中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [12]
金属研究所 [10]
昆明植物研究所 [5]
南海海洋研究所 [1]
西双版纳热带植物园 [1]
新疆理化技术研究所 [1]
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期刊论文 [35]
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Divalent tranylcypromine derivative as lysine-specific demethylase 1 inhibitor
期刊论文
OAI收割
MEDICINAL CHEMISTRY RESEARCH, 2021, 页码: 8
作者:
Sun, Yin
;
Li, Na
;
Su, Mingbo
;
Wang, Xiaowen
;
Zhao, Dongmei
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2021/05/24
Divalent tranylcypromine
LSD1 inhibitor
MV4-11 antiproliferative activity
CD86 mRNA expression
Linker
Selectivity
Antiproliferative abietane quinone diterpenoids from the roots of Salvia deserta
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 104, 期号: 11, 页码: 1-12
作者:
Zheng, XF (Zheng, Xiaofeng)[ 1 ]
;
Kadir, A (Kadir, Abdukriem)[ 1,2 ]
;
Zheng, GJ (Zheng, Guijuan)[ 1 ]
;
Jin, PF (Jin, Pengfei)[ 1 ]
;
Qin, DM (Qin, Dongmei)[ 3 ]
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2021/01/05
Salvia deserta Schang (Lamiaceae)
Abietane quinone diterpenoids
Calculated C-13 NMR-DP4+analysis
Mo-2(OAc)(4)-induced ECD
Antiproliferative activity
New New cytotoxic ergostane-type sterols from the Chinese soft coral Sinularia sp.
期刊论文
OAI收割
STEROIDS, 2019, 卷号: 149, 页码: 5
作者:
Jiang, Cheng-Shi
;
Ru, Tong
;
Huan, Xia-Juan
;
Miao, Ze-Hong
;
Guo, Yue-Wei
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2020/07/01
Soft coral
Sinularia sp.
Ergostane
Antiproliferative activity
Apoptosis
Antiproliferative Aspidosperma-Type Monoterpenoid Indole Alkaloids from Bousigonia mekongensis Inhibit Tubulin Polymerization
期刊论文
OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 7, 页码: 10
作者:
Zhang, Yu
;
Goto, Masuo
;
Oda, Akifumi
;
Hsu, Pei-Ling
;
Guo, Ling-Li
  |  
收藏
  |  
浏览/下载:81/0
  |  
提交时间:2019/07/29
aspidosperma-type
monoterpenoid indole alkaloids
antiproliferative activity
tubulin inhibitor
Bousigonia mekongensis
Tranylcypromine and 6-trifluoroethyl thienopyrimidine hybrid as LSD1 inhibitor
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 844-847
作者:
Wang, Xiaowen
;
Su, Mingbo
;
Li, You
;
Liu, Tongchao
;
Wang, Yujie
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/07/01
LSD1 inhibitor
Tranylcypromine
Menin-MLL1 protei n-protein interaction inhibitor
MV4-11 antiproliferative activity
Structure activity relationship
Targeting the PI3K/Akt/mTOR signaling pathway by pterostilbene attenuates mantle cell lymphoma progression
期刊论文
OAI收割
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2018, 卷号: 50, 期号: 8, 页码: 782-792
作者:
Yu, Dandan
;
Zhang, Yong
;
Chen, Gege
;
Xie, Yongsheng
;
Xu, Zhijian
  |  
收藏
  |  
浏览/下载:64/0
  |  
提交时间:2019/01/08
mantle cell lymphoma
pterostilbene
antiproliferative activity
PI3K/Akt/mTOR pathway
synergistic cytotoxicity
Design, synthesis and pharmacological evaluation of ALK and Hsp90 dual inhibitors bearing resorcinol and 2,4-diaminopyrimidine motifs
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 76-86
作者:
Geng, Kaijun
;
Liu, Hongchun
;
Song, Zilan
;
Zhang, Chi
;
Zhang, Minmin
  |  
收藏
  |  
浏览/下载:187/0
  |  
提交时间:2019/01/08
Heat shock protein 90 (Hsp90)
Tyrosine kinase ALK
Dual inhibitor
Drug resistance
Antiproliferative activity
targetingthepi3kaktmtorsignalingpathwaybypterostilbeneattenuatesmantlecelllymphomaprogression
期刊论文
OAI收割
actabiochimicaetbiophysicasinica, 2018, 卷号: 50, 期号: 8, 页码: 782
作者:
Yu Dandan
;
Zhang Yong
;
Chen Gege
;
Xie Yongsheng
;
Xu Zhijian
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/07/01
PROTEIN-KINASE PATHWAY
CANCER IN-VITRO
TRANSDUCTION PATHWAYS
CYCLE ARREST
APOPTOSIS
ACTIVATION
PATHOGENESIS
INHIBITION
ANTICANCER
EXPRESSION
mantle cell lymphoma
pterostilbene
antiproliferative activity
PI3K/Akt/mTOR pathway
synergistic cytotoxicity
Meroterpenoids with Antitumor Activities from Guava (Psidium guajava)
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2017, 卷号: 65, 期号: 24, 页码: 4993-4999
作者:
Qin, Xu-Jie
;
Yu, Qian
;
Yan, Huan
;
Khan, Afsar
;
Feng, Mi-Yan
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2017/07/31
guava
meroterpenoids
cytotoxicity
DNA topoisomerase I inhibitors
antiproliferative activity
Synthesis and antiproliferative activities of 5H-benzo[b]carbazole-6,11-diones
期刊论文
OAI收割
Journal of China Pharmaceutical University, 2017, 卷号: 48, 期号: 2, 页码: 157-166
作者:
Cao Sufen
;
Xie Qin
;
Chen Yi
;
Duan Wenhu
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08
5H-benzo[b]carbazole-6,11-dione
synthesis
antiproliferative activity