中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共19条,第1-10条 帮助

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Discovery of a potent and orally bioavailable 3,3-dimethyl-2-oxoindoline STING inhibitor 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 301, 页码: 18
作者:  
Li, Wenxin;  Wang, Xiyuan;  Zang, Shumin;  Zhou, Rongyao;  Zhou, Hongfei
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Discovery of isoindoline-2(1H)-carboxamide STING inhibitors as anti-inflammatory agents 期刊论文  OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 13
作者:  
Zhou, Xiaoqian;  Zang, Shumin;  Yao, Shanyan;  Zhou, Hongfei;  Wang, Xiyuan
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Discovery of 3,4-dihydroisoquinoline-2(1H)-carboxamide STING inhibitors as anti-inflammatory agents 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 297, 页码: 20
作者:  
Zhou, Xiaoqian;  Yue, Hangtian;  Wang, Xiyuan;  Zang, Shumin;  Li, Han
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Dual targeting of VEGFR2 and CSF1R with SYHA1813 confers novel strategy for treating both BRAF wild-type and mutant melanoma 期刊论文  OAI收割
CANCER CELL INTERNATIONAL, 2025, 卷号: 25, 期号: 1, 页码: 12
作者:  
Shi, Wenhao;  Tang, Haotian;  Tong, Linjiang;  Song, Peiran;  Huang, Yuqing
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Discovery of a non-nucleotide stimulator of interferon genes (STING) agonist with systemic antitumor effect 期刊论文  OAI收割
MEDCOMM, 2025, 卷号: 6, 期号: 1, 页码: e70001
作者:  
Wang, Xiyuan;  Zhan, Zhengsheng;  Wang, Zhen;  Zhang, Yan;  Zhao, Kaiyan
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A Novel IRAK4 Inhibitor DW18134 Ameliorates Peritonitis and Inflammatory Bowel Disease 期刊论文  OAI收割
MOLECULES, 2024, 卷号: 29, 期号: 8, 页码: 17
作者:  
Huang, Yuqing;  Ning, Yi;  Chen, Zhiwei;  Song, Peiran;  Tang, Haotian
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Preclinical and early clinical studies of a novel compound SYHA1813 that efficiently crosses the blood-brain barrier and exhibits potent activity against glioblastoma 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4748-4764
作者:  
Liu, Yingqiang;  Zhan, Zhengsheng;  Kang, Zhuang
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Design, synthesis, and STING-agonistic activity of benzo[b]thiophene-2-carboxamide derivatives 期刊论文  OAI收割
MOLECULAR DIVERSITY, 2023, 页码: 10
作者:  
Zhou, Rongyao;  Wang, Xiyuan;  Zhang, Deqiang;  Zhan, Zhengsheng;  Duan, Wenhu
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Design, Synthesis and Bioactivity of [3.3.3]Propellane-Based Voltage-Gated Calcium Channel alpha 2 delta Subunit Ligands 期刊论文  OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2023, 卷号: 43, 期号: 6, 页码: 2226-2238
作者:  
He Jinyan;  Tian Fuyun;  Wu Qingqing;  Zheng Yueming;  Chen Yuting
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Discovery of 10H-Benzo[b]pyrido[2,3-e][1,4]oxazine AXL Inhibitors via Structure-Based Drug Design Targeting c-Met Kinase 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:  
Zhan, Zhengsheng;  Ji, Yinchun;  Su, Haixia;  Fang, Chen;  Peng, Xia
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