中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
金属研究所 [2]
福建物质结构研究所 [1]
化学研究所 [1]
上海药物研究所 [1]
采集方式
OAI收割 [5]
内容类型
期刊论文 [5]
发表日期
2020 [1]
2009 [3]
2006 [1]
学科主题
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Design of G-protein-coupled bile acid receptor 1 (GPBAR1, TGR5) soft drugs with reduced gallbladder-filling effects
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 12
作者:
Han, Fanghui
;
Ning, Mengmeng
;
Cao, Hua
;
Ye, Yangliang
;
Feng, Ying
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/12/21
Soft drug
TGR5
GLP-1
Gallbladder-filling effects
Rapid metabolism
Carboxylic ester
Crystal Structures of 2-Aminobenzothiazole-based Inhibitors in Complexes with Urokinase-type Plasminogen Activator
期刊论文
OAI收割
Chinese Journal of Structural Chemistry, 2009, 卷号: 28, 期号: 11, 页码: 1427-1432
L. G. Jiang, H. Y. Yu, C. Yuan, J. D. Wang, L. Q. Chen, E. J. Meehan, Z. X. Huang and M. D. Huang
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2012/11/06
urokinase-type plasminogen activator
2-aminobenzothiazole
2-amino-benzothiazole-6-carboxylic acid ethyl ester
P1 group
selective inhibitors
system
subsite
design
Design, Synthesis, and Biological Evaluation of 5H-Thiazolo3,2-apyrimidine-6-carboxylic Acid Ethyl Ester Derivatives as a Novel Series of Acetylcholinesterase Inhibitors
期刊论文
OAI收割
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 3, 页码: 332-337
作者:
Zhi Hui
;
Chen Lanmei
;
Zhang Linlin
;
Liu Sijie
;
Wan David Chi Cheong
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2021/02/02
Acetylcholinesterase inhibitor
Docking screening
Heterocycle
Biological activity
5H-Thiazolo3,2-a pyrimidine-6-carboxylic acid ethyl ester derivative
Design, Synthesis, and Biological Evaluation of 5H-Thiazolo3,2-apyrimidine-6-carboxylic Acid Ethyl Ester Derivatives as a Novel Series of Acetylcholinesterase Inhibitors
期刊论文
OAI收割
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 3, 页码: 332-337
作者:
Zhi Hui
;
Chen Lanmei
;
Zhang Linlin
;
Liu Sijie
;
Wan David Chi Cheong
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/02/02
Acetylcholinesterase inhibitor
Docking screening
Heterocycle
Biological activity
5H-Thiazolo3,2-a pyrimidine-6-carboxylic acid ethyl ester derivative
Labeling analysis of neuropeptides with 7-methoxycoumarin-3-carboxylic acid N-succinimidyl ester
期刊论文
OAI收割
CHEMICAL JOURNAL OF CHINESE UNIVERSITIES-CHINESE, 2006, 卷号: 27, 期号: 12, 页码: 2297-2299
作者:
Jun, Li
;
Liu Xiang-Jun
;
Rui, Zhao
;
Xiong Shao-Xiang
;
Ma Hui-Min
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/04/09
Neuropeptides
Labeling Analysis
7-methoxycoumarin-3-carboxylic Acid N-succimidyl Ester