中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共17条,第1-10条 帮助

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Discovery of indole derivatives as STING degraders 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 21
作者:  
An, Yuxiang;  Zhang, Yan;  Luo, Xin;  Lan, Yaohan;  Geng, Meiyu
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/08/20
First ATG101-recruiting small molecule degrader for selective CDK9 degradation via autophagy-lysosome pathway 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 5, 页码: 2612-2624
作者:  
Zhong, Ye;  Xu, Jing;  Cao, Huiying;  Gao, Jie;  Ding, Shaoyue
  |  收藏  |  浏览/下载:17/0  |  提交时间:2025/07/25
Cross-Linking Profiling of Molecular Glue Degrader-Induced E3 Ligase Interactome to Expand Target Space 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 13
作者:  
Xu, Yali;  Zhao, Wensi;  Nie, Hui-Jun;  Wang, Jiamin;  Fu, Jingjing
  |  收藏  |  浏览/下载:20/0  |  提交时间:2025/05/27
Recent advances in targeted degradation in the RAS pathway 期刊论文  OAI收割
FUTURE MEDICINAL CHEMISTRY, 2025, 卷号: 17, 期号: 6, 页码: 693-708
作者:  
Ge, Zhiming;  Fan, Zisheng;  He, Wei;  Zhou, Guizhen;  Zhou, Yidi
  |  收藏  |  浏览/下载:14/0  |  提交时间:2025/04/24
Discovery of a Potent, selective and orally bioavailable CDK9 degrader for targeting transcription regulation in Triple-Negative breast cancer 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 153, 页码: 16
作者:  
Nie, Hui-Jun;  Li, Ben-Fu;  Sun, Jingya;  Yuan, Yali;  Zhang, Zhi-Gao
  |  收藏  |  浏览/下载:43/0  |  提交时间:2024/11/26
Discovery of KW0113 as a First and Effective PROTAC Degrader of DNMT1 Protein 期刊论文  OAI收割
CHEMMEDCHEM, 2024, 页码: 16
作者:  
Wang, Huihui;  Wang, Zhaoliang;  Hu, Linghao;  Yang, Bingjie;  Zong, Liangyi
  |  收藏  |  浏览/下载:30/0  |  提交时间:2024/12/16
SIP-metagenomics reveals key drivers of rhizospheric Benzo[a]pyrene bioremediation via bioaugmentation with indigenous soil microbes☆ 期刊论文  OAI收割
ENVIRONMENTAL POLLUTION, 2024, 卷号: 360, 页码: 12
作者:  
Zhao, Xuan;  Cheng, Xianghui;  Cai, Xixi;  Wang, Shuang;  Li, Jibing
  |  收藏  |  浏览/下载:39/0  |  提交时间:2024/09/13
Targeting EGFR with molecular degraders as a promising strategy to overcome resistance to EGFR inhibitors 期刊论文  OAI收割
FUTURE MEDICINAL CHEMISTRY, 2024, 页码: 22
作者:  
Wang, Qiangfeng;  Zhu, Yumeng;  Pei, Junping
  |  收藏  |  浏览/下载:42/0  |  提交时间:2024/10/21
Cultivation and characterization of functional-yet-uncultivable phenanthrene degraders by stable-isotope-probing and metagenomic-binning directed cultivation (SIP-MDC) 期刊论文  OAI收割
ENVIRONMENT INTERNATIONAL, 2024, 卷号: 185, 页码: 11
作者:  
Li, Jibing;  Luo, Chunling;  Cai, Xixi;  Dai, Yeliang;  Zhang, Dayi
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/09/12
In Situ Discrimination and Cultivation of Active Degraders in Soils by Genome-Directed Cultivation Assisted by SIP-Raman-Activated Cell Sorting 期刊论文  OAI收割
ENVIRONMENTAL SCIENCE & TECHNOLOGY, 2023, 卷号: 57, 期号: 44, 页码: 17087-17098
作者:  
Li, Jibing;  Zhang, Dayi;  Luo, Chunling;  Li, Bei;  Zhang, Gan
  |  收藏  |  浏览/下载:21/0  |  提交时间:2024/09/14