中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [22]
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浏览/检索结果:
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Discovery, Structure-Activity Relationship and In Vitro Anticancer Activity of Small-Molecule Inhibitors of the Protein-Protein Interactions between AF9/ENL and AF4 or DOT1L
期刊论文
OAI收割
CANCERS, 2023, 卷号: 15, 期号: 21, 页码: 28
作者:
Li, Xin
;
Wu, Xiaowei
;
Nie, Shenyou
;
Zhao, Jidong
;
Yao, Yuan
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/12/19
MLL-rearranged leukemia
super elongation complexes
small-molecule inhibitor
protein-protein interaction
cancer therapeutics
Design, synthesis of novel benzimidazole derivatives as ENL inhibitors suppressing leukemia cells viability via downregulating the expression of MYC
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 248, 页码: 14
作者:
Guo, Siqi
;
Jia, Tongguan
;
Xu, Xiaoming
;
Yang, Feng
;
Xiao, Senhao
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/04/10
ENL Inhibitor
YEATS domain
Histone lysine acetylation
Benzimidazole derivatives
Acute myeloid leukemia
Novel figuring method for a multilayer Laue lens
期刊论文
OAI收割
Optics Express, 2022, 卷号: 30, 期号: 26, 页码: 46838-46848
作者:
Ji, Bin
;
Yue, Shuaipeng,
;
Zhou, Liang
;
Li, Ming
;
Chang, Guangcai,
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2023/11/10
Single-order focus multilayer Laue lens
期刊论文
OAI收割
Applied Optics, 2022, 卷号: 61, 期号: 27, 页码: 8028-8033
作者:
Ji, Bin
;
Yue, Shuaipeng,
;
Zhou, Liang
;
Chang, Guangcai
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2023/11/09
Phase noise reduction of a 2 µm passively mode-locked laser through hybrid III-V/silicon integration
期刊论文
OAI收割
Optica, 2021, 卷号: 8, 期号: 6, 页码: 855-860
作者:
X. Li
;
J. X. B. Sia
;
W. J. Wang
;
Z. L. Qiao
;
X. Guo
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/06/13
Discovery of novel CBP bromodomain inhibitors through TR-FRET-based high-throughput screening
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 2, 页码: 286-292
作者:
Zhang, Feng-cai
;
Sun, Zhong-ya
;
Liao, Li-ping
;
Zuo, Yu
;
Zhang, Dan
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2020/07/01
CBP bromodomain
small-molecule inhibitor
high-throughput screening
TR-FRET
molecular modeling
human leukemia MV4-11 cells
Characterization of functional transposable element enhancers in acute myeloid leukemia
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2020, 卷号: 63, 期号: 5, 页码: 675-687
作者:
Zeng, Yingying
;
Cao, Yaqiang
;
Liu, Denghui
;
Zhang, Xiaoli
;
Han, Jing-Dong J.
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收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/12/21
SET ENRICHMENT ANALYSIS
C-JUN
GENE
GENOME
CHROMATIN
EVOLUTION
MLL-AF9
PROTEIN
DNA
DIFFERENTIATION
The expression of histone methyltransferases and distribution of selected histone methylations in testes of yak and cattle-yak hybrid
期刊论文
OAI收割
THERIOGENOLOGY, 2020, 卷号: 144
作者:
Li, Yong-Chang
;
Wang, Guo-Wen
;
Xu, Shang-Rong
;
Zhang, Xiao-Na
;
Yang, Qi-En
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收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/11/25
Yak
Hybrid male sterility
Histone methylation
Spermatogenesis
Meiosis
The Development of Inhibitors Targeting the Mixed Lineage Leukemia 1 (MLL1)-WD Repeat Domain 5 Protein (WDR5) Protein-Protein Interaction
期刊论文
OAI收割
CURRENT MEDICINAL CHEMISTRY, 2020, 卷号: 27, 期号: 33, 页码: 5530-5542
作者:
Ye, Xiaoqing
;
Chen, Gang
;
Jin, Jia
;
Zhang, Binzhong
;
Wang, Yinda
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2020/12/24
WDR5
MLL1
histone methyltransferase
small-molecular inhibitor
epigenetics
human acute leukemia
Repetition frequency variation of a 2 m GaSb-based passively mode-locked laser Invited
期刊论文
OAI收割
Hongwai yu Jiguang Gongcheng/Infrared and Laser Engineering, 2020, 卷号: 49, 期号: 12, 页码: 5
作者:
X. Li,H. Wang,Z. Qiao,Y. Zhang,Z. Niu,C. Tong and C. Liu
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2021/07/06