中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
采集方式
内容类型
发表日期
学科主题
筛选

浏览/检索结果: 共98条,第1-10条 帮助

条数/页: 排序方式:
Rapid Discovery of Celastrol Derivatives as Potent and Selective PRDX1 Inhibitors via Microplate-Based Parallel Compound Library and In Situ Screening 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 13, 页码: 13609-13627
作者:  
Chen, Shuang;  Wang, Zhenyu;  Gao, Jia;  Wang, Yanlin;  Liang, Jiayin
  |  收藏  |  浏览/下载:19/0  |  提交时间:2025/08/20
Understanding the coupled relationship between regional longevity and physical geographical environment in Hechi, Guangxi, China 期刊论文  OAI收割
SCIENTIFIC REPORTS, 2024, 卷号: 14, 期号: 1, 页码: 32154
作者:  
Deng, Qucheng;  Liu, Yaqing;  Wei, Yongping;  Liang, Wei;  Zhu, Kaixian
  |  收藏  |  浏览/下载:36/0  |  提交时间:2025/02/24
Berberine Derivative B68 Promotes Tumor Immune Clearance by Dual-Targeting BMI1 for Senescence Induction and CSN5 for PD-L1 Degradation 期刊论文  OAI收割
ADVANCED SCIENCE, 2024, 页码: 21
作者:  
Hu, Hongmei;  Wang, Qun;  Yu, Dianping;  Tao, Xiaoyu;  Guo, Mengmeng
  |  收藏  |  浏览/下载:55/0  |  提交时间:2025/02/28
The Association Between Environmental Factors and Longevity in Hezhou, China Based on the Drinking Water Quality 期刊论文  OAI收割
EXPOSURE AND HEALTH, 2024, 卷号: N/A
作者:  
Deng, Qucheng;  Liu, Yaqing;  Zhu, Kaixian;  Han, Xuerong;  Erpeng, Yang
  |  收藏  |  浏览/下载:58/0  |  提交时间:2025/01/17
Application of ensemble learning for predicting GABAA receptor agonists 期刊论文  OAI收割
COMPUTERS IN BIOLOGY AND MEDICINE, 2024, 卷号: 169, 页码: 13
作者:  
Xiao, Fu;  Ding, Xiaoyu;  Shi, Yan;  Wang, Dingyan;  Wang, Yitian
  |  收藏  |  浏览/下载:71/0  |  提交时间:2024/03/25
Design, synthesis and biological evaluation of chalcone derivatives as potent and orally active hCYP3A4 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 9
作者:  
Lu, Shiwei;  Zhang, Feng;  Gong, Jiahao;  Huang, Jian;  Zhu, Guanghao
  |  收藏  |  浏览/下载:72/0  |  提交时间:2023/12/08
Design, synthesis and biological evaluation of salicylanilides as novel allosteric inhibitors of human pancreatic lipase 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 91, 页码: 11
作者:  
Zhao, Yitian;  Zhang, Min;  Hou, Xudong;  Han, Jiaxin;  Qin, Xiaoya
  |  收藏  |  浏览/下载:75/0  |  提交时间:2023/10/17
Discovery of Small-Molecule Degraders of the CDK9-Cyclin T1 Complex for Targeting Transcriptional Addiction in Prostate Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 16, 页码: 11034-11057
作者:  
Li, Jiacheng;  Liu, Ting;  Song, Yuanli
  |  收藏  |  浏览/下载:50/0  |  提交时间:2024/03/21
Chemo- and Site-Selective Lysine Modification of Peptides and Proteins under Native Conditions Using the Water-Soluble Zolinium 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 14
作者:  
Sun, Haiguo;  Xi, Mengyu;  Jin, Qiang;  Zhu, Zhengdan;  Zhang, Yani
  |  收藏  |  浏览/下载:76/0  |  提交时间:2022/09/30
Design, Synthesis, and Biological Evaluation of Peptidomimetic Aldehydes as Broad-Spectrum Inhibitors against Enterovirus and SARS-CoV-2 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 4, 页码: 2794-2808
作者:  
Dai, Wenhao;  Jochmans, Dirk;  Xie, Hang;  Yang, Hang;  Li, Jian
  |  收藏  |  浏览/下载:66/0  |  提交时间:2022/08/16