中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
上海药物研究所 [6]
水生生物研究所 [3]
中国科学院大学 [1]
采集方式
OAI收割 [9]
iSwitch采集 [1]
内容类型
期刊论文 [10]
发表日期
2023 [1]
2020 [1]
2019 [1]
2018 [2]
2016 [2]
2014 [1]
更多
学科主题
Biochemist... [1]
筛选
浏览/检索结果:
共10条,第1-10条
帮助
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
题名升序
题名降序
提交时间升序
提交时间降序
作者升序
作者降序
发表日期升序
发表日期降序
Discovery, Structure-Activity Relationship and In Vitro Anticancer Activity of Small-Molecule Inhibitors of the Protein-Protein Interactions between AF9/ENL and AF4 or DOT1L
期刊论文
OAI收割
CANCERS, 2023, 卷号: 15, 期号: 21, 页码: 28
作者:
Li, Xin
;
Wu, Xiaowei
;
Nie, Shenyou
;
Zhao, Jidong
;
Yao, Yuan
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2023/12/19
MLL-rearranged leukemia
super elongation complexes
small-molecule inhibitor
protein-protein interaction
cancer therapeutics
The Development of Inhibitors Targeting the Mixed Lineage Leukemia 1 (MLL1)-WD Repeat Domain 5 Protein (WDR5) Protein-Protein Interaction
期刊论文
OAI收割
CURRENT MEDICINAL CHEMISTRY, 2020, 卷号: 27, 期号: 33, 页码: 5530-5542
作者:
Ye, Xiaoqing
;
Chen, Gang
;
Jin, Jia
;
Zhang, Binzhong
;
Wang, Yinda
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/12/24
WDR5
MLL1
histone methyltransferase
small-molecular inhibitor
epigenetics
human acute leukemia
The identification of novel small-molecule inhibitors targeting WDR5-MLL1 interaction through fluorescence polarization based high-throughput screening
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 4, 页码: 638-645
作者:
Ye, Xiaoqing
;
Zhang, Rukang
;
Lian, Fulin
;
Zhang, Weiyao
;
Lu, Wenchao
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
WDR5-MLL1 interaction
Leukemia
Small-molecule
High-throughput screening
Fluorescence polarization (FP)
Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1751-1758
作者:
Song, Yakai
;
Li, Linjuan
;
Chen, Yantao
;
Liu, Jingqiu
;
Xiao, Senhao
  |  
收藏
  |  
浏览/下载:60/0
  |  
提交时间:2019/01/08
DOT1L
MLL-rearranged leukemia
AlphaLISA
HTS
Novel inhibitors
Piribedil disrupts the MLL1-WDR5 interaction and sensitizes MLL-rearranged acute myeloid leukemia (AML) to doxorubicin-induced apoptosis
期刊论文
OAI收割
CANCER LETTERS, 2018, 卷号: 431, 页码: 150-160
作者:
Zhang, Xiong
;
Zheng, Xingling
;
Yang, Hong
;
Yan, Juan
;
Fu, Xuhong
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2019/01/08
MLL leukemia
Piribedil
H3K4 methylation
Cell cycle
Apoptosis
Design and synthesis of benzylpiperidine inhibitors targeting the menin-mll1 interface
期刊论文
iSwitch采集
Bioorganic & medicinal chemistry letters, 2016, 卷号: 26, 期号: 18, 页码: 4472-4476
作者:
Ren, Jing
;
Xu, Wei
;
Tang, Le
;
Su, Minbo
;
Chen, Danqi
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2019/05/09
Menin
Mixed lineage leukemia
Mll1
Sar
Inhibitor
Design and synthesis of benzylpiperidine inhibitors targeting the menin-MLL1 interface
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 18, 页码: 4472-4476
作者:
Ren, Jing
;
Xu, Wei
;
Tang, Le
;
Su, Minbo
;
Chen, Danqi
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
Menin
Mixed lineage leukemia
MLL1
SAR
Inhibitor
ELL Inhibits E2F1 Transcriptional Activity by Enhancing E2F1 Deacetylation via Recruitment of Histone Deacetylase 1
期刊论文
OAI收割
MOLECULAR AND CELLULAR BIOLOGY, 2014, 卷号: 34, 期号: 4, 页码: 765-775
作者:
Zhang, Wei
;
Ji, Wei
;
Liu, Xing
;
Ouyang, Gang
;
Xiao, Wuhan
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2014/08/13
RNA-POLYMERASE-II
ELONGATION-FACTOR ELL
MIXED-LINEAGE LEUKEMIA
DNA-DAMAGE
COMPLEX SEC
CELL-DEATH
MLL-ELL
PROTEIN
GENE
TRANSACTIVATION
E2F-1 Directly Regulates Thrombospondin 1 Expression
期刊论文
OAI收割
PLOS ONE, 2010, 卷号: 5, 期号: 10, 页码: -e13442
作者:
Ji, Wei
;
Zhang, Wei
;
Xiao, Wuhan
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2010/12/23
CELL-CYCLE CONTROL
ENDOTHELIAL-CELLS
RB/E2F PATHWAY
LEUKEMIA
MICE
ANGIOGENESIS
GENE
MLL
APOPTOSIS
CD36
Elongation Factor ELL (Eleven-Nineteen Lysine-rich Leukemia) Acts as a Transcription Factor for Direct Thrombospondin-1 Regulation
期刊论文
OAI收割
JOURNAL OF BIOLOGICAL CHEMISTRY, 2009, 卷号: 284, 期号: 28, 页码: 19142-19152
作者:
Zhou, Jiangang
;
Feng, Xi
;
Ban, Bin
;
Liu, Jingxia
;
Wang, Zhou
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2010/10/13
MIXED LINEAGE LEUKEMIA
ACUTE MYELOID-LEUKEMIA
MLL-ELL
TUMOR-GROWTH
STEM-CELLS
GENE
EXPRESSION
ANGIOGENESIS
P53
POLYMERASE