中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [22]
昆明动物研究所 [3]
中国科学院大学 [1]
上海生物化学与细胞生... [1]
上海营养与健康研究所 [1]
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OAI收割 [27]
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期刊论文 [26]
学位论文 [2]
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2025 [3]
2022 [2]
2019 [1]
2018 [3]
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2016 [4]
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Science & ... [2]
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(+)-Borneol Enhances the Antiseizure Effects of Retigabine by both Pharmacokinetic and Pharmacodynamic Interaction
期刊论文
OAI收割
NEUROCHEMICAL RESEARCH, 2025, 卷号: 50, 期号: 3, 页码: 13
作者:
Xu, Haiyan
;
Wu, Zhidan
;
Wang, Pei
;
Gong, Jili
;
Qiu, Li
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/06/23
Epilepsy
Retigabine
(+)-Borneol
Synergistic interaction
KCNQ channels
Phosphatidylinositol 4,5-bisphosphate activation mechanism of human KCNQ5
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 14, 页码: 11
作者:
Yang, Zhenni
;
Zheng, Yueming
;
Ma, Demin
;
Wang, Long
;
Zhang, Jiatong
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/06/23
KCNQ
PIP2
ligand activation
structure
mechanism
Electrophysiological Abnormalities and Pharmacological Corrections of Pathogenic Missense Variants in KCNQ3
期刊论文
OAI收割
NEUROSCIENCE BULLETIN, 2025, 页码: 11
作者:
Wu, Xiaorong
;
Gong, Jili
;
Qiu, Li
;
Yang, Guimei
;
Yuan, Hui
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/05/27
KCNQ3
Self-limited familial neonatal epilepsy
Neurodevelopmental disorder
Pynegabine
Amitriptyline
Electrophysiology
Epilepsy phenotype and response to KCNQ openers in mice harboring the Kcnq2 R207W voltage-sensor mutation
期刊论文
OAI收割
NEUROBIOLOGY OF DISEASE, 2022, 卷号: 174, 页码: 10
作者:
Tian, Fuyun
;
Cao, Birong
;
Xu, Haiyan
;
Zhan, Li
;
Nan, Fajun
  |  
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2022/12/13
KCNQ2
Epilepsy
Mouse model
HN37 (pynegabine)
Diversity-oriented synthesis of marine polybrominated diphenyl ethers as potential KCNQ potassium channel activators
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 126, 页码: 105909
作者:
Liu, Lai-Xin
;
Gu, Ru-Rong
;
Jin, Yang
;
Chen, Xue-Qin
;
Li, Xu-Wen
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/03/21
Marine Natural product
Polybrominated diphenyl ethers
KCNQ potassium channel
Discovery of Novel Retigabine Derivatives as Potent KCNQ4 and KCNQ5 Channel Agonists with Improved Specificity
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 10, 期号: 1, 页码: 27-33
作者:
Wang, Lei
;
Qiao, Guan-Hua
;
Hu, Hai-Ning
;
Gao, Zhao-Bing
;
Nan, Fa-Jun
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2020/07/01
KCNQ channel
retigabine
subtype selectivity
agonist
以离子通道为基础的动物生存策略研究进展
学位论文
OAI收割
北京: 中国科学院大学, 2018
作者:
罗雷
  |  
收藏
  |  
浏览/下载:129/0
  |  
提交时间:2019/09/27
Trpv1
失活
Kcnq
Sstx
Retigabine
Desensitization
A Statistical Thermodynamic Model for Ligands Interacting With Ion Channels: Theoretical Model and Experimental Validation of the KCNQ2 Channel
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9
作者:
Bai, Fang
;
Pi, Xiaoping
;
Li, Ping
;
Zhou, Pingzheng
;
Yang, Huaiyu
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2019/01/08
KCNQ2 potassium channel
hill equation
thermodynamic model
patch clamp electrophysiology
activators
Centipedes subdue giant prey by blocking KCNQ channels
期刊论文
OAI收割
PNAS, 2018, 卷号: 115, 期号: 7, 页码: 1646–1651
作者:
Rose Ombati
;
Xiancui Lu
;
Jianmin Cui
;
Qiumin Lu
;
Longhua Zhang
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2018/09/26
Centipede
Toxicity
Sstx
Kcnq
Mitochondrial dynamics controls anti-tumour innate immunity by regulating CHIP-IRF1 axis stability
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2017, 卷号: 8, 期号: -, 页码: 1805
作者:
Gao, Zhengjun
;
Li, Yiyuan
;
Wang, Fei
;
Huang, Tao
;
Fan, Keqi
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/12/09
Electrophysiology
Long QT syndrome
KCNQ1
Selectivity filter