中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共59条,第1-10条 帮助

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Discovery of a novel DDRs kinase inhibitor XBLJ-13 for the treatment of idiopathic pulmonary fibrosis 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  
Dong, Ying;  Tang, Bi-xi;  Wang, Qi;  Zhou, Li-wei;  Li, Cong
  |  收藏  |  浏览/下载:52/0  |  提交时间:2022/01/04
Anlotinib in Locally Advanced or Metastatic Medullary Thyroid Carcinoma: A Randomized, Double-Blind Phase IIB Trial 期刊论文  OAI收割
CLINICAL CANCER RESEARCH, 2021, 卷号: 27
作者:  
Li, Dapeng;  Chi, Yihebali;  Chen, Xiaohong;  Ge, Minghua;  Zhang, Yuan
  |  收藏  |  浏览/下载:40/0  |  提交时间:2021/08/31
Discovery and characterization of a novel highly potent and selective type II native and drug-resistant V299L mutant BCR-ABL inhibitor (CHMFL-ABL-039) for Chronic Myeloid Leukemia (CML) 期刊论文  OAI收割
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 6, 页码: 877-885
作者:  
Wu, Jiaxin;  Wang, Aoli;  Li, Xixiang;  Chen, Cheng;  Qi, Ziping
  |  收藏  |  浏览/下载:76/0  |  提交时间:2019/11/27
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:  
Wang, Qiang;  Liu, Feiyang;  Qi, Shuang;  Qi, Ziping;  Yan, Xiao-E.
  |  收藏  |  浏览/下载:62/0  |  提交时间:2019/06/10
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFRα kinase inhibi 期刊论文  OAI收割
Eur. J. Med. Chem., 2018
作者:  
Qiang Wang;  Feiyang Liu;  Qi S(亓爽);  Ziping Qi;  Beilei Wang
  |  收藏  |  浏览/下载:25/0  |  提交时间:2020/10/20
SOMCL-085, a novel multi-targeted FGFR inhibitor, displays potent anticancer activity in FGFR-addicted human cancer models 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 2, 页码: 243-250
作者:  
Jiang, Xi-fei;  Dai, Yang;  Peng, Xia;  Shen, Yan-yan;  Su, Yi
  |  收藏  |  浏览/下载:53/0  |  提交时间:2019/01/08
somcl085anovelmultitargetedfgfrinhibitordisplayspotentanticanceractivityinfgfraddictedhumancancermodels 期刊论文  OAI收割
actapharmacologicasinica, 2018, 卷号: 39, 期号: 2, 页码: 243
作者:  
Jiang Xifei;  Dai Yang;  Peng Xia;  Shen Yanyan;  Su Yi
  |  收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
Reversible De-differentiation of Mature White Adipocytes into Preadipocyte-like Precursors during Lactation 期刊论文  OAI收割
CELL METABOLISM, 2018, 卷号: 28, 期号: 2, 页码: 282-+
作者:  
Wang, Qiong A.;  Zhang, Fang;  Vishvanath, Lavanya;  Ye, Risheng;  Shao, Mengle
  |  收藏  |  浏览/下载:10/0  |  提交时间:2020/12/09
Dihydroartemisinin selectively inhibits PDGFR alpha-positive ovarian cancer growth and metastasis through inducing degradation of PDGFR alpha protein 期刊论文  OAI收割
CELL DISCOVERY, 2017, 卷号: 3
作者:  
Li, Xiaoguang;  Ba, Qian;  Liu, Yanling;  Yue, Qingxi;  Chen, Peizhan
  |  收藏  |  浏览/下载:43/0  |  提交时间:2019/01/08
Lyn mediates FIP1L1-PDGFRA signal pathway facilitating IL-5RA intracellular signal through FIP1L1-PDGFRA/JAK2/Lyn/Akt network complex in CEL 期刊论文  OAI收割
ONCOTARGET, 2017, 卷号: 8, 期号: 39, 页码: 64984-64998
作者:  
Li, Bin;  Li, Cui;  Peng, Zhenzi;  Wang, Jun;  Dong, Yeping
  |  收藏  |  浏览/下载:13/0  |  提交时间:2020/12/09
Lyn  CEL