中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [11]
兰州化学物理研究所 [4]
西北高原生物研究所 [3]
昆明植物研究所 [3]
生态环境研究中心 [3]
长春应用化学研究所 [3]
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OAI收割 [34]
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期刊论文 [31]
学位论文 [3]
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2022 [1]
2020 [4]
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2017 [1]
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Chemistry [4]
Medicinal [3]
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浏览/检索结果:
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HIF-1alpha/VEGF pathway mediates 1,3,6,8-tetrabromo-9 H-carbazole-induced angiogenesis: a potential vascular toxicity of an emerging contaminant
期刊论文
OAI收割
JOURNAL OF HAZARDOUS MATERIALS, 2022, 卷号: 432, 期号: 0, 页码: 128718
作者:
Xu, Tong
;
Hu, Xiaoxu
;
Yang, Guanglei
;
Liu, Yiyun
;
Zhang, Qian
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2022/11/08
ARYL-HYDROCARBON RECEPTOR
HALOGENATED CARBAZOLES
TUMOR ANGIOGENESIS
HYPOXIA
DIOXIN
VEGF
HIF-1-ALPHA
SYSTEM
CANCER
OXYGEN
TCDD 对红系细胞分化相关基因的调控作用及机制探索
学位论文
OAI收割
北京: 中国科学院大学;中国科学院生态环境研究中心, 2020
作者:
马永超
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/06/16
二恶英,Tf-1 细胞,芳香烃受体,促红细胞生成素,乙酰胆碱酯酶
dioxins, Tf-1 Cells, Aryl Hydrocarbon Receptors, Erythropoietin, Acetylcholinesterase
Synthesis and biological evaluation of heterocyclic bis-aryl amides as novel Src homology 2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 11, 页码: 5
作者:
Satheeshkumar, Rajendran
;
Zhu, Rui
;
Feng, Bo
;
Huang, Chao
;
Gao, Ya
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2020/07/01
Heterocyclic bis-aryl amides
PTP1B
SHP2
Inhibitors
Structure-activity relationships (SAR)
Discovery of aryl sulfonamide-selective Nav1.7 inhibitors with a highly hydrophobic ethanoanthracene core
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 293-302
作者:
Wang, Jin-tao
;
Zheng, Yue-ming
;
Chen, Yue-ting
;
Gu, Min
;
Gao, Zhao-bing
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2020/07/01
Nav1
7 sodium channel
aryl sulfonamide
maprotiline
compound 10o
electrophysiology
acetic acid-induced visceral pain
analgesic activity
Direct decarboxylative C-H 3-arylation of quinoxalin-2(H)-ones with aryl acyl peroxides leading to 3-arylquinoxalin-2(1H)-ones
期刊论文
OAI收割
TETRAHEDRON LETTERS, 2020, 卷号: 61, 期号: 47
作者:
Lv, Yufen
;
Bao, Pengli
;
Yue, Huilan
;
Wei, Wei
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/11/25
3-arylquinoxalin-2(1H)-ones
Catalyst-free
C-H 3-arylation
Aryl acyl peroxides
Synthesis and biological evaluation of 3-aryl-4-indolyl-maleimides as potent mutant isocitrate dehydrogenase-1 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 4, 页码: 589-603
作者:
Liu, Xiaoqi
;
Hu, Yuanyuan
;
Gao, Anhui
;
Xu, Meng
;
Gao, Lixin
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/07/01
3-Aryl-4-indolyl-maleimides
IDH1/R132H inhibitors
Tumor 2-HG
Synthesis
Direct C-H3 3-Arylation of Quinoxalin-2(H)-ones with Aryl Diazonium Salts under Visible-Light Irradiation
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2018, 卷号: 38, 期号: 12
作者:
Wang Leilei
;
Bao Pengli
;
Liu Weiwei
;
Liu Sitong
;
Hu Changsong
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2019/11/26
visible-light
Eosin Y catalysis
C-H arylation
aryl diazonium salt
3-arylquinoxalin-2(1H)-one
Metal-Free Synthesis of 1,2,4-Triazines via a Coupled Domino Process in One-Pot
期刊论文
OAI收割
Current Organic Chemistry, 2017, 卷号: 21, 期号: 2, 页码: 183-188
作者:
Wang, Jing
;
Tang, Dong
;
Li, Zhuo-Mei
;
Wu, Ping
;
Meng X(孟旭)
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2017/02/20
1,2,4-Triazines
domino strategy
aryl alkenes
amidrazones
Kornblum oxidation
metal-free
Synthesis of Novel 3-aryl-1-oxa-2,8-diazaspiro[4.5]dec-2-ene Derivatives and Their Biological Evaluation Against Protein Tyrosine Phosphatase 1B
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2015, 卷号: 86, 期号: 5, 页码: 1161-1167
作者:
Wang, Wen-Long
;
Chen, Xia
;
Gao, Li-Xin
;
Sheng, Li
;
Li, Jing-Ya
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
3-aryl-1-oxa-2,8-diazaspiro[4.5]dec-2-ene derivatives
inhibitors
one-pot synthesis
protein tyrosine phosphatase 1B
structure-activity relationships
Rh(I)-catalyzed asymmetric 1,2-additions of arylboronic acids to isatins with chiral sulfur-alkene hybrid ligands
期刊论文
OAI收割
TETRAHEDRON LETTERS, 2014, 卷号: 55, 期号: 33, 页码: 4581-4584
作者:
Feng, Xiangqing
;
Nie, Yanzhao
;
Zhang, Lanqiong
;
Yang, Jing
;
Du, Haifeng
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/04/09
3-aryl-3-hydroxy-2-oxindoles
Chiral Sulfur-alkene Ligands
Rhodium-catalyzed
Asymmetric Catalysis
1
2-addition