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浏览/检索结果: 共70条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序提交时间升序提交时间降序作者升序作者降序发表日期升序发表日期降序 Antidepressant and anxiolytic profiles of newly synthesized arginine vasopressin 期刊论文  OAI收割 出版物, 3111, 期号: 0, 页码: 1-62 作者:  M Iijima;  T Yoshimizu;  T Shimazaki;  K Tokugawa;  K Fukumoto   |  收藏  |  浏览/下载：622/0  |  提交时间：2017/07/24 Arginine Vasopressin  V1b Receptor Antagonist  Depression  Anxiety  Hpa Axis   The antidepressant-like effect and proposed mechanism of action of TPN672MA, a novel serotonin-dopamine receptor modulator for the treatment of schizophrenia 期刊论文  OAI收割 PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 2024, 卷号: 242, 页码: 13 作者:  Cheng, Jiaxin;  Wu, Chunhui;  Wang, Yu;  Wang, Zhen;  He, Yang   |  收藏  |  浏览/下载：12/0  |  提交时间：2024/09/24 TPN672MA  5-HT 1A receptor agonist  D 2 /D 3 receptor partial agonist  5-HT 2A receptor antagonist  Antidepressant-like  Mechanism   Design and Synthesis Studies of α-Methylene-γ-butyrolactones Antagonists of GPR52 期刊论文  OAI收割 CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2023, 卷号: 43, 期号: 11, 页码: 3916-3929 作者:  Shen, Donghang;  Li, Xin;  Guo, Shimeng;  Xie, Xin;  Nan, Fajun   |  收藏  |  浏览/下载：29/0  |  提交时间：2024/02/27 Huntingdon's disease  G protein-coupled receptor  GPR52  alpha-methylene-gamma-butyrolactones  antagonist   Synthesis of Hydantoin Androgen Receptor Antagonists and Study on Their Antagonistic Activity 期刊论文  OAI收割 MOLECULES, 2022, 卷号: 27, 期号: 18, 页码: 22 作者:  Ma, Longjun;  Zhou, Yan;  Yang, Dehua;  Wang, Ming-Wei;  Lu, Wei   |  收藏  |  浏览/下载：49/0  |  提交时间：2022/11/11 androgen receptor  antagonist  enzalutamide  hydantoin analogs  antiproliferative   Constructing an MCF-7 breast cancer cell-based transient transfection assay for screening RAR? (Ant)agonistic activities of emerging phenolic compounds 期刊论文  OAI收割 JOURNAL OF HAZARDOUS MATERIALS, 2022, 卷号: 435, 期号: 0, 页码: 129024 作者:  Xu, Hanqing;  Su, Jiahui;  Ku, Tingting;  Liu, Qian S.;  Liang, Jiefeng   |  收藏  |  浏览/下载：37/0  |  提交时间：2022/11/08 ACID RECEPTOR-ALPHA  RETINOIC ACID  GENE-EXPRESSION  DEPENDENT TRANSCRIPTION  GROWTH-INHIBITION  IN-VITRO  RXR  CONTAMINANTS  ANTAGONIST  ACTIVATION   Medulloblastoma: Molecular understanding, treatment evolution, and new developments 期刊论文  OAI收割 PHARMACOLOGY & THERAPEUTICS, 2020, 卷号: 210, 页码: 13 作者:  Liu, Xiaohua;  Ding, Chunyong;  Tan, Wenfu;  Zhang, Ao   |  收藏  |  浏览/下载：49/0  |  提交时间：2020/07/01 Medulloblastoma  Pediatric brain tumor  Oncogenic driver gene  Hedgehog pathway inhibitor  Smoothened receptor antagonist   Revealing the Positive Binding Cooperativity Mechanism between the Orthosteric and the Allosteric Antagonists of CCR2 by Metadynamics and Gaussian Accelerated Molecular Dynamics Simulations 期刊论文  OAI收割 ACS CHEMICAL NEUROSCIENCE, 2020, 卷号: 11, 期号: 4, 页码: 628-637 作者:  An, Xiaoli;  Bai, Qifeng;  Bing, Zhitong;  Liu, Hongli;  Zhang, Qianqian   |  收藏  |  浏览/下载：29/0  |  提交时间：2022/01/18 CC chemokine receptor 2  orthosteric antagonist  allosteric antagonist  binding cooperativity  metadynamics simulation  Gaussian accelerated MD simulation   Systematic characterization of AT1 receptor antagonists with label-free dynamic mass redistribution assays 期刊论文  OAI收割 JOURNAL OF PHARMACOLOGICAL AND TOXICOLOGICAL METHODS, 2020, 卷号: 102 作者:  Qu, Lala;  Wang, Jixia;  Hou, Tao;  Zhou, Han;  Wang, Zhiwei   |  收藏  |  浏览/下载：25/0  |  提交时间：2020/11/25 Angiotensin II type 1 receptor  Antagonist  Binding property  Dynamic mass redistribution assay   Discovery of Novel Androgen Receptor Ligands by Structure-based Virtual Screening and Bioassays 期刊论文  OAI收割 GENOMICS PROTEOMICS & BIOINFORMATICS, 2019, 卷号: 16, 期号: 6, 页码: 416-427 作者:  Hou, Tingjun;  Li, Dan;  Chang, Shan;  Xu, Lei;  Sun, Huiyong   |  收藏  |  浏览/下载：278/0  |  提交时间：2019/06/24 Androgen receptor  AR ligand  Virtual screening  AR agonist  AR antagonist   How Does Agonist and Antagonist Binding Lead to Different Conformational Ensemble Equilibria of the kappa-Opioid Receptor: Insight from Long-Time Gaussian Accelerated Molecular Dynamics Simulation 期刊论文  OAI收割 ACS CHEMICAL NEUROSCIENCE, 2019, 卷号: 10, 期号: 3, 页码: 1575-1584 作者:  An, Xiaoli;  Bai, Qifeng;  Bing, Zhitong;  Zhou, Shuangyan;  Shi, Danfeng   |  收藏  |  浏览/下载：68/0  |  提交时间：2019/11/10 kappa-opioid receptor  Gaussian accelerated molecular dynamics simulation  agonist  antagonist  conformational change