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Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共294条,第1-10条 帮助

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Discovery of novel antimyeloma agents targeting TRIP13 by molecular modeling and bioassay 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2025, 页码: 14
作者:  
Bunu, Samuel Jacob;  Cai, Haiyan;  Zhou, Zhaoyin;  Zhang, Yanlei;  Lai, Yue
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Design, Synthesis, and Biological Evaluation of Peptidomimetic Tetrahydropyrrole Spirodihydroindolones as SARS-CoV-2 3CL Protease Inhibitors 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 16, 期号: 5, 页码: 790-796
作者:  
Hu, Liuyan;  Zhao, Zhi;  Zhang, Shujing;  Yang, Lei;  Cui, Wenjie
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Development of RelB-targeting small-molecule inhibitors of non-canonical NF-kB signaling with antitumor efficacy 期刊论文  OAI收割
MOLECULAR THERAPY, 2025, 卷号: 33, 期号: 4, 页码: 1519-1534
作者:  
Li, Cuifeng;  Wei, Shuqi;  Sun, Donglin;  Yang, Zhuo;  Wang, Qi
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/05/27
REG3A secreted by peritumoral acinar cells enhances pancreatic ductal adenocarcinoma progression via activation of EGFR signaling 期刊论文  OAI收割
CELL COMMUNICATION AND SIGNALING, 2025, 卷号: 23, 期号: 1, 页码: 19
作者:  
Ren, Xiaojing;  Teng, Yunfei;  Xie, Kunxin;  He, Xiao;  Chen, Gang
  |  收藏  |  浏览/下载:18/0  |  提交时间:2025/04/01
Novel conjugated 5-alkenyl rhodanine tethered 1,4-benzodioxane derivatives as dual-chitinases inhibitors to hinder the growth of Asian corn borer 期刊论文  OAI收割
MEDICINAL CHEMISTRY RESEARCH, 2025, 页码: 13
作者:  
Chen, Jinxiu;  Shi, Dongmei;  Jiang, Zhiyang;  Zou, Renxuan;  Zhang, Jingyu
  |  收藏  |  浏览/下载:7/0  |  提交时间:2025/04/01
Exploratory research on the effective chemical basis of tanreqing injection for treating acute lung injury: In vivo, in vitro and in silico 期刊论文  OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2025, 卷号: 337, 页码: 11
作者:  
Tang, Bixi;  Xie, Like;  Wang, Yangyang;  Shi, Yulong;  Kan, Weijuan
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/11/26
B(MIDA)-directed site-selective intermolecular halofluoroalkylation of alkenes: synthesis of diversely functionalized building blocks 期刊论文  OAI收割
CHEMICAL SCIENCE, 2025, 页码: 8
作者:  
Wu, Hengbo;  Luo, Ruitong;  Peng, Jingjing;  Han, Zijian;  Zhang, Renjie
  |  收藏  |  浏览/下载:13/0  |  提交时间:2025/04/01
Discovery of peptidomimetic spiropyrrolidine derivatives as novel 3CLpro inhibitors against SARS-CoV-2 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 281, 页码: 22
作者:  
Guma, Samuel Desta;  Zhou, Zhaoyin;  Song, Kang;  Yang, Feipu;  Suo, Jin
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/12/11
F-CPI: A Multimodal Deep Learning Approach for Predicting Compound Bioactivity Changes Induced by Fluorine Substitution 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 13
作者:  
Zhang, Qian;  Yin, Wenhai;  Chen, Xinyao;  Zhou, Aimin;  Zhang, Guixu
  |  收藏  |  浏览/下载:13/0  |  提交时间:2025/02/28
Identification of USP2 as a novel target to induce degradation of KRAS in myeloma cells 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 12, 页码: 5235-5248
作者:  
Wang, Yingying;  Zhang, Youping;  Luo, Hao;  Wei, Wei;  Liu, Wanting
  |  收藏  |  浏览/下载:18/0  |  提交时间:2025/04/01