中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Design, Synthesis, and Pharmacological Evaluation of Quinazoline and Quinoline Derivatives as Potent ENPP1 Inhibitors for Cancer Immunotherapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 18
作者:  
He, Jie;  Ma, Xiaoyu;  Sun, Jia;  Chen, Manman;  Xu, Lan
  |  收藏  |  浏览/下载:8/0  |  提交时间:2025/04/01
Discovery of Urea Derivatives of Celastrol as Selective Peroxiredoxin 1 Inhibitors against Colorectal Cancer Cells 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 9, 页码: 7176-7196
作者:  
Li, Yang;  Zhu, Yuyuan;  Shang, Fan-Fan;  Xu, Lin;  Jiang, Defang
  |  收藏  |  浏览/下载:33/0  |  提交时间:2024/06/27
Design, Synthesis, and Pharmacological Evaluation of Spiro[carbazole-3,3′-pyrrolidine] Derivatives as cGAS Inhibitors for Treatment of Acute Lung Injury 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 24
作者:  
Chen, Mingjie;  Lei, Shuyue;  Zhou, Zihua;  Wang, Meng;  Feng, Chunlan
  |  收藏  |  浏览/下载:35/0  |  提交时间:2024/05/22
Design, Synthesis, and Pharmacological Evaluation of Isoindoline Analogues as New HPK1 Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 23, 页码: 16201-16221
作者:  
  |  收藏  |  浏览/下载:35/0  |  提交时间:2024/02/27
Photochemically controlled activation of STING by CAIX-targeting photocaged agonists to suppress tumor cell growth 期刊论文  OAI收割
CHEMICAL SCIENCE, 2023, 卷号: 14, 期号: 22, 页码: 5956-5964
作者:  
Ding, Chunyong;  Du, Mengyan;  Xiong, Zhi;  Wang, Xue;  Li, Hongji
  |  收藏  |  浏览/下载:39/0  |  提交时间:2023/10/17
Celastrol suppresses colorectal cancer via covalent targeting peroxiredoxin 1 期刊论文  OAI收割
Signal Transduction and Targeted Therapy, 2023, 卷号: 8, 期号: 3, 页码: 1159-1174
作者:  
Xu, Heng;  Zhao, Hongfang;  Ding, Chunyong;  Jiang, Defang;  Zhao, Zijie
  |  收藏  |  浏览/下载:29/0  |  提交时间:2024/03/27
Acid-Ionizable Iron Nanoadjuvant Augments STING Activation for Personalized Vaccination Immunotherapy of Cancer 期刊论文  OAI收割
ADVANCED MATERIALS, 2023, 页码: 15
作者:  
Chen, Fangmin;  Li, Tianliang;  Zhang, Huijuan;  Saeed, Madiha;  Liu, Xiaoying
  |  收藏  |  浏览/下载:46/0  |  提交时间:2023/04/10
Structure-Activity relationship study of benzothiophene oxobutanoic acid analogues leading to novel stimulator of interferon gene (STING) agonists 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 241, 页码: 16
作者:  
Shen, Ancheng;  Li, Xiyuan;  Zhang, Yan;  Ma, Jing;  Xiao, Ruoxuan
  |  收藏  |  浏览/下载:30/0  |  提交时间:2023/04/10
Design, synthesis and pharmacological evaluation of new PARP1 inhibitors by merging pharmacophores of olaparib and the natural product alantolactone 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 240, 页码: 114574
作者:  
Kayumov, Muzaffar;  Jia, Li;  Pardaev, Azizbek;  Song, Shan-Shan;  Mirzaakhmedov, Sharafitdin
  |  收藏  |  浏览/下载:35/0  |  提交时间:2024/03/21
Synthesis and pharmacological validation of fluorescent diarylsulfonylurea analogues as NLRP3 inhibitors and imaging probes 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 237, 页码: 13
作者:  
Zhao, Jiannan;  Li, Yongling;  Ma, Jing;  Liu, Jingting;  Xiao, Ruoxuan
  |  收藏  |  浏览/下载:105/0  |  提交时间:2022/08/16
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