyang
;
Chen, Beijing
;
Teng, Dan
;
Zhao, Hongshen
;
Liao, Yilie
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2025/04/01
Prediction of Solvate Based on Graph Attention Network
期刊论文
OAI收割
CRYSTAL GROWTH & DESIGN, 2025, 卷号: 25, 期号: 2, 页码: 297-308
作者:
Sun, Shihui
;
Wang, Jian-Rong
;
Tang, Lei
;
Fan, Zhehuan
;
Li, Xutong
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2025/04/01
Age-related decline in CD8
+
tissue resident memory T cells compromises antitumor immunity
期刊论文
OAI收割
NATURE AGING, 2024, 卷号: 4, 期号: 12, 页码: 1828-+
作者:
Pei, Siyu
;
Deng, Xiuyu
;
Yang, Ruirui
;
Wang, Hui
;
Shi, Jian-Hong
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2025/02/28
SurfDock is a surface-informed diffusion generative model for reliable and accurate protein-ligand complex prediction
期刊论文
OAI收割
NATURE METHODS, 2024, 页码: 24
作者:
Cao, Duanhua
;
Chen, Mingan
;
Zhang, Runze
;
Wang, Zhaokun
;
Huang, Manlin
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2025/01/06
Prediction of Multi-Pharmacokinetics Property in Multi-Species: Bayesian Neural Network Stacking Model with Uncertainty
期刊论文
OAI收割
MOLECULAR PHARMACEUTICS, 2024, 页码: 16
作者:
Zhang, Yuanyuan
;
Xie, Zhiyin
;
Xiao, Fu
;
Yu, Jie
;
Fan, Zhehuan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/12/11
pharmacokinetic parameters
machine learning
uncertainty
stacking
multitask learning
ADME
Asymmetric macrocyclization enabled by Rh(III)-catalyzed C-H activation: Enantioenriched macrocyclic inhibitor of Zika virus infection
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2024, 卷号: 35, 期号: 11, 页码: 6
作者:
Chen, Chao
;
Yu, Wenwen
;
Huang, Guangen
;
Ren, Xuelian
;
Chen, Xiangli
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/09/26
C -H activation
Carboamidation
Enantioselective macrocyclization
Anti-Zika virus activity
Unraveling the CDK9/PP2A/ERK Network in Transcriptional Pause Release and Complement Activation in KRAS-mutant Cancers
期刊论文
OAI收割
ADVANCED SCIENCE, 2024, 页码: 20
作者:
Wang, Yafang
;
Xu, Lansong
;
Ling, Lijun
;
Yao, Mingyue
;
Shi, Shangxuan
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2024/10/21
KRAS
CDK9
ERK
complement activation
immunosuppression
Reducing overconfident errors in molecular property classification using Posterior Network
期刊论文
OAI收割
PATTERNS, 2024, 卷号: 5, 期号: 6, 页码: 100991
作者:
Fan, Zhehuan
;
Yu, Jie
;
Zhang, Xiang
;
Chen, Yijie
;
Sun, Shihui
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/06/04