中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共8条,第1-8条 帮助

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Discovery and characterization of a novel highly potent and selective type II native and drug-resistant V299L mutant BCR-ABL inhibitor (CHMFL-ABL-039) for Chronic Myeloid Leukemia (CML) 期刊论文  OAI收割
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 6, 页码: 877-885
作者:  
Wu, Jiaxin;  Wang, Aoli;  Li, Xixiang;  Chen, Cheng;  Qi, Ziping
  |  收藏  |  浏览/下载:88/0  |  提交时间:2019/11/27
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:  
Wang, Qiang;  Liu, Feiyang;  Qi, Shuang;  Qi, Ziping;  Yan, Xiao-E.
  |  收藏  |  浏览/下载:76/0  |  提交时间:2019/06/10
Discovery and characterization of a novel potent type II native and mutant BCR-ABL inhibitor (CHMFL-074) for Chronic Myeloid Leukemia (CML) 期刊论文  OAI收割
ONCOTARGET, 2016, 卷号: 7, 期号: 29, 页码: 45562-45574
作者:  
Liu, Feiyang;  Wang, Beilei;  Wang, Qiang;  Qi, Ziping;  Chen, Cheng
收藏  |  浏览/下载:49/0  |  提交时间:2017/11/21
Establishment of the active catalytic domain of human PDGFR beta tyrosine kinase-based ELISA assay for inhibitor screening 期刊论文  OAI收割
BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS, 2007, 卷号: 1770, 期号: 10, 页码: 1490-1497
作者:  
Zhang, Xiu-Hua;  Guo, Xiao-Ning;  Zhong, Li;  Luo, Xiao-Min;  Jiang, Hua-Liang
  |  收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
TKI-31 inhibits angiogenesis by combined suppression signaling pathway of VEGFR2 and PDGFR beta 期刊论文  OAI收割
CANCER BIOLOGY & THERAPY, 2006, 卷号: 5, 期号: 3, 页码: 323-330
作者:  
Zhong, L;  Guo, XN;  Zhang, XH;  Sun, QM;  Tong, LJ
  |  收藏  |  浏览/下载:26/0  |  提交时间:2019/01/08