中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
上海药物研究所 [28]
西北高原生物研究所 [18]
合肥物质科学研究院 [5]
上海营养与健康研究所 [3]
广州生物医药与健康研... [2]
中国科学院大学 [1]
更多
采集方式
OAI收割 [58]
iSwitch采集 [1]
内容类型
期刊论文 [57]
会议论文 [1]
学位论文 [1]
发表日期
2021 [2]
2019 [1]
2018 [5]
2017 [3]
2016 [3]
2015 [13]
更多
学科主题
Cell Biolo... [5]
Oncology [5]
Biochemist... [1]
Biochemist... [1]
Biophysics [1]
Endocrinol... [1]
更多
筛选
浏览/检索结果:
共59条,第1-10条
帮助
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
提交时间升序
提交时间降序
发表日期升序
发表日期降序
题名升序
题名降序
作者升序
作者降序
Discovery of a novel DDRs kinase inhibitor XBLJ-13 for the treatment of idiopathic pulmonary fibrosis
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Dong, Ying
;
Tang, Bi-xi
;
Wang, Qi
;
Zhou, Li-wei
;
Li, Cong
  |  
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2022/01/04
idiopathic pulmonary fibrosis
DDRs
kinase inhibitor
indazole derivatives
XBLJ-13
nintedanib
bleomycin-induced pulmonary fibrosismouse model
Anlotinib in Locally Advanced or Metastatic Medullary Thyroid Carcinoma: A Randomized, Double-Blind Phase IIB Trial
期刊论文
OAI收割
CLINICAL CANCER RESEARCH, 2021, 卷号: 27
作者:
Li, Dapeng
;
Chi, Yihebali
;
Chen, Xiaohong
;
Ge, Minghua
;
Zhang, Yuan
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2021/08/31
Discovery and characterization of a novel highly potent and selective type II native and drug-resistant V299L mutant BCR-ABL inhibitor (CHMFL-ABL-039) for Chronic Myeloid Leukemia (CML)
期刊论文
OAI收割
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 6, 页码: 877-885
作者:
Wu, Jiaxin
;
Wang, Aoli
;
Li, Xixiang
;
Chen, Cheng
;
Qi, Ziping
  |  
收藏
  |  
浏览/下载:76/0
  |  
提交时间:2019/11/27
BCR-ABL
PDGFR
chronic myeloid leukemia
kinase inhibitor
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFRα kinase inhibi
期刊论文
OAI收割
Eur. J. Med. Chem., 2018
作者:
Qiang Wang
;
Feiyang Liu
;
Qi S(亓爽)
;
Ziping Qi
;
Beilei Wang
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2020/10/20
SOMCL-085, a novel multi-targeted FGFR inhibitor, displays potent anticancer activity in FGFR-addicted human cancer models
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 2, 页码: 243-250
作者:
Jiang, Xi-fei
;
Dai, Yang
;
Peng, Xia
;
Shen, Yan-yan
;
Su, Yi
  |  
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2019/01/08
human cancer
anticancer drug
SOMCL-085
receptor tyrosine kinase
FGFR
xenograft nude mouse model
somcl085anovelmultitargetedfgfrinhibitordisplayspotentanticanceractivityinfgfraddictedhumancancermodels
期刊论文
OAI收割
actapharmacologicasinica, 2018, 卷号: 39, 期号: 2, 页码: 243
作者:
Jiang Xifei
;
Dai Yang
;
Peng Xia
;
Shen Yanyan
;
Su Yi
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
human cancer
anticancer drug
SOMCL-085
receptor tyrosine kinase
FGFR
xenograft nude mouse model
Reversible De-differentiation of Mature White Adipocytes into Preadipocyte-like Precursors during Lactation
期刊论文
OAI收割
CELL METABOLISM, 2018, 卷号: 28, 期号: 2, 页码: 282-+
作者:
Wang, Qiong A.
;
Zhang, Fang
;
Vishvanath, Lavanya
;
Ye, Risheng
;
Shao, Mengle
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2020/12/09
liver kinase B1
metformin
pancreatic cancer
Snail
ubiquitination
Dihydroartemisinin selectively inhibits PDGFR alpha-positive ovarian cancer growth and metastasis through inducing degradation of PDGFR alpha protein
期刊论文
OAI收割
CELL DISCOVERY, 2017, 卷号: 3
作者:
Li, Xiaoguang
;
Ba, Qian
;
Liu, Yanling
;
Yue, Qingxi
;
Chen, Peizhan
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2019/01/08
Dihydroartemisinin
Epithelial-mesenchymal transition
metastasis
ovarian cancer
PDGFR alpha
Lyn mediates FIP1L1-PDGFRA signal pathway facilitating IL-5RA intracellular signal through FIP1L1-PDGFRA/JAK2/Lyn/Akt network complex in CEL
期刊论文
OAI收割
ONCOTARGET, 2017, 卷号: 8, 期号: 39, 页码: 64984-64998
作者:
Li, Bin
;
Li, Cui
;
Peng, Zhenzi
;
Wang, Jun
;
Dong, Yeping
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/12/09
Lyn
CEL