机构

• 上海药物研究所 [6]
• 中国科学院大学 [1]

采集方式

• OAI收割 [6]
• iSwitch采集 [1]

内容类型

• 期刊论文 [7]

发表日期

• 2023 [1]
• 2022 [3]
• 2020 [1]
• 2016 [2]

学科主题

筛选

浏览/检索结果: 共7条，第1-7条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序发表日期升序发表日期降序提交时间升序提交时间降序作者升序作者降序 Discovery of new small molecule inhibitors of the BPTF bromodomain 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2023, 卷号: 134, 页码: 106453 作者:  Liang, Xiaochen;  Cao, Yu;  Duan, Zhe;  Wang, Mingchen;  Zhang, Naixia   |  收藏  |  浏览/下载：16/0  |  提交时间：2024/03/27 BPTF bromodomain  BPTF inhibitors  HTRF  c-Myc   Discovery of novel benzimidazole derivatives as potent p300 bromodomain inhibitors with anti-proliferative activity in multiple cancer cells 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 66, 页码: 16 作者:  Chen, Zonglong;  Li, Jiayi;  Yang, Hong;  He, Yulong;  Shi, Qiongyu   |  收藏  |  浏览/下载：60/0  |  提交时间：2022/08/16 P300  Bromodomain inhibitors  CBP30  SBDD   Design, synthesis and biological evaluation of (R)-5-methylpyrrolidin-2-ones as p300 bromodomain inhibitors with Anti-Tumor activities in multiple tumor lines 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2022, 卷号: 124, 页码: 15 作者:  Liu, Ruiqi;  Yang, Hong;  Chen, Zonglong;  Zhou, Kaixin;  Shi, Qiongyu   |  收藏  |  浏览/下载：61/0  |  提交时间：2022/08/16 Epigenetics  p300  CBP  Bromodomain inhibitors  CCS1477   Discovery of CECR2 Bromodomain Inhibitors with High Selectivities over BPTF Bromodomain 期刊论文  OAI收割 CHINESE JOURNAL OF CHEMISTRY, 2022, 页码: 2072-2080 作者:  Lu, Haibo;  Zu, Shijia;  Duan, Zhe;  Feng, Yueyao;  Wang, Jie   |  收藏  |  浏览/下载：44/0  |  提交时间：2022/08/16 CECR2 bromodomain  BPTF bromodomain  Inhibitors  Structure-activity relationships  chemical probe   A patent review of BRD4 inhibitors (2013-2019) 期刊论文  OAI收割 EXPERT OPINION ON THERAPEUTIC PATENTS, 2020, 卷号: 30, 期号: 1, 页码: 57-81 作者:  Lu, Tian;  Lu, Wenchao;  Luo, Cheng   |  收藏  |  浏览/下载：38/0  |  提交时间：2020/07/01 Bromodomain-containing protein 4 (BRD4)  bromodomain and extra-terminal (BET) family  small molecule inhibitors  cancer  patent  therapeutic potential   Nmr-based platform for fragment-based lead discovery used in screening brd4-targeted compounds 期刊论文  iSwitch采集 Acta pharmacologica sinica, 2016, 卷号: 37, 期号: 7, 页码: 984-993 作者:  Yu, Jun-lan;  Chen, Tian-tian;  Zhou, Chen;  Lian, Fu-lin;  Tang, Xu-long 收藏  |  浏览/下载：33/0  |  提交时间：2019/05/09 Fragment-based lead discovery  Nmr  Bromodomain  Brd4 inhibitors   NMR-based platform for fragment-based lead discovery used in screening BRD4-targeted compounds 期刊论文  OAI收割 ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 7, 页码: 984-993 作者:  Yu, Jun-lan;  Chen, Tian-tian;  Zhou, Chen;  Lian, Fu-lin;  Tang, Xu-long   |  收藏  |  浏览/下载：29/0  |  提交时间：2019/01/08 fragment-based lead discovery  NMR  bromodomain  BRD4 inhibitors