中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [20]
上海神经科学研究所 [13]
金属研究所 [5]
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武汉物理与数学研究所 [2]
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iSwitch采集 [1]
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期刊论文 [53]
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2025 [3]
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2019 [1]
2017 [1]
2016 [2]
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AI-driven breakthroughs in ion channel drug discovery: the future is now
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 2
作者:
Zheng, Ming-yue
;
Gao, Zhao-bing
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2026/01/29
ion channel
artificial intelligence
deep learning
drug discovery
NMDA receptor
New advances in small molecule drugs targeting NMDA receptors
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 19
作者:
Zeng, Yue
;
Qu, Zhi-yan
;
Zhu, Qian-wen
;
Wang, Hai-ying
;
Zhou, Yu
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/12/04
N
-methyl-
D
-aspartate (NMDA) receptor
small-molecule modulators
depression
CNS disorders
channel blocker
allosteric modulator
An efficient deep learning-based strategy to screen inhibitors for GluN1/GluN3A receptor
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 9
作者:
Wang, Ze-chen
;
Zeng, Yue
;
Sun, Jin-yuan
;
Chen, Xue-qin
;
Wu, Hao-chen
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2025/04/24
deep learning
scoring function
GluN1/GluN3A receptor
N
-methyl-
D
-aspartate (NMDA) receptor
virtual screening
drug discovery
Design, Synthesis and Bioactivity of NYX-2925
L
-Proline Derivatives as
N
-Methyl-D-aspartate (NMDA) Receptor Partial Agonists
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 4, 页码: 1247-1263
作者:
Wu Youjin
;
Jin Zhengsheng
;
Liu Yongjia
;
Huang Wenqian
;
Zhao Guilong
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2024/08/22
N-methyl-D-aspartate (NMDA) receptor
partial agonist
NYX-2925
synthesis
bioactivity
Temporal transformer-spatial graph convolutional network: an intelligent classification model for anti N-methyl-D-aspartate receptor encephalitis based on electroencephalogram signal
期刊论文
OAI收割
FRONTIERS MEDIA SA, 2023, 卷号: 17
作者:
Dang, Ruochen
;
Yu, Tao
;
Hu, Bingliang
;
Wang, Yuqi
;
Pan, Zhibin
  |  
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2023/10/10
anti NMDA receptor encephalitis
viral encephalitis
EEG
transformer
graph network
classification
Cholecystokinin release triggered by NMDA receptors produces LTP and sound-sound associative memory
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2019, 卷号: 116, 期号: 13, 页码: 6397-6406
作者:
He, Jufang
;
Xu, Fuqiang
;
Guo, Yiping
;
Tortorella, Micky
;
Chan, Ying-Shing
  |  
收藏
  |  
浏览/下载:166/0
  |  
提交时间:2019/06/24
cholecystokinin
NMDA receptor
long-term potentiation
memory
entorhinal cortex
Incorporation of Dihydroartemisinin into Memantine Through a Propriate Spacer to Make Hybrid with Enhanced Effects to Protect PC12 Cells from Corticosterone-caused Impairments
期刊论文
OAI收割
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2017, 卷号: 33, 期号: 4, 页码: 611-622
作者:
Zhang Lei
;
Zhou Fan
;
Zhang Laitao
;
Peng Lizhi
;
Guo Cuiping
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/01/08
Artemisinin
Memantine
Neuroprotection
N-Methyl-D-aspartate(NMDA) receptor
Depression
Timosaponin derivative YY-23 acts as a non-competitive NMDA receptor antagonist and exerts a rapid antidepressant-like effect in mice
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 2, 页码: 166-176
作者:
Zhang, Qi
;
Guo, Fei
;
Fu, Zhi-wen
;
Zhang, Bing
;
Huang, Cheng-gang
  |  
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2019/01/08
Rhizoma Anemarrhenae
timosaponin
YY-23
depression
NMDA receptor antagonist
chronic mild stress
chronic social defeat stress
fluoxetine
Large-Scale Persistent Network Reconfiguration Induced by Ketamine in Anesthetized Monkeys: Relevance to Mood Disorders
期刊论文
OAI收割
BIOLOGICAL PSYCHIATRY, 2016, 卷号: 79, 期号: 9, 页码: 765-775
作者:
Lv, Q
;
Yang, LQ
;
Li, GL
;
Wang, ZW
;
Shen, ZM
收藏
  |  
浏览/下载:72/0
  |  
提交时间:2016/09/14
STATE FUNCTIONAL CONNECTIVITY
TREATMENT-RESISTANT DEPRESSION
NMDA RECEPTOR BLOCKADE
MAJOR DEPRESSION
NONHUMAN-PRIMATES
PREFRONTAL CORTEX
BRAIN NETWORKS
ARCHITECTURE
HUMANS
ANTIDEPRESSANTS
Neural circuits containing olfactory neurons are involved in the prepulse inhibition of the startle reflex in rats
期刊论文
OAI收割
FRONTIERS IN BEHAVIORAL NEUROSCIENCE, 2015, 卷号: 9
作者:
Niu, Haichen
;
He, Xiaobin
;
Zhou, Ting
;
Shi, Xi
;
Zhang, Qiang
收藏
  |  
浏览/下载:71/0
  |  
提交时间:2015/06/23
olfactory dysfunction
sensory stimulus
prepulse inhibition (PPI)
NMDA receptor
neural trace