中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
昆明植物研究所 [43]
上海药物研究所 [19]
青岛生物能源与过程研... [1]
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期刊论文 [64]
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2023 [1]
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Identification of 3H-benzo[b] [1,4] diazepine derivatives as PPAR alpha agonists by in silico studies and biochemical evaluation
期刊论文
OAI收割
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, 2023, 页码: 16
作者:
Li, Yue
;
Lv, Mengjia
;
Shen, Meiling
;
Gu, Xi
;
Zhang, Li
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
NAFLD
PPAR alpha agonist
virtual screening
biochemical evaluation
Development and structure-activity relationships of tanshinones as selective 11β-hydroxysteroid dehydrogenase 1 inhibitors
期刊论文
OAI收割
NATURAL PRODUCTS AND BIOPROSPECTING, 2022, 卷号: 12, 期号: 6, 页码: 1
作者:
Deng Xu
;
Huang Suling
;
Ren Jian
;
Pan Zhenghong
;
Shen Yu
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/05/22
Metabolic syndrome
Tanshinones
Selective 11β-HSD1 inhibitors
Structure-activity relationships
Discovery of novel inhibitors against main protease (Mpro) of SARS-CoV-2 via virtual screening and biochemical evaluation
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 110, 页码: 8
作者:
Guo, Sheng
;
Xie, Hang
;
Lei, Yu
;
Liu, Bin
;
Zhang, Li
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2021/08/17
SARS-CoV-2
Main protease
Virtual screening
Biochemical evaluation
Heterogeneous Fenton-like reaction followed by GAC filtration improved removal efficiency of NOM and DBPs without adjusting pH
期刊论文
OAI收割
SEPARATION AND PURIFICATION TECHNOLOGY, 2021, 卷号: 260, 页码: -
作者:
Zhang, Yao
;
Lu, Zhili
;
Zhang, Zeyu
;
Shi, Baoyou
;
Hu, Chun
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2021/12/23
Heterogeneous Fenton-like reaction
Granular activated carbon filtration
Natural organic matter
Disinfection by-products
Genotoxicity
Which species does the virus like most: Binding modes study between SARS-CoV-2 S protein and ACE2 receptor
期刊论文
OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2021, 卷号: 105, 页码: 107893
作者:
Guo,Sheng
;
Yang,Jing
;
Lei,Yu
;
Liu,Bin
;
Zhang,Wei
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/04/02
SARS-CoV-2
COVID-19
Homology modeling
Molecular dynamics simulation
Binding free energy
CORONAVIRUS SPIKE PROTEIN
ACTIVATION
GROMACS
ENTRY
Enantioselective access to tricyclic tetrahydropyran derivatives by a remote hydrogen bonding mediated intramolecular IEDHDA reaction
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 7188
作者:
Jin,Min
;
Tang,Congyun
;
Li,Yingying
;
Yang,Shuai
;
Yang,Ying-Tao
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/04/02
DIELS-ALDER REACTION
BIOMIMETIC TOTAL-SYNTHESIS
ORTHO-QUINONE METHIDES
BRONSTED ACID
CYCLIZATION
ACTIVATION
OLEFINS
CYCLOADDITIONS
CATALYSIS
ENTRY
Discovery of novel inhibitors against main protease (Mpro) of SARS-CoV-2 via virtual screening and biochemical evaluation
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 110, 页码: 104767
作者:
Guo,Sheng
;
Xie,Hang
;
Lei,Yu
;
Liu,Bin
;
Zhang,Li
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/04/02
SARS-CoV-2
Main protease
Virtual screening
Biochemical evaluation
Discovery of novel modulators targeting human TRPC5: Docking-based virtual screening, molecular dynamics simulation and binding af fi nity predication
期刊论文
OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2021, 卷号: 102, 页码: 107795
作者:
Liu,Bin
;
Zhang,Wei
;
Guo,Sheng
;
Zuo,Zhili
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/04/02
hTRPC5
Homology modeling
Molecular docking
Molecular dynamics simulation
Virtual screening
INHIBITOR
CHANNELS
GROMACS
POTENT
AMBER
IDENTIFICATION
CONSTRAINTS
INTEGRATION
AMYGDALA
Oligosaccharides from fucosylated glycosaminoglycan prevent breast cancer metastasis in mice by inhibiting heparanase activity and angiogenesis
期刊论文
OAI收割
PHARMACOLOGICAL RESEARCH, 2021, 卷号: 166, 页码: 105527
作者:
Zhou,Lutan
;
Yin,Ronghua
;
Gao,Na
;
Sun,Huifang
;
Chen,Dingyuan
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2022/04/02
Oligosaccharides
Heparanase
Angiogenesis
Metastasis
FIBROBLAST-GROWTH-FACTOR
TUMOR-GROWTH
SULFATE PROTEOGLYCANS
MAMMALIAN HEPARANASE
COMBINATION
MECHANISMS
DISCOVERY
BINDING
TARGET
PI-88
INDITTO2 transposon conveys auxin-mediated DRO1 transcription for rice drought avoidance
期刊论文
OAI收割
PLANT CELL AND ENVIRONMENT, 2021, 卷号: 44, 期号: 6, 页码: 1846-1857
作者:
Zhao,Yiting
;
Wu,Lixia
;
Fu,Qijing
;
Wang,Dong
;
Li,Jing
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/04/02
DNA transposable elements
indoleacetic acid
Oryza
stress