中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
采集方式
内容类型
发表日期
学科主题
筛选

浏览/检索结果: 共10条,第1-10条 帮助

条数/页: 排序方式:
Discovery, Structure-Activity Relationship and In Vitro Anticancer Activity of Small-Molecule Inhibitors of the Protein-Protein Interactions between AF9/ENL and AF4 or DOT1L 期刊论文  OAI收割
CANCERS, 2023, 卷号: 15, 期号: 21, 页码: 28
作者:  
Li, Xin;  Wu, Xiaowei;  Nie, Shenyou;  Zhao, Jidong;  Yao, Yuan
  |  收藏  |  浏览/下载:27/0  |  提交时间:2023/12/19
The Development of Inhibitors Targeting the Mixed Lineage Leukemia 1 (MLL1)-WD Repeat Domain 5 Protein (WDR5) Protein-Protein Interaction 期刊论文  OAI收割
CURRENT MEDICINAL CHEMISTRY, 2020, 卷号: 27, 期号: 33, 页码: 5530-5542
作者:  
Ye, Xiaoqing;  Chen, Gang;  Jin, Jia;  Zhang, Binzhong;  Wang, Yinda
  |  收藏  |  浏览/下载:29/0  |  提交时间:2020/12/24
The identification of novel small-molecule inhibitors targeting WDR5-MLL1 interaction through fluorescence polarization based high-throughput screening 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 4, 页码: 638-645
作者:  
Ye, Xiaoqing;  Zhang, Rukang;  Lian, Fulin;  Zhang, Weiyao;  Lu, Wenchao
  |  收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1751-1758
作者:  
Song, Yakai;  Li, Linjuan;  Chen, Yantao;  Liu, Jingqiu;  Xiao, Senhao
  |  收藏  |  浏览/下载:60/0  |  提交时间:2019/01/08
Piribedil disrupts the MLL1-WDR5 interaction and sensitizes MLL-rearranged acute myeloid leukemia (AML) to doxorubicin-induced apoptosis 期刊论文  OAI收割
CANCER LETTERS, 2018, 卷号: 431, 页码: 150-160
作者:  
Zhang, Xiong;  Zheng, Xingling;  Yang, Hong;  Yan, Juan;  Fu, Xuhong
  |  收藏  |  浏览/下载:49/0  |  提交时间:2019/01/08
Design and synthesis of benzylpiperidine inhibitors targeting the menin-mll1 interface 期刊论文  iSwitch采集
Bioorganic & medicinal chemistry letters, 2016, 卷号: 26, 期号: 18, 页码: 4472-4476
作者:  
Ren, Jing;  Xu, Wei;  Tang, Le;  Su, Minbo;  Chen, Danqi
收藏  |  浏览/下载:42/0  |  提交时间:2019/05/09
Design and synthesis of benzylpiperidine inhibitors targeting the menin-MLL1 interface 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 18, 页码: 4472-4476
作者:  
Ren, Jing;  Xu, Wei;  Tang, Le;  Su, Minbo;  Chen, Danqi
  |  收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
ELL Inhibits E2F1 Transcriptional Activity by Enhancing E2F1 Deacetylation via Recruitment of Histone Deacetylase 1 期刊论文  OAI收割
MOLECULAR AND CELLULAR BIOLOGY, 2014, 卷号: 34, 期号: 4, 页码: 765-775
作者:  
Zhang, Wei;  Ji, Wei;  Liu, Xing;  Ouyang, Gang;  Xiao, Wuhan
收藏  |  浏览/下载:31/0  |  提交时间:2014/08/13
E2F-1 Directly Regulates Thrombospondin 1 Expression 期刊论文  OAI收割
PLOS ONE, 2010, 卷号: 5, 期号: 10, 页码: -e13442
作者:  
Ji, Wei;  Zhang, Wei;  Xiao, Wuhan
收藏  |  浏览/下载:19/0  |  提交时间:2010/12/23
Elongation Factor ELL (Eleven-Nineteen Lysine-rich Leukemia) Acts as a Transcription Factor for Direct Thrombospondin-1 Regulation 期刊论文  OAI收割
JOURNAL OF BIOLOGICAL CHEMISTRY, 2009, 卷号: 284, 期号: 28, 页码: 19142-19152
作者:  
Zhou, Jiangang;  Feng, Xi;  Ban, Bin;  Liu, Jingxia;  Wang, Zhou
收藏  |  浏览/下载:42/0  |  提交时间:2010/10/13