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中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共306条,第1-10条 帮助

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Covalent sortase A inhibitor, α, β-unsaturated aldehydes, prevents Staphylococcus aureus infection 期刊论文  OAI收割
MICROBIAL PATHOGENESIS, 2025, 卷号: 204, 页码: 12
作者:  
Wang, Jianchao;  He, Yuan;  Chu, Chenliang;  Wu, Ziqi;  Zhang, Ting
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:  
Wu, Xinyuan;  Li, Shunyao;  Liang, Ting;  Yu, Qing;  Zhang, Yiwei
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Dynamic Cap-Mediated Substrate Access and Potent Inhibitor Design of Monkeypox Virus I7L Protease 期刊论文  OAI收割
ADVANCED SCIENCE, 2025, 页码: 13
作者:  
Su, Haixia;  Wu, Guoqing;  Xiong, Muya;  Wang, Yuhang;  Cao, Junyuan
  |  收藏  |  浏览/下载:2/0  |  提交时间:2025/05/27
Discovery of Covalent and Cell-Active ALKBH5 Inhibitors with Potent Antileukemia Effects In Vivo 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 9
作者:  
Wu, Hengbo;  Lai, Gan-Qiang;  Cheng, Ruixiang;  Huang, Hui;  Wang, Ju
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/04/24
Discovery of novel covalent stabilizers for p53 Y220C using structure-based drug discovery methods 期刊论文  OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 14
作者:  
Wen, Yiming;  Xu, Peijia;  Chen, Yijie;  Meng, Jingyi;  Zheng, Mingyue
  |  收藏  |  浏览/下载:13/0  |  提交时间:2025/04/01
In vitro and In vivo Drug Metabolism Analysis of BPI-460372-A Covalent TEAD1/3/4 Inhibitor 期刊论文  OAI收割
CURRENT DRUG METABOLISM, 2025, 页码: 15
作者:  
Liu, Xiaoyun;  Zhong, Dafang;  Tang, Chongzhuang;  Xu, Xiaofeng;  Lan, Hong
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/04/24
Identifying a non-conserved site for achieving allosteric covalent inhibition of CECR2 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 16
作者:  
Tang, Cai-ling;  Li, Yuan-qing;  Du, Xi-kun;  Fang, Xiao-xia;  Guang, Yi-man
  |  收藏  |  浏览/下载:15/0  |  提交时间:2025/04/01
Design and development of a series of 4-(piperazin-1-yl)pyrimidines as irreversible menin inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 280, 页码: 20
作者:  
Luo, Menglan;  Ye, Yunfei;  Tang, Lu;  Kan, Weijuan;  Chen, Lin
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/11/26
Photocatalytic overall water splitting Z-schemes for hydrogen production with the X@CTF-0/β-Sb (X = S, Se) heterostructures 期刊论文  OAI收割
COLLOIDS AND SURFACES A-PHYSICOCHEMICAL AND ENGINEERING ASPECTS, 2024, 卷号: 703, 页码: 135437
作者:  
Sun, Qing-Guo;  Yang, Chuan-Lu;  Li, Xiaohu;  Liu, Yuliang;  Zhao, Wenkai
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/11/27
Synergistic immune augmentation enabled by covalently conjugating TLR4 and NOD2 agonists 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 278, 页码: 15
作者:  
Ding, Dong;  Gao, Runing;  Lei, Yujuan;  Liu, Jianing;  Zhou, Chengkai
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/10/21
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