中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
广州生物医药与健康... [19]
上海药物研究所 [1]
大连化学物理研究所 [1]
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OAI收割 [21]
内容类型
期刊论文 [21]
发表日期
2018 [1]
2016 [7]
2015 [4]
2014 [4]
2013 [5]
学科主题
Science & ... [8]
Pharmacolo... [6]
Engineerin... [2]
Materials ... [2]
Research &... [2]
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Y08060: A Selective BET Inhibitor for Treatment of Prostate Cancer
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 9, 期号: 3, 页码: 262-267
作者:
Xiang, Quping
;
Zhang, Yan
;
Li, Jiaguo
;
Xue, Xiaoqian
;
Wang, Chao
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2019/06/20
Bromodomain
Brd4
Prostate Cancer
Epigenetics
Enhanced renoprotective effect of IGF-1 modified human umbilical cord-derived mesenchymal stem cells on gentamicin-induced acute kidney injury
期刊论文
OAI收割
SCIENTIFIC REPORTS, 2016, 卷号: 6
Liu, Pengfei
;
Feng, Yetong
;
Dong, Delu
;
Liu, Xiaobo
;
Chen, Yaoyu
;
Wang, Yi
;
Zhou, Yulai
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2016/12/16
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
;
Xue, Xiaoqian
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2018/12/13
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
作者:
Xue, Xiaoqian
;
Song, Yu
;
Qian, Chao-Nan
;
Yan, Weiqun
;
Xing, Yanli
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2018/12/13
Enhanced renoprotective effect of IGF-1 modified human umbilical cord-derived mesenchymal stem cells on gentamicin-induced acute kidney injury
期刊论文
OAI收割
SCIENTIFIC REPORTS, 2016, 卷号: 6
作者:
Liu, Pengfei
;
Liu, Xiaobo
;
Feng, Yetong
;
Dong, Delu
;
Zhou, Yulai
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian
;
Zhang, Yan
;
Liu, Zhaoxuan
;
Song, Ming
;
Xing, Yanli
;
Xiang, Qiuping
;
Wang, Zhen
;
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2016/12/16
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
Song, Yu
;
Xue, Xiaoqian
;
Wu, Xishan
;
Wang, Rui
;
Xing, Yanli
;
Yan, Weiqun
;
Zhou, Yulai
;
Qian, Chao-Nan
;
Zhang, Yan
;
Xu, Yong
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2016/12/16
Discovery and structural optimization of 4-(4-(benzyloxy) phenyl)-3,4-dihydropyrimidin-2(1H)-ones as RORc inverse agonists
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 11, 页码: 1516
作者:
Wu Xishan
;
Wang Rui
;
Xing Yanli
;
Xue Xiaoqian
;
Zhang Yan
  |  
收藏
  |  
浏览/下载:85/0
  |  
提交时间:2020/12/24
GAMMA-T
ORPHAN RECEPTORS
CELL-DIFFERENTIATION
LIGAND
IDENTIFICATION
MODULATORS
DERIVATIVES
PROTEIN
INHIBITORS
DOCKING
nuclear receptor
RORc
inverse agonist
SAR
structure-based optimization
autoimmune disease
Effects of SOX2 on Proliferation, Migration and Adhesion of Human Dental Pulp Stem Cells
期刊论文
OAI收割
PLOS ONE, 2015, 卷号: 10, 期号: 10
作者:
Dong, Delu
;
Liu, Pengfei
;
Cai, Jinglei
;
Chen, Yaoyu
;
Liu, Xiaobo
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2018/12/13
Protective effect of vitamin E against acute kidney injury
期刊论文
OAI收割
BIO-MEDICAL MATERIALS AND ENGINEERING, 2015, 卷号: 26, 页码: S2133-S2144
作者:
Feng, Yetong
;
Liu, Pengfei
;
Zhao, Lei
;
Zhou, Yulai
;
Wang, Yi
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2018/12/13