中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [19]
采集方式
OAI收割 [19]
内容类型
期刊论文 [18]
会议论文 [1]
发表日期
2026 [1]
2025 [4]
2024 [1]
2023 [3]
2022 [2]
2021 [1]
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学科主题
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浏览/检索结果:
共19条,第1-10条
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Discovery of a potent and orally bioavailable 3,3-dimethyl-2-oxoindoline STING inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 301, 页码: 18
作者:
Li, Wenxin
;
Wang, Xiyuan
;
Zang, Shumin
;
Zhou, Rongyao
;
Zhou, Hongfei
  |  
收藏
  |  
Discovery of isoindoline-2(1
H
)-carboxamide STING inhibitors as anti-inflammatory agents
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 13
作者:
Zhou, Xiaoqian
;
Zang, Shumin
;
Yao, Shanyan
;
Zhou, Hongfei
;
Wang, Xiyuan
  |  
收藏
  |  
Discovery of 3,4-dihydroisoquinoline-2(1H)-carboxamide STING inhibitors as anti-inflammatory agents
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 297, 页码: 20
作者:
Zhou, Xiaoqian
;
Yue, Hangtian
;
Wang, Xiyuan
;
Zang, Shumin
;
Li, Han
  |  
收藏
  |  
Dual targeting of VEGFR2 and CSF1R with SYHA1813 confers novel strategy for treating both BRAF wild-type and mutant melanoma
期刊论文
OAI收割
CANCER CELL INTERNATIONAL, 2025, 卷号: 25, 期号: 1, 页码: 12
作者:
Shi, Wenhao
;
Tang, Haotian
;
Tong, Linjiang
;
Song, Peiran
;
Huang, Yuqing
  |  
收藏
  |  
Discovery of a non-nucleotide stimulator of interferon genes (STING) agonist with systemic antitumor effect
期刊论文
OAI收割
MEDCOMM, 2025, 卷号: 6, 期号: 1, 页码: e70001
作者:
Wang, Xiyuan
;
Zhan, Zhengsheng
;
Wang, Zhen
;
Zhang, Yan
;
Zhao, Kaiyan
  |  
收藏
  |  
A Novel IRAK4 Inhibitor DW18134 Ameliorates Peritonitis and Inflammatory Bowel Disease
期刊论文
OAI收割
MOLECULES, 2024, 卷号: 29, 期号: 8, 页码: 17
作者:
Huang, Yuqing
;
Ning, Yi
;
Chen, Zhiwei
;
Song, Peiran
;
Tang, Haotian
  |  
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  |  
Preclinical and early clinical studies of a novel compound SYHA1813 that efficiently crosses the blood-brain barrier and exhibits potent activity against glioblastoma
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4748-4764
作者:
Liu, Yingqiang
;
Zhan, Zhengsheng
;
Kang, Zhuang
  |  
收藏
  |  
Design, synthesis, and STING-agonistic activity of benzo[
b
]thiophene-2-carboxamide derivatives
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2023, 页码: 10
作者:
Zhou, Rongyao
;
Wang, Xiyuan
;
Zhang, Deqiang
;
Zhan, Zhengsheng
;
Duan, Wenhu
  |  
收藏
  |  
Design, Synthesis and Bioactivity of [3.3.3]Propellane-Based Voltage-Gated Calcium Channel alpha 2 delta Subunit Ligands
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2023, 卷号: 43, 期号: 6, 页码: 2226-2238
作者:
He Jinyan
;
Tian Fuyun
;
Wu Qingqing
;
Zheng Yueming
;
Chen Yuting
  |  
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  |  
Discovery of 10H-Benzo[b]pyrido[2,3-e][1,4]oxazine AXL Inhibitors via Structure-Based Drug Design Targeting c-Met Kinase
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:
Zhan, Zhengsheng
;
Ji, Yinchun
;
Su, Haixia
;
Fang, Chen
;
Peng, Xia
  |  
收藏
  |